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Found 458 with Last Name = 'thomas' and Initial = 'aj'
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM285708(US10077289, Compound 16 | [(2S,3R,4R)-3-Hydroxy-4-...)
Affinity DataKi:  0.720nMpH: 7.8Assay Description:The protease-free PPIase assay measures the rate of cis to trans conversion of a peptide substrate catalyzed by the enzyme cyclophilin A. Addition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM50022815((3S,6S,9S,12R,15S,18S,21S,24S,30S,33S)-30-ethyl-33...)
Affinity DataKi:  1.5nMpH: 7.8Assay Description:The protease-free PPIase assay measures the rate of cis to trans conversion of a peptide substrate catalyzed by the enzyme cyclophilin A. Addition of...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM285706(US10077289, Compound 14 | [(2S,3R,4R)-7-(5-Fluoro-...)
Affinity DataKi:  1.5nMpH: 7.8Assay Description:The protease-free PPIase assay measures the rate of cis to trans conversion of a peptide substrate catalyzed by the enzyme cyclophilin A. Addition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM285715(US10077289, Compound 23 | [(2S,3R,4R)-3-Hydroxy-4-...)
Affinity DataKi:  2.10nMpH: 7.8Assay Description:The protease-free PPIase assay measures the rate of cis to trans conversion of a peptide substrate catalyzed by the enzyme cyclophilin A. Addition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM285710(US10077289, Compound 18 | [(2S,3R,4R)-3-Hydroxy-4-...)
Affinity DataKi:  2.20nMpH: 7.8Assay Description:The protease-free PPIase assay measures the rate of cis to trans conversion of a peptide substrate catalyzed by the enzyme cyclophilin A. Addition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM285701(US10077289, Compound 9 | [(2S,3R,4R)-1-(1H-Benzimi...)
Affinity DataKi:  2.30nMpH: 7.8Assay Description:The protease-free PPIase assay measures the rate of cis to trans conversion of a peptide substrate catalyzed by the enzyme cyclophilin A. Addition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM285707(US10077289, Compound 15 | [(2S,3R,4R)-3-Hydroxy-4-...)
Affinity DataKi:  2.5nMpH: 7.8Assay Description:The protease-free PPIase assay measures the rate of cis to trans conversion of a peptide substrate catalyzed by the enzyme cyclophilin A. Addition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM285725(US10077289, Compound 33 | [2S,3R,4R)-3-Hydroxy-4-m...)
Affinity DataKi:  3.10nMpH: 7.8Assay Description:The protease-free PPIase assay measures the rate of cis to trans conversion of a peptide substrate catalyzed by the enzyme cyclophilin A. Addition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM285726(US10077289, Compound 34 | [2S,3R,4R)-3-Hydroxy-4-m...)
Affinity DataKi:  3.10nMpH: 7.8Assay Description:The protease-free PPIase assay measures the rate of cis to trans conversion of a peptide substrate catalyzed by the enzyme cyclophilin A. Addition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM285714(US10077289, Compound 22 | [(2S,3R,4R)-3-Hydroxy-4-...)
Affinity DataKi:  3.20nMpH: 7.8Assay Description:The protease-free PPIase assay measures the rate of cis to trans conversion of a peptide substrate catalyzed by the enzyme cyclophilin A. Addition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM285713(US10077289, Compound 21 | [(2S,3R,4R)-3-Hydroxy-4-...)
Affinity DataKi:  3.20nMpH: 7.8Assay Description:The protease-free PPIase assay measures the rate of cis to trans conversion of a peptide substrate catalyzed by the enzyme cyclophilin A. Addition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM285705(US10077289, Compound 13 | [(2S,3R,4R)-3-Hydroxy-4-...)
Affinity DataKi:  3.20nMpH: 7.8Assay Description:The protease-free PPIase assay measures the rate of cis to trans conversion of a peptide substrate catalyzed by the enzyme cyclophilin A. Addition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM285716(US10077289, Compound 24 | [(2S,3R,4R)-3-Hydroxy-4-...)
Affinity DataKi:  3.5nMpH: 7.8Assay Description:The protease-free PPIase assay measures the rate of cis to trans conversion of a peptide substrate catalyzed by the enzyme cyclophilin A. Addition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM285704(US10077289, Compound 12 | [(2S,3R,4R)-3-Hydroxy-4-...)
Affinity DataKi:  3.80nMpH: 7.8Assay Description:The protease-free PPIase assay measures the rate of cis to trans conversion of a peptide substrate catalyzed by the enzyme cyclophilin A. Addition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM285717(US10077289, Compound 25 | [(2S,3R,4R)-3-Hydroxy-4-...)
Affinity DataKi:  3.80nMpH: 7.8Assay Description:The protease-free PPIase assay measures the rate of cis to trans conversion of a peptide substrate catalyzed by the enzyme cyclophilin A. Addition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM285720(US10077289, Compound 28 | [(2S,3R,4R)-3-Hydroxy-4-...)
Affinity DataKi:  3.90nMpH: 7.8Assay Description:The protease-free PPIase assay measures the rate of cis to trans conversion of a peptide substrate catalyzed by the enzyme cyclophilin A. Addition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM285709(US10077289, Compound 17 | [(2S,3R,4R)-3-Hydroxy-4-...)
