TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Ludwig-Maximilians-Universit£T M£Nchen
Curated by ChEMBL
Ludwig-Maximilians-Universit£T M£Nchen
Curated by ChEMBL
Affinity DataIC50: 1.04E+4nMAssay Description:Inhibition of human recombinant N-terminally 6X-His-tagged SIRT2 after 4 hrs in presence of NAD+ by fluorescent deacetyalse assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Ludwig-Maximilians-Universit£T M£Nchen
Curated by ChEMBL
Ludwig-Maximilians-Universit£T M£Nchen
Curated by ChEMBL
Affinity DataIC50: 1.56E+4nMAssay Description:Inhibition of human recombinant N-terminally 6X-His-tagged SIRT2 after 4 hrs in presence of NAD+ by fluorescent deacetyalse assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Homo sapiens (Human))
Ludwig-Maximilians-Universit£T M£Nchen
Curated by ChEMBL
Ludwig-Maximilians-Universit£T M£Nchen
Curated by ChEMBL
Affinity DataIC50: 2.36E+4nMAssay Description:Inhibition of human recombinant N-terminally 6X-His-tagged SIRT3 after 4 hrs in presence of NAD+ by fluorescent deacetyalse assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Homo sapiens (Human))
Ludwig-Maximilians-Universit£T M£Nchen
Curated by ChEMBL
Ludwig-Maximilians-Universit£T M£Nchen
Curated by ChEMBL
Affinity DataIC50: 2.51E+4nMAssay Description:Inhibition of human recombinant N-terminally 6X-His-tagged SIRT3 after 4 hrs in presence of NAD+ by fluorescent deacetyalse assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Ludwig-Maximilians-Universit£T M£Nchen
Curated by ChEMBL
Ludwig-Maximilians-Universit£T M£Nchen
Curated by ChEMBL
Affinity DataIC50: 2.80E+4nMAssay Description:Inhibition of human recombinant N-terminally His6-tagged SIRT2 after 4 hrs by homogeneous fluorescent deacetylase assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Ludwig-Maximilians-Universit£T M£Nchen
Curated by ChEMBL
Ludwig-Maximilians-Universit£T M£Nchen
Curated by ChEMBL
Affinity DataIC50: 2.84E+4nMAssay Description:Inhibition of human recombinant N-terminally 6X-His-tagged SIRT2 after 4 hrs in presence of NAD+ by fluorescent deacetyalse assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Ludwig-Maximilians-Universit£T M£Nchen
Curated by ChEMBL
Ludwig-Maximilians-Universit£T M£Nchen
Curated by ChEMBL
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibition of human recombinant N-terminally His6-tagged SIRT2 after 4 hrs by homogeneous fluorescent deacetylase assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
University Of East Anglia
Curated by ChEMBL
University Of East Anglia
Curated by ChEMBL
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of human recombinant GST-tagged SIRT1 after 4 hrs by homogeneous fluorescent deacetylase assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Ludwig-Maximilians-Universit£T M£Nchen
Curated by ChEMBL
Ludwig-Maximilians-Universit£T M£Nchen
Curated by ChEMBL
Affinity DataIC50: 3.34E+4nMAssay Description:Inhibition of human recombinant N-terminally 6X-His-tagged SIRT2 after 4 hrs in presence of NAD+ by fluorescent deacetyalse assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Ludwig-Maximilians-Universit£T M£Nchen
Curated by ChEMBL
Ludwig-Maximilians-Universit£T M£Nchen
Curated by ChEMBL
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of human recombinant N-terminally His6-tagged SIRT2 after 4 hrs by homogeneous fluorescent deacetylase assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
University Of East Anglia
Curated by ChEMBL
University Of East Anglia
Curated by ChEMBL
Affinity DataIC50: 4.06E+4nMAssay Description:Inhibition of human recombinant N-terminally GST-tagged SIRT1 after 4 hrs in presence of NAD+ by fluorescent deacetyalse assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
University Of East Anglia
Curated by ChEMBL
University Of East Anglia
Curated by ChEMBL
Affinity DataIC50: 4.16E+4nMAssay Description:Inhibition of human recombinant N-terminally GST-tagged SIRT1 after 4 hrs in presence of NAD+ by fluorescent deacetyalse assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Ludwig-Maximilians-Universit£T M£Nchen
Curated by ChEMBL
Ludwig-Maximilians-Universit£T M£Nchen
Curated by ChEMBL
Affinity DataIC50: 4.30E+4nMAssay Description:Inhibition of human recombinant N-terminally His6-tagged SIRT2 after 4 hrs by homogeneous fluorescent deacetylase assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Ludwig-Maximilians-Universit£T M£Nchen
Curated by ChEMBL
Ludwig-Maximilians-Universit£T M£Nchen
Curated by ChEMBL
Affinity DataIC50: 5.20E+4nMAssay Description:Inhibition of human recombinant N-terminally His6-tagged SIRT2 after 4 hrs by homogeneous fluorescent deacetylase assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Ludwig-Maximilians-Universit£T M£Nchen
Curated by ChEMBL
Ludwig-Maximilians-Universit£T M£Nchen
Curated by ChEMBL
Affinity DataIC50: 8.72E+4nMAssay Description:Inhibition of human recombinant N-terminally 6X-His-tagged SIRT2 after 4 hrs in presence of NAD+ by fluorescent deacetyalse assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Ludwig-Maximilians-Universit£T M£Nchen
Curated by ChEMBL
Ludwig-Maximilians-Universit£T M£Nchen
Curated by ChEMBL
Affinity DataIC50: 1.23E+5nMAssay Description:Inhibition of human recombinant N-terminally 6X-His-tagged SIRT2 after 4 hrs in presence of NAD+ by fluorescent deacetyalse assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Ludwig-Maximilians-Universit£T M£Nchen
Curated by ChEMBL
Ludwig-Maximilians-Universit£T M£Nchen
Curated by ChEMBL
Affinity DataIC50: 1.23E+5nMAssay Description:Inhibition of human recombinant N-terminally His6-tagged SIRT2 after 4 hrs by homogeneous fluorescent deacetylase assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Ludwig-Maximilians-Universit£T M£Nchen
Curated by ChEMBL
Ludwig-Maximilians-Universit£T M£Nchen
Curated by ChEMBL
Affinity DataIC50: 1.35E+5nMAssay Description:Inhibition of human recombinant N-terminally 6X-His-tagged SIRT2 after 4 hrs in presence of NAD+ by fluorescent deacetyalse assayMore data for this Ligand-Target Pair
Affinity DataKd: 1.12E+4nMAssay Description:Binding affinity at human recombinant ARTD8 expressed in Escherichia coli BL21 (DE3) R3 pRARE cells by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 7.60E+3nMAssay Description:Binding affinity at human recombinant ARTD8 expressed in Escherichia coli BL21 (DE3) R3 pRARE cells by isothermal titration calorimetryMore data for this Ligand-Target Pair