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Found 167 with Last Name = 'tenney' and Initial = 'k'
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM227589(Radicicol)
Affinity DataIC50:  19nMAssay Description:Inhibition of HSP90 (unknown origin)More data for this Ligand-Target Pair
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Colorado Mesa University

Curated by ChEMBL
LigandPNGBDBM50267199(CHEMBL4079583)
Affinity DataIC50:  100nMAssay Description:Inhibition of human MetAP1More data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
University Of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM22372(4-[(2R,3S)-4-(3,4-dihydroxyphenyl)-2,3-dimethylbut...)
Affinity DataIC50:  110nMAssay Description:Inhibition of human N-terminal His6-tagged 5-lipoxygenase arachidonic acid by UV-vis spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAcetolactate synthase catalytic subunit, mitochondrial(Saccharomyces cerevisiae)
University Of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50134315(7-hydroxy-11-hydroxymethyl-12-methyl-14,15-dithia-...)
Affinity DataIC50:  200nMAssay Description:Inhibition of Saccharomyces cerevisiae acetolactate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 2(Homo sapiens (Human))
Colorado Mesa University

Curated by ChEMBL
LigandPNGBDBM50267200(CHEMBL4077166)
Affinity DataIC50:  200nMAssay Description:Inhibition of human MetAP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 2(Homo sapiens (Human))
Colorado Mesa University

Curated by ChEMBL
LigandPNGBDBM50267194(CHEMBL4089242)
Affinity DataIC50:  380nMAssay Description:Inhibition of human MetAP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Colorado Mesa University

Curated by ChEMBL
LigandPNGBDBM17847(CHEMBL327579 | pyridine-2-carboxylic acid inhibito...)
Affinity DataIC50:  400nMAssay Description:Inhibition of human MetAP1More data for this Ligand-Target Pair
TargetMethionine aminopeptidase 2(Homo sapiens (Human))
Colorado Mesa University

Curated by ChEMBL
LigandPNGBDBM50295174(Bengamide A | CHEMBL256279)
Affinity DataIC50:  400nMAssay Description:Inhibition of human MetAP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 2(Homo sapiens (Human))
Colorado Mesa University

Curated by ChEMBL
LigandPNGBDBM50267193(CHEMBL4078211)
Affinity DataIC50:  400nMAssay Description:Inhibition of human MetAP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
University Of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50240936(2-[(2E,6E)-3,7-Dimethyl-9-(2,6,6-trimethyl-cyclohe...)
Affinity DataIC50:  450nMAssay Description:Inhibition of human N-terminal His6-tagged 5-lipoxygenase arachidonic acid by UV-vis spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
University Of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50320449((-)-ZILEUTON | CHEMBL1164975)
Affinity DataIC50:  500nMAssay Description:Inhibition of human N-terminal His6-tagged 5-lipoxygenase arachidonic acid by UV-vis spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
University Of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50240865((4aS,6aS,12aR,12bS)-10-Hydroxy-4,4,6a,12b-tetramet...)
Affinity DataIC50:  680nMAssay Description:Inhibition of human N-terminal His6-tagged 5-lipoxygenase arachidonic acid by UV-vis spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Colorado Mesa University

Curated by ChEMBL
LigandPNGBDBM50295174(Bengamide A | CHEMBL256279)
Affinity DataIC50:  700nMAssay Description:Inhibition of human MetAP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Colorado Mesa University

Curated by ChEMBL
LigandPNGBDBM50267193(CHEMBL4078211)
Affinity DataIC50:  700nMAssay Description:Inhibition of human MetAP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Homo sapiens (Human))
University Of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM22372(4-[(2R,3S)-4-(3,4-dihydroxyphenyl)-2,3-dimethylbut...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of human reticulocyte N-terminal His6-tagged 15-lipoxygenase by UV-vis spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Colorado Mesa University

Curated by ChEMBL
LigandPNGBDBM68281(Bengamide A)
Affinity DataIC50:  1.90E+3nMAssay Description:The determined effects of seven bengamide analogs on the enzymatic activity of both recombinated human MetAP1 and MetAP2 in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Colorado Mesa University

Curated by ChEMBL
LigandPNGBDBM68286(Bengamide N | Bengamide O)
Affinity DataIC50:  2.70E+3nMAssay Description:The determined effects of seven bengamide analogs on the enzymatic activity of both recombinated human MetAP1 and MetAP2 in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Colorado Mesa University

Curated by ChEMBL
LigandPNGBDBM50267195(CHEMBL4061080)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of human MetAP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX12(Homo sapiens (Human))
University Of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50320447(CHEMBL1164369 | isojaspic acid)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of human 12-lipoxygenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
University Of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50320451(CHEMBL1163875 | puupehedione)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of human N-terminal His6-tagged 5-lipoxygenase arachidonic acid by UV-vis spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThioredoxin reductase 1, cytoplasmic(Homo sapiens (Human))
University Of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50315537(CHEMBL1089316 | chaetocin)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of thioredoxin reductase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Homo sapiens (Human))
University Of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50320448(CHEMBL1163939 | jaspic acid)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of human reticulocyte N-terminal His6-tagged 15-lipoxygenase by UV-vis spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50232491(3,5-dibromo-2-(2',4'-dibromophenoxy)phenol | 3,5-d...)
Affinity DataIC50:  4.78E+3nMAssay Description:Inhibition of Bak binding to Mcl-1 by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Homo sapiens (Human))
University Of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50320447(CHEMBL1164369 | isojaspic acid)
Affinity DataIC50:  5.30E+3nMAssay Description:Inhibition of human 15-lipoxygenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Colorado Mesa University

