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Found 11 with Last Name = 'teng' and Initial = 'k'
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50280897(CHEMBL281660 | Tetradecanoic acid (2S,3R)-2-(2-hyd...)
Affinity DataKi:  880nMAssay Description:Inhibition of [3H]-PDBU binding to Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50282658(((2R,3R)-2-Hydroxymethyl-5-oxo-tetrahydro-furan-3-...)
Affinity DataKi:  1.47E+3nMAssay Description:Inhibition of [3H]-PDBU binding to Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50280896(CHEMBL276429 | Tetradecanoic acid (2S,3R)-2-hydrox...)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition of [3H]-PDBU binding to Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50282661(CHEMBL29762 | Tetradecanoic acid (2R,3S)-2-hydroxy...)
Affinity DataKi:  3.10E+3nMAssay Description:Inhibition of [3H]-PDBU binding to Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50282657(CHEMBL29668 | [(2S,3R)-2-(2-Hydroxy-ethyl)-5-oxo-t...)
Affinity DataKi:  1.86E+4nMAssay Description:Inhibition of [3H]-PDBU binding to Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetFarnesyl pyrophosphate synthase(Homo sapiens (Human))
Academia Sinica

LigandPNGBDBM12578(2-(imidazol-1-yl)-1-hydroxyethylidene-1,1-bisphosp...)
Affinity DataIC50:  4nMAssay Description:To measure the kinetic constants by radioactive assays, 0.2 μM wild-type E. coli OPPS and the wild-type or mutant S. cerevisiae GGPPS and human ...More data for this Ligand-Target Pair
TargetIspB protein(Escherichia coli (Enterobacteria))
Academia Sinica

LigandPNGBDBM12578(2-(imidazol-1-yl)-1-hydroxyethylidene-1,1-bisphosp...)
Affinity DataIC50:  220nMAssay Description:The assays were performed by mixing either 0.2 μM E. coli OPPS, Y107A/F108A S. cerevisiae GGPPS, or Y96A/F97A human GGPPS with various concentra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIspB protein(Escherichia coli (Enterobacteria))
Academia Sinica

LigandPNGBDBM12578(2-(imidazol-1-yl)-1-hydroxyethylidene-1,1-bisphosp...)
Affinity DataIC50:  290nMAssay Description:To measure the kinetic constants by radioactive assays, 0.2 μM wild-type E. coli OPPS and the wild-type or mutant S. cerevisiae GGPPS and human ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGeranylgeranyl pyrophosphate synthase BTS1(Saccharomyces cerevisiae (Yeast))
Academia Sinica

LigandPNGBDBM12578(2-(imidazol-1-yl)-1-hydroxyethylidene-1,1-bisphosp...)
Affinity DataIC50:  660nMAssay Description:To measure the kinetic constants by radioactive assays, 0.2 μM wild-type E. coli OPPS and the wild-type or mutant S. cerevisiae GGPPS and human ...More data for this Ligand-Target Pair
TargetGeranylgeranyl pyrophosphate synthase BTS1 [Y107A,F108A](Saccharomyces cerevisiae (Yeast))
Academia Sinica

LigandPNGBDBM12578(2-(imidazol-1-yl)-1-hydroxyethylidene-1,1-bisphosp...)
Affinity DataIC50:  710nMAssay Description:The assays were performed by mixing either 0.2 μM E. coli OPPS, Y107A/F108A S. cerevisiae GGPPS, or Y96A/F97A human GGPPS with various concentra...More data for this Ligand-Target Pair
TargetGeranylgeranyl pyrophosphate synthase(Homo sapiens (Human))
Academia Sinica

LigandPNGBDBM12578(2-(imidazol-1-yl)-1-hydroxyethylidene-1,1-bisphosp...)
Affinity DataIC50: >1.00E+5nMAssay Description:To measure the kinetic constants by radioactive assays, 0.2 μM wild-type E. coli OPPS and the wild-type or mutant S. cerevisiae GGPPS and human ...More data for this Ligand-Target Pair