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Found 30 with Last Name = 'true' and Initial = 'ra'
TargetGlutamate receptor ionotropic, kainate 4(Homo sapiens (Human))
Allelix Biopharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM50002369((2S-(2alpha,3beta,4beta))-2-carboxy-4-(1-methyleth...)
Affinity DataKi:  2.29nMMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 4(Homo sapiens (Human))
Allelix Biopharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM17660((2S)-2-amino-3-(3,5-dioxo-1,2,4-oxadiazolidin-2-yl...)
Affinity DataKi:  6.43nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 4(Homo sapiens (Human))
Allelix Biopharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM50252103((2S,3S,4S)-2-CARBOXY-4-[(1Z,3E,5R)-5-CARBOXY-1-MET...)
Affinity DataKi:  10.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 4(Homo sapiens (Human))
Allelix Biopharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM50013055(2-aminopentanedioateglutamate | L-Glutamate | glut...)
Affinity DataKi:  18.3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50001266(5,7-DICHLORO-4-HYDROXYQUINOLINE-2-CARBOXYLIC ACID ...)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]glycine from glycine site on the NMDA receptor.More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM22778(6,7-Dichloro-1,4-dihydro-quinoxaline-2,3-dione | 6...)
Affinity DataKi:  210nMAssay Description:Displacement of [3H]glycine from glycine site on the NMDA receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50002707(7,8-Dichloro-5H-[1,2,4]triazolo[4,3-a]quinoxalin-4...)
Affinity DataKi:  630nMAssay Description:Displacement of [3H]glycine from glycine site on the NMDA receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50002696(7,8-Dichloro-5H-imidazo[1,2-a]quinoxalin-4-one | C...)
Affinity DataKi:  1.26E+3nMAssay Description:Displacement of [3H]glycine from glycine site on the NMDA receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50002700(1-Butyl-7,8-dichloro-5H-[1,2,4]triazolo[4,3-a]quin...)
Affinity DataKi:  1.48E+3nMAssay Description:Displacement of [3H]glycine from glycine site on the NMDA receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 4(Homo sapiens (Human))
Allelix Biopharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM50002370((R,S)-alpha-amino-3-hydroxy-5-methyl-4-isooxazole-...)
Affinity DataKi:  1.97E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50002710(7,9-Dichloro-5H-[1,2,4]triazolo[4,3-a]quinoxalin-4...)
Affinity DataKi:  2.85E+3nMAssay Description:Displacement of [3H]glycine from glycine site on the NMDA receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 4(Homo sapiens (Human))
Allelix Biopharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM50240399((2R,3R,4S)-3-(carboxymethyl)-4-isopropylpyrrolidin...)
Affinity DataKi:  3.84E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50002701(7,8-Dichloro-1-propyl-5H-[1,2,4]triazolo[4,3-a]qui...)
Affinity DataKi:  3.92E+3nMAssay Description:Displacement of [3H]glycine from glycine site on the NMDA receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50002711(7,8-Dichloro-1-ethyl-5H-[1,2,4]triazolo[4,3-a]quin...)
Affinity DataKi:  4.58E+3nMAssay Description:Displacement of [3H]glycine from glycine site on the NMDA receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50002704(7-Nitro-5H-[1,2,4]triazolo[4,3-a]quinoxalin-4-one ...)
Affinity DataKi:  7.35E+3nMAssay Description:Displacement of [3H]glycine from glycine site on the NMDA receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 4(Homo sapiens (Human))
Allelix Biopharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM82560(CAS_2379-57-9 | DNQX | NSC_3140)
Affinity DataKi:  8.49E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50002712(8-Nitro-5H-1,2,3,5,9b-pentaaza-cyclopenta[a]naphth...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]glycine from glycine site on the NMDA receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50002695(7,8-Dichloro-5H-1,2,3,5,9b-pentaaza-cyclopenta[a]n...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]glycine from glycine site on the NMDA receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50002708(7-Nitro-5H-1,2,3,5,9b-pentaaza-cyclopenta[a]naphth...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]glycine from glycine site on the NMDA receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50002709(8,9-Dichloro-6H-pyrazolo[1,5-c]quinazolin-5-one | ...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]glycine from glycine site on the NMDA receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50002705(8-Chloro-6H-pyrazolo[1,5-c]quinazolin-5-one | CHEM...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]glycine from glycine site on the NMDA receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50002706(7,8-Dichloro-1-phenyl-5H-[1,2,4]triazolo[4,3-a]qui...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]glycine from glycine site on the NMDA receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50002703(7,8-Dichloro-1-methyl-5H-[1,2,4]triazolo[4,3-a]qui...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]glycine from glycine site on the NMDA receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50002702(7,8-Dichloro-1-trifluoromethyl-5H-[1,2,4]triazolo[...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]glycine from glycine site on the NMDA receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50002699(7,8-Difluoro-5H-[1,2,4]triazolo[4,3-a]quinoxalin-4...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]glycine from glycine site on the NMDA receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 4(Homo sapiens (Human))
Allelix Biopharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM50002343(2-Methylamino-succinic acid | CHEMBL275325 | NMDA)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 4(Homo sapiens (Human))
Allelix Biopharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM50289504(7-Cyano-3-hydroxy-6-nitro-quinoxalin-2-ol anion | ...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2C(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM85211(t-2,4-PDC | t-PDC)
Affinity DataIC50: <1.00E+5nMAssay Description:Tested for the ability to displace [3H]CGS-19,755 (10 nM) binding in rat forebrain membranes for NMDA receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGlutamate receptor ionotropic, NMDA 2C(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50212606(CHEMBL176910 | LY-301900)
Affinity DataIC50: <1.00E+5nMAssay Description:Tested for the ability to displace [3H]CGS-19,755 (10 nM) binding in rat forebrain membranes for NMDA receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGlutamate receptor ionotropic, NMDA 2C(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50280814((2S,4R)-4-(1H-Tetrazol-5-yl)-pyrrolidine-2-carboxy...)
Affinity DataIC50: >1.00E+5nMAssay Description:Tested for the ability to displace [3H]-CGS-19,755 (10 nM) binding in rat forebrain membranes for NMDA receptorMore data for this Ligand-Target Pair
In DepthDetails Article