Curated by ChEMBL
LigandPNGBDBM68285(Bengamide M)
Affinity DataIC50:  5.40E+3nMAssay Description:The determined effects of seven bengamide analogs on the enzymatic activity of both recombinated human MetAP1 and MetAP2 in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX12(Homo sapiens (Human))
University Of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM22372(4-[(2R,3S)-4-(3,4-dihydroxyphenyl)-2,3-dimethylbut...)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibition of human platelet N-terminal His6-tagged 12-lipoxygenase by UV-vis spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Homo sapiens (Human))
University Of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50240865((4aS,6aS,12aR,12bS)-10-Hydroxy-4,4,6a,12b-tetramet...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of human reticulocyte N-terminal His6-tagged 15-lipoxygenase by UV-vis spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Homo sapiens (Human))
University Of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50320451(CHEMBL1163875 | puupehedione)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of human reticulocyte N-terminal His6-tagged 15-lipoxygenase by UV-vis spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX12(Homo sapiens (Human))
University Of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50320448(CHEMBL1163939 | jaspic acid)
Affinity DataIC50:  7.90E+3nMAssay Description:Inhibition of human platelet N-terminal His6-tagged 12-lipoxygenase by UV-vis spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Colorado Mesa University

Curated by ChEMBL
LigandPNGBDBM50267194(CHEMBL4089242)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human MetAP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 2(Homo sapiens (Human))
Colorado Mesa University

Curated by ChEMBL
LigandPNGBDBM68281(Bengamide A)
Affinity DataIC50:  1.05E+4nMAssay Description:The determined effects of seven bengamide analogs on the enzymatic activity of both recombinated human MetAP1 and MetAP2 in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50292443(3,4,5-tribromo-2-(2', 4'-dibromo-phenoxy)phenol | ...)
Affinity DataIC50: >1.25E+4nMAssay Description:Inhibition of Bak binding to Mcl-1 by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
University Of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50320448(CHEMBL1163939 | jaspic acid)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of human N-terminal His6-tagged 5-lipoxygenase arachidonic acid by UV-vis spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50135851(2,3,4,5-tetrabromo-6-(3,5-dibromo-2-hydroxy-phenox...)
Affinity DataIC50: >1.48E+4nMAssay Description:Inhibition of Bak binding to Mcl-1 by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Homo sapiens (Human))
University Of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50320447(CHEMBL1164369 | isojaspic acid)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of human reticulocyte N-terminal His6-tagged 15-lipoxygenase by UV-vis spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50480591(CHEMBL374480)
Affinity DataIC50: >1.63E+4nMAssay Description:Inhibition of Bak binding to Mcl-1 by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50480592(CHEMBL149159)
Affinity DataIC50: >1.67E+4nMAssay Description:Inhibition of Bak binding to Mcl-1 by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50480593(CHEMBL572122)
Affinity DataIC50: >1.67E+4nMAssay Description:Inhibition of Bak binding to Mcl-1 by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50150788(2,3,5-tribromo-6-(3,5-dibromo-2-hydroxy-phenoxy)-p...)
Affinity DataIC50: >1.67E+4nMAssay Description:Inhibition of Bak binding to Mcl-1 by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50480589(CHEMBL558681)
Affinity DataIC50: >1.67E+4nMAssay Description:Inhibition of Bak binding to Mcl-1 by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50480590(CHEMBL402539)
Affinity DataIC50: >1.72E+4nMAssay Description:Inhibition of Bak binding to Mcl-1 by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM57619(2,4-dibromo-6-(2,4-dibromophenoxy)phenol | 2-[2,4-...)
Affinity DataIC50: >1.77E+4nMAssay Description:Inhibition of Bak binding to Mcl-1 by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 2(Homo sapiens (Human))
Colorado Mesa University

Curated by ChEMBL
LigandPNGBDBM68282(Bengamide B)
Affinity DataIC50:  1.79E+4nMAssay Description:The determined effects of seven bengamide analogs on the enzymatic activity of both recombinated human MetAP1 and MetAP2 in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
University Of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50320447(CHEMBL1164369 | isojaspic acid)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of human N-terminal His6-tagged 5-lipoxygenase arachidonic acid by UV-vis spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX12(Homo sapiens (Human))
University Of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50320451(CHEMBL1163875 | puupehedione)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of human platelet N-terminal His6-tagged 12-lipoxygenase by UV-vis spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Homo sapiens (Human))
University Of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50240936(2-[(2E,6E)-3,7-Dimethyl-9-(2,6,6-trimethyl-cyclohe...)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of human reticulocyte N-terminal His6-tagged 15-lipoxygenase by UV-vis spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX12(Homo sapiens (Human))
University Of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50240865((4aS,6aS,12aR,12bS)-10-Hydroxy-4,4,6a,12b-tetramet...)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of human platelet N-terminal His6-tagged 12-lipoxygenase by UV-vis spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Colorado Mesa University

Curated by ChEMBL
LigandPNGBDBM68283(Bengamide G)
Affinity DataIC50:  2.68E+4nMAssay Description:The determined effects of seven bengamide analogs on the enzymatic activity of both recombinated human MetAP1 and MetAP2 in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Colorado Mesa University

Curated by ChEMBL
LigandPNGBDBM68282(Bengamide B)
Affinity DataIC50:  2.93E+4nMAssay Description:The determined effects of seven bengamide analogs on the enzymatic activity of both recombinated human MetAP1 and MetAP2 in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX12(Homo sapiens (Human))
University Of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50320447(CHEMBL1164369 | isojaspic acid)
Affinity DataIC50:  3.10E+4nMAssay Description:Inhibition of human platelet N-terminal His6-tagged 12-lipoxygenase by UV-vis spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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