BindingDB PrimarySearch

Found 1501 with Last Name = 'uno' and Initial = 'h'

Alpha-1D adrenergic receptor(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50060964((R)-5-(2-((2-(2-ethoxyphenoxy)ethyl)amino)propyl)-...)

Ki: 0.180nMAssay Description:Displacement of [125I] HEAT from human alpha1D adrenergic receptor expressed in Chlorocebus aethiops COS1 cell membranes incubated for 60 mins by liq...More data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532486(CHEMBL4564992)

Ki: 0.300nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532486(CHEMBL4564992)

Ki: 0.300nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

PDB
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Neuronal acetylcholine receptor subunit alpha-2/beta-2(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL

BDBM50210335(CHEMBL3898434)

Ki: 0.300nMAssay Description:Displacement of [3H]epibatidine from rat alpha2beta2 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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Neuronal acetylcholine receptor subunit alpha-2/beta-2(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL

BDBM50210334(CHEMBL3948977)

Ki: 0.300nMAssay Description:Displacement of [3H]epibatidine from rat alpha2beta2 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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Alpha-1D adrenergic receptor(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50456840(CHEMBL4207824)

Ki: 0.300nMAssay Description:Displacement of 7-methoxy-[3H]-prazosin from human alpha1D-adrenoreceptor expressed in CHOK1 cell membranes after 60 mins by TopCount liquid scintill...More data for this Ligand-Target Pair

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Neuronal acetylcholine receptor subunit alpha-2/beta-2(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL

BDBM50216347((1R,4R)-2-(3-pyridinyl)-2,5-diazabicyclo[2.2.1]hep...)

Ki: 0.300nMAssay Description:Displacement of [3H]epibatidine from rat alpha2beta2 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532518(CHEMBL4440420)

Ki: 0.5nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532506(CHEMBL4536431)

Ki: 0.5nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532506(CHEMBL4536431)

Ki: 0.5nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532508(CHEMBL4471576)

Ki: 0.5nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Neuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL

BDBM50210335(CHEMBL3898434)

Ki: 0.5nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532518(CHEMBL4440420)

Ki: 0.5nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532508(CHEMBL4471576)

Ki: 0.5nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sphingosine 1-phosphate receptor 5(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL

BDBM50250631(CHEMBL4093489)

Ki: 0.574nMAssay Description:Displacement of [33P]-S1P from human S1P5 receptor expressed in CHO-K1 cells after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair

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Sphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Ono Pharmaceutical

Curated by ChEMBL

BDBM50250631(CHEMBL4093489)

Ki: 0.626nMAssay Description:Agonist activity at human S1P5 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 30 mins by E...More data for this Ligand-Target Pair

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Alpha-1D adrenergic receptor(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50164686(CHEMBL3798124)

Ki: 0.660nMAssay Description:Displacement of 7-methoxy-[3H]-prazosin from human alpha1D adrenergic receptor expressed in CHO-K1 cell membranes incubated for 60 mins by liquid sci...More data for this Ligand-Target Pair

Reactome pathway KEGG
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Neuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL

BDBM50210334(CHEMBL3948977)

Ki: 0.700nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532502(CHEMBL4538923)

Ki: 0.700nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532502(CHEMBL4538923)

Ki: 0.700nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sphingosine 1-phosphate receptor 1(Rattus norvegicus)
Ono Pharmaceutical

Curated by ChEMBL

BDBM50250631(CHEMBL4093489)

Ki: 0.772nMAssay Description:Displacement of [33P]-S1P from human S1P2 receptor expressed in CHO-K1 cells after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532512(CHEMBL4539105)

Ki: 0.800nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532512(CHEMBL4539105)

Ki: 0.800nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Neuronal acetylcholine receptor subunit alpha-2/beta-2(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL

BDBM50210337(CHEMBL3970672)

Ki: 0.800nMAssay Description:Displacement of [3H]epibatidine from rat alpha2beta2 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
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Neuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL

