Affinity DataKi: 0.0150nMAssay Description:Displacement of [3H]-diprenorphine from human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0190nMAssay Description:Displacement of [3H]-diprenorphine from human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0200nMAssay Description:Displacement of [3H]-diprenorphine from human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0250nMAssay Description:Displacement of [3H]-diprenorphine from human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0290nMAssay Description:Displacement of [3H]-diprenorphine from rat recombinant MOR expressed in rat C6 cells after 2 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0290nMAssay Description:Displacement of [3H]-diprenorphine from rat recombinant MOR expressed in rat C6 cells after 2 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0300nMAssay Description:Displacement of [3H]-diprenorphine from rat recombinant MOR expressed in rat C6 cells after 2 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0310nMAssay Description:Displacement of [3H]-diprenorphine from rat recombinant MOR expressed in rat C6 cells after 2 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0330nMAssay Description:Displacement of [3H]-diprenorphine from human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0380nMAssay Description:Displacement of [3H]-diprenorphine from rat recombinant MOR expressed in rat C6 cells after 2 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0410nMAssay Description:Displacement of [3H]-diprenorphine from human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0430nM Kon: 0.0000145M-1s-1 Koff: 3.39E+5s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 0.0430nMAssay Description:Displacement of [3H]-diprenorphine from rat recombinant MOR expressed in rat C6 cells after 2 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0430nMAssay Description:Antagonist activity at human mu opioid receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.0470nMAssay Description:Displacement of [3H]-diprenorphine from human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0510nMAssay Description:Displacement of [3H]-diprenorphine from human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0510nMAssay Description:Displacement of [3H]-diprenorphine from human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0540nMAssay Description:Displacement of [3H]-diprenorphine from rat recombinant MOR expressed in rat C6 cells after 2 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0570nMAssay Description:Displacement of [3H]-diprenorphine from human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0590nMAssay Description:Displacement of [3H]-diprenorphine from human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0600nMAssay Description:Displacement of [3H]-diprenorphine from human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0600nMAssay Description:Binding affinity for human leukocyte elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 0.0600nMAssay Description:Displacement of [3H]-diprenorphine from rat recombinant MOR expressed in rat C6 cells after 2 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0620nMAssay Description:Displacement of [3H]-diprenorphine from human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0650nMAssay Description:Displacement of [3H]-diprenorphine from human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0670nMAssay Description:Displacement of [3H]-diprenorphine from human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0670nMAssay Description:Displacement of [3H]-diprenorphine from human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0670nMAssay Description:Displacement of [3H]-diprenorphine from human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0680nM Kon: 0.0000759M-1s-1 Koff: 1.12E+6s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 0.0690nMAssay Description:Displacement of [3H]-diprenorphine from human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0700nMAssay Description:Antagonist activity at human mu opioid receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.0700nMAssay Description:Displacement of [3H]citalopram from SERTMore data for this Ligand-Target Pair
Affinity DataKi: 0.0710nM Kon: 0.0000550M-1s-1 Koff: 7.76E+5s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 0.0740nMAssay Description:Displacement of [3H]-diprenorphine from human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0780nMAssay Description:Displacement of [3H]-diprenorphine from human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0800nMAssay Description:Antagonist activity at human mu opioid receptor by GTP-gamma S binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.0820nMAssay Description:Displacement of [3H]-diprenorphine from human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0820nMAssay Description:Displacement of [3H]-diprenorphine from human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0860nMAssay Description:Displacement of [3H]-diprenorphine from human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0860nMAssay Description:Displacement of [3H]-diprenorphine from human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0860nMAssay Description:Displacement of [3H]-diprenorphine from human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0900nMAssay Description:Displacement of [3H]-diprenorphine from human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0910nMAssay Description:Displacement of [3H]-diprenorphine from rat recombinant MOR expressed in rat C6 cells after 2 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0920nMAssay Description:Displacement of [3H]-diprenorphine from human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Displacement of [3H]-diprenorphine from human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nM Kon: 0.00000617M-1s-1 Koff: 6.46E+4s-1Assay Description:Component deacylation rate constant for interaction with human leukocyte elastaseChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 0.110nMAssay Description:Displacement of [3H]-diprenorphine from human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.110nMAssay Description:Displacement of [3H]-diprenorphine from human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.110nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair