Compile Data Set for Download or QSAR
maximum 50k data
Found 30 with Last Name = 'tian' and Initial = 'gr'
TargetCarboxypeptidase A1(Homo sapiens (Human))
Yanbian University

Curated by ChEMBL
LigandPNGBDBM50373038(CHEMBL407567)
Affinity DataKi:  150nMAssay Description:Inhibition of CPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCarboxypeptidase A1(Homo sapiens (Human))
Yanbian University

Curated by ChEMBL
LigandPNGBDBM50301283((R)-2-benzyl-5-nitro-4-oxopentanoic acid | CHEMBL5...)
Affinity DataKi:  160nMAssay Description:Inhibition of Carboxypeptidase A assessed as amount of Cl-CPL consumed by UV spectrometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase A1(Homo sapiens (Human))
Yanbian University

Curated by ChEMBL
LigandPNGBDBM50301281((+/-)-2-benzyl-5,5,5-trifluoro-4-oxopentanoic acid...)
Affinity DataKi:  200nMAssay Description:Inhibition of Carboxypeptidase A assessed as amount of Cl-CPL consumed by UV spectrometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase A1(Homo sapiens (Human))
Yanbian University

Curated by ChEMBL
LigandPNGBDBM50301282((+/-)-2-benzyl-5-nitro-4-oxopentanoic acid | CHEMB...)
Affinity DataKi:  430nMAssay Description:Inhibition of Carboxypeptidase A assessed as amount of Cl-CPL consumed by UV spectrometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase A1(Homo sapiens (Human))
Yanbian University

Curated by ChEMBL
LigandPNGBDBM50373036(CHEMBL259621)
Affinity DataKi:  450nMAssay Description:Inhibition of CPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCarboxypeptidase A1(Homo sapiens (Human))
Yanbian University

Curated by ChEMBL
LigandPNGBDBM50373037(CHEMBL261332)
Affinity DataKi:  790nMAssay Description:Inhibition of CPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase A1(Homo sapiens (Human))
Yanbian University

Curated by ChEMBL
LigandPNGBDBM50373039(CHEMBL407566)
Affinity DataKi:  2.08E+3nMAssay Description:Inhibition of CPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase A1(Homo sapiens (Human))
Yanbian University

Curated by ChEMBL
LigandPNGBDBM50301280((+/-)-2-benzyl-5-bromo-4-oxopentanoic acid | CHEMB...)
Affinity DataKi:  1.50E+4nMAssay Description:Inhibition of Carboxypeptidase A assessed as amount of Cl-CPL consumed by UV spectrometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase A1(Homo sapiens (Human))
Yanbian University

Curated by ChEMBL
LigandPNGBDBM50301284((S)-2-benzyl-5-nitro-4-oxopentanoic acid | CHEMBL5...)
Affinity DataKi:  3.10E+4nMAssay Description:Inhibition of Carboxypeptidase A assessed as amount of Cl-CPL consumed by UV spectrometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase A1(Homo sapiens (Human))
Yanbian University

Curated by ChEMBL
LigandPNGBDBM50373035(CHEMBL259221)
Affinity DataKi:  6.26E+4nMAssay Description:Inhibition of CPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase A1(Homo sapiens (Human))
Yanbian University

Curated by ChEMBL
LigandPNGBDBM50373037(CHEMBL261332)
Affinity DataKi:  6.80E+4nMAssay Description:Inhibition of CPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase A1(Homo sapiens (Human))
Yanbian University

Curated by ChEMBL
LigandPNGBDBM50301279((+/-)-2-benzyl-4-oxopentanoic acid | CHEMBL568460)
Affinity DataKi:  2.07E+5nMAssay Description:Inhibition of Carboxypeptidase A assessed as amount of Cl-CPL consumed by UV spectrometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50147178((Z)-Octadec-9-enoic acid phenylamide | CHEMBL15611...)
Affinity DataIC50:  20nMAssay Description:Inhibitory activity against rat liver microsomal Acyl coenzyme A:cholesterol acyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50147178((Z)-Octadec-9-enoic acid phenylamide | CHEMBL15611...)
Affinity DataIC50:  140nMAssay Description:Inhibitory activity against human Acyl coenzyme A:cholesterol acyltransferase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50150482(Acetic acid 3-acetoxy-4-acetoxymethyl-12-hydroxy-4...)
Affinity DataIC50:  170nMAssay Description:Inhibitory activity against rat liver microsomal Acyl coenzyme A:cholesterol acyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50147178((Z)-Octadec-9-enoic acid phenylamide | CHEMBL15611...)
Affinity DataIC50:  170nMAssay Description:Inhibitory activity against human Acyl coenzyme A:cholesterol acyltransferase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50150482(Acetic acid 3-acetoxy-4-acetoxymethyl-12-hydroxy-4...)
Affinity DataIC50:  640nMAssay Description:Inhibitory activity against human Acyl coenzyme A:cholesterol acyltransferase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50150483((9Z,12Z)-Octadeca-9,12-dienoic acid amide | CHEMBL...)
Affinity DataIC50:  4.50E+4nMAssay Description:Inhibitory activity against human Acyl coenzyme A:cholesterol acyltransferase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50150483((9Z,12Z)-Octadeca-9,12-dienoic acid amide | CHEMBL...)
Affinity DataIC50:  5.30E+4nMAssay Description:Inhibitory activity against human Acyl coenzyme A:cholesterol acyltransferase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM23028((9Z)-octadec-9-enamide | 14C-labeled oleamide | CH...)
Affinity DataIC50:  6.30E+4nMAssay Description:Inhibitory activity against human Acyl coenzyme A:cholesterol acyltransferase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM23028((9Z)-octadec-9-enamide | 14C-labeled oleamide | CH...)
Affinity DataIC50:  8.50E+4nMAssay Description:Inhibitory activity against human Acyl coenzyme A:cholesterol acyltransferase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50150483((9Z,12Z)-Octadeca-9,12-dienoic acid amide | CHEMBL...)
Affinity DataIC50:  1.50E+5nMAssay Description:Inhibitory activity against rat liver microsomal Acyl coenzyme A:cholesterol acyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM23028((9Z)-octadec-9-enamide | 14C-labeled oleamide | CH...)
Affinity DataIC50:  1.70E+5nMAssay Description:Inhibitory activity against rat liver microsomal Acyl coenzyme A:cholesterol acyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM22231((9Z,12Z)-octadeca-9,12-dienoic acid | CHEMBL267476...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity against human Acyl coenzyme A:cholesterol acyltransferase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50150484((Z)-9-octadecenoic acid | (Z)-Octadec-9-enoic acid...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity against human Acyl coenzyme A:cholesterol acyltransferase 1More data for this Ligand-Target Pair
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM22231((9Z,12Z)-octadeca-9,12-dienoic acid | CHEMBL267476...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity against human Acyl coenzyme A:cholesterol acyltransferase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50150484((Z)-9-octadecenoic acid | (Z)-Octadec-9-enoic acid...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity against human Acyl coenzyme A:cholesterol acyltransferase 2More data for this Ligand-Target Pair
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM22231((9Z,12Z)-octadeca-9,12-dienoic acid | CHEMBL267476...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity against rat liver microsomal Acyl coenzyme A:cholesterol acyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50150482(Acetic acid 3-acetoxy-4-acetoxymethyl-12-hydroxy-4...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity against human Acyl coenzyme A:cholesterol acyltransferase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50150484((Z)-9-octadecenoic acid | (Z)-Octadec-9-enoic acid...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity against rat liver microsomal Acyl coenzyme A:cholesterol acyltransferaseMore data for this Ligand-Target Pair