Affinity DataKi:  3.90nMpH: 7.8Assay Description:The protease-free PPIase assay measures the rate of cis to trans conversion of a peptide substrate catalyzed by the enzyme cyclophilin A. Addition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM285697(US10077289, Compound 5 | [(2S,3R,4R)-3-Hydroxy-4-m...)
Affinity DataKi:  4.10nMpH: 7.8Assay Description:The protease-free PPIase assay measures the rate of cis to trans conversion of a peptide substrate catalyzed by the enzyme cyclophilin A. Addition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM285727(US10077289, Compound 35 | [2S,3R,4R)-3-Hydroxy-4-m...)
Affinity DataKi:  4.40nMpH: 7.8Assay Description:The protease-free PPIase assay measures the rate of cis to trans conversion of a peptide substrate catalyzed by the enzyme cyclophilin A. Addition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM285693(US10077289, Compound 2 | [(2S,3R,4R)-3-Hydroxy-4-m...)
Affinity DataKi:  4.60nMpH: 7.8Assay Description:The protease-free PPIase assay measures the rate of cis to trans conversion of a peptide substrate catalyzed by the enzyme cyclophilin A. Addition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM285695(US10077289, Compound 4 | [(2S,3R,4R)-5-(1-(N,N-Dim...)
Affinity DataKi:  5.10nMpH: 7.8Assay Description:The protease-free PPIase assay measures the rate of cis to trans conversion of a peptide substrate catalyzed by the enzyme cyclophilin A. Addition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM285698(US10077289, Compound 6 | [(2S,3R,4R)-3-Hydroxy-5-(...)
Affinity DataKi:  5.10nMpH: 7.8Assay Description:The protease-free PPIase assay measures the rate of cis to trans conversion of a peptide substrate catalyzed by the enzyme cyclophilin A. Addition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM285711(US10077289, Compound 19 | [(2S,3R,4R)-3-Hydroxy-4-...)
Affinity DataKi:  5.40nMpH: 7.8Assay Description:The protease-free PPIase assay measures the rate of cis to trans conversion of a peptide substrate catalyzed by the enzyme cyclophilin A. Addition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM285729(US10077289, Compound 37 | [(2S,3R,4R)-3-Hydroxy-4-...)
Affinity DataKi:  5.60nMpH: 7.8Assay Description:The protease-free PPIase assay measures the rate of cis to trans conversion of a peptide substrate catalyzed by the enzyme cyclophilin A. Addition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM285699(US10077289, Compound 7 | [(2S,3R,4R)-3-Hydroxy-4-m...)
Affinity DataKi:  5.60nMpH: 7.8Assay Description:The protease-free PPIase assay measures the rate of cis to trans conversion of a peptide substrate catalyzed by the enzyme cyclophilin A. Addition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM285703(US10077289, Compound 11 | [(2S,3R,4S)-3-Hydroxy-4-...)
Affinity DataKi:  5.60nMpH: 7.8Assay Description:The protease-free PPIase assay measures the rate of cis to trans conversion of a peptide substrate catalyzed by the enzyme cyclophilin A. Addition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM285712(US10077289, Compound 20 | [(2S,3R,4R)-3-Hydroxy-7-...)
Affinity DataKi:  5.70nMpH: 7.8Assay Description:The protease-free PPIase assay measures the rate of cis to trans conversion of a peptide substrate catalyzed by the enzyme cyclophilin A. Addition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM285719(US10077289, Compound 27 | [(2S,3R,4R)-3-Hydroxy-4-...)
Affinity DataKi:  6.80nMpH: 7.8Assay Description:The protease-free PPIase assay measures the rate of cis to trans conversion of a peptide substrate catalyzed by the enzyme cyclophilin A. Addition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM285702(US10077289, Compound 10 | [(2S,3R,4R)-1-(1H-Benzim...)
Affinity DataKi:  7.10nMpH: 7.8Assay Description:The protease-free PPIase assay measures the rate of cis to trans conversion of a peptide substrate catalyzed by the enzyme cyclophilin A. Addition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM285700(US10077289, Compound 8 | [(2S,3R,4R)-3-Hydroxy-4-m...)
Affinity DataKi:  7.40nMpH: 7.8Assay Description:The protease-free PPIase assay measures the rate of cis to trans conversion of a peptide substrate catalyzed by the enzyme cyclophilin A. Addition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM285728(US10077289, Compound 36 | [(2S,3R,4R)-3-Hydroxy-4-...)
Affinity DataKi:  7.70nMpH: 7.8Assay Description:The protease-free PPIase assay measures the rate of cis to trans conversion of a peptide substrate catalyzed by the enzyme cyclophilin A. Addition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM285724(US10077289, Compound 32 | [(2S,3R,4R)-3-Hydroxy-4-...)
Affinity DataKi:  8.30nMpH: 7.8Assay Description:The protease-free PPIase assay measures the rate of cis to trans conversion of a peptide substrate catalyzed by the enzyme cyclophilin A. Addition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM285694(US10077289, Compound 3 | [(2S,3R,4R)-3-Hydroxy-4-m...)
Affinity DataKi:  8.60nMpH: 7.8Assay Description:The protease-free PPIase assay measures the rate of cis to trans conversion of a peptide substrate catalyzed by the enzyme cyclophilin A. Addition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM285723(US10077289, Compound 31 | [(2S,3R,4R)-3-Hydroxy-4-...)
Affinity DataKi:  9.5nMpH: 7.8Assay Description:The protease-free PPIase assay measures the rate of cis to trans conversion of a peptide substrate catalyzed by the enzyme cyclophilin A. Addition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM285721(US10077289, Compound 29 | [(2S,3R,4R)-3-Hydroxy-4-...)
Affinity DataKi:  11nMpH: 7.8Assay Description:The protease-free PPIase assay measures the rate of cis to trans conversion of a peptide substrate catalyzed by the enzyme cyclophilin A. Addition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM285718(US10077289, Compound 26 | [(2S,3R,4R)-3-Hydroxy-7-...)
Affinity DataKi:  12.2nMpH: 7.8Assay Description:The protease-free PPIase assay measures the rate of cis to trans conversion of a peptide substrate catalyzed by the enzyme cyclophilin A. Addition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM285722(US10077289, Compound 30 | [(2S,3R,4R)-3-Hydroxy-4-...)
Affinity DataKi:  14nMpH: 7.8Assay Description:The protease-free PPIase assay measures the rate of cis to trans conversion of a peptide substrate catalyzed by the enzyme cyclophilin A. Addition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM285692(US10077289, Compound 1 | [(2S,3R,4R)-3-Hydroxy-4-m...)
Affinity DataKi:  15nMpH: 7.8Assay Description:The protease-free PPIase assay measures the rate of cis to trans conversion of a peptide substrate catalyzed by the enzyme cyclophilin A. Addition of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM50004665((oxotremorine)1-(4-Pyrrolidin-1-yl-but-2-ynyl)-pyr...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of 0.1 nM [3H]cis-methyldioxolane binding to rat neocortex muscarinic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50009300(CHEMBL11081 | N-Methyl-N-(4-pyrrolidin-1-yl-but-2-...)
Affinity DataIC50:  4.5nMAssay Description:Inhibition of 0.1 nM [3H]cis-methyldioxolane binding to rat neocortex muscarinic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50073501(1-Ethyl-4-phenyl-1,2,5,6-tetrahydro-pyridine-3-car...)
Affinity DataIC50:  8.80nMAssay Description:Displacement of [3H]NMS binding to human Muscarinic acetylcholine receptor M1 using membranes from transfected CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50073492(1-Ethyl-4-phenyl-1,2,5,6-tetrahydro-pyridine-3-car...)
Affinity DataIC50:  9.60nMAssay Description:Displacement of [3H]NMS binding to human Muscarinic acetylcholine receptor M1 using membranes from transfected CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50073465(1-Ethyl-4-phenyl-1,2,5,6-tetrahydro-pyridine-3-car...)
Affinity DataIC50:  12nMAssay Description:Displacement of [3H]NMS binding to human Muscarinic acetylcholine receptor M1 using membranes from transfected CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50073488(1-Ethyl-4-phenyl-1,2,3,6-tetrahydro-pyridine-3-car...)
Affinity DataIC50:  13nMAssay Description:Displacement of [3H]NMS binding to human Muscarinic acetylcholine receptor M1 using membranes from transfected CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50073454(1-Ethyl-4-phenyl-1,2,5,6-tetrahydro-pyridine-3-car...)
Affinity DataIC50:  15nMAssay Description:Displacement of [3H]NMS binding to human Muscarinic acetylcholine receptor M1 using membranes from transfected CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50073479(1-Ethyl-4-phenyl-1,2,3,6-tetrahydro-pyridine-3-car...)
Affinity DataIC50:  17nMAssay Description:Displacement of [3H]NMS binding to human Muscarinic acetylcholine receptor M1 using membranes from transfected CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50073503(1-Ethyl-4-phenyl-1,2,5,6-tetrahydro-pyridine-3-car...)
Affinity DataIC50:  18nMAssay Description:Displacement of [3H]NMS binding to human Muscarinic acetylcholine receptor M1 using membranes from transfected CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50073487(1-Ethyl-4-phenyl-1,2,5,6-tetrahydro-pyridine-3-car...)
Affinity DataIC50:  21nMAssay Description:Displacement of [3H]NMS binding to human Muscarinic acetylcholine receptor M2 using membranes from transfected CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50280524(2-Methyl-6-pyrrolidin-1-yl-hex-4-ynal oxime | CHEM...)
Affinity DataIC50:  21nMAssay Description:Inhibition of 0.1 nM [3H]cis-methyldioxolane binding to rat neocortex muscarinic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50009291(CHEMBL75358 | N-(4-Dimethylamino-but-2-ynyl)-N-met...)
Affinity DataIC50:  22nMAssay Description:Inhibition of 0.1 nM [3H]cis-methyldioxolane binding to rat neocortex muscarinic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
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