BDBM50210337(CHEMBL3970672)

Ki: 0.800nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Alpha-1D adrenergic receptor(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50456841(CHEMBL4218307)

Ki: 0.850nMAssay Description:Displacement of 7-methoxy-[3H]-prazosin from human alpha1D-adrenoreceptor expressed in CHOK1 cell membranes after 60 mins by TopCount liquid scintill...More data for this Ligand-Target Pair

Reactome pathway KEGG
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Alpha-1D adrenergic receptor(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50164745(CHEMBL3800606)

Ki: 0.860nMAssay Description:Displacement of 7-methoxy-[3H]-prazosin from human alpha1D adrenergic receptor expressed in CHO-K1 cell membranes incubated for 60 mins by liquid sci...More data for this Ligand-Target Pair

Reactome pathway KEGG
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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532507(CHEMBL4593797)

Ki: 0.900nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

PDB
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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532507(CHEMBL4593797)

Ki: 0.900nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
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Neuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL

BDBM50216347((1R,4R)-2-(3-pyridinyl)-2,5-diazabicyclo[2.2.1]hep...)

Ki: 1nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Alpha-1D adrenergic receptor(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50164769(CHEMBL3799553)

Ki: 1.10nMAssay Description:Displacement of 7-methoxy-[3H]-prazosin from human alpha1D adrenergic receptor expressed in CHO-K1 cell membranes incubated for 60 mins by liquid sci...More data for this Ligand-Target Pair

Reactome pathway KEGG
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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532489(CHEMBL4434692)

Ki: 1.10nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
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Neuronal acetylcholine receptor subunit alpha-2/beta-2(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL

BDBM50088438(1-(pyridin-3-yl)-1,4-diazepane | 1-Pyridin-3-yl-[1...)

Ki: 1.10nMAssay Description:Displacement of [3H]epibatidine from rat alpha2beta2 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532489(CHEMBL4434692)

Ki: 1.10nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
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Alpha-1D adrenergic receptor(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50456848(CHEMBL4208816)

Ki: 1.10nMAssay Description:Displacement of 7-methoxy-[3H]-prazosin from human alpha1D-adrenoreceptor expressed in CHOK1 cell membranes after 60 mins by TopCount liquid scintill...More data for this Ligand-Target Pair

Reactome pathway KEGG
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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532503(CHEMBL4458060)

Ki: 1.40nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532521(CHEMBL4524740)

Ki: 1.40nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532503(CHEMBL4458060)

Ki: 1.40nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

PDB
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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532521(CHEMBL4524740)

Ki: 1.40nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

PDB
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Alpha-1D adrenergic receptor(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50456851(CHEMBL4213029)

Ki: 1.5nMAssay Description:Displacement of 7-methoxy-[3H]-prazosin from human alpha1D-adrenoreceptor expressed in CHOK1 cell membranes after 60 mins by TopCount liquid scintill...More data for this Ligand-Target Pair

Reactome pathway KEGG
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Alpha-1D adrenergic receptor(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50164687(CHEMBL3799292)

Ki: 1.60nMAssay Description:Displacement of 7-methoxy-[3H]-prazosin from human alpha1D adrenergic receptor expressed in CHO-K1 cell membranes incubated for 60 mins by liquid sci...More data for this Ligand-Target Pair

Reactome pathway KEGG
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Coagulation factor X(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL

BDBM50273137((3-{[(3-Carbamimidoyl-phenyl)-({4-[1-(1-imino-ethy...)

Ki: 1.73nMAssay Description:Inhibition of human factor 10a by Dixon-plot methodMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532505(CHEMBL4535404)

Ki: 1.80nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532505(CHEMBL4535404)

Ki: 1.80nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL

BDBM50400743(CHEMBL2203549)

Ki: 2.10nMAssay Description:Binding affinity to sigma 1 receptorMore data for this Ligand-Target Pair

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Sodium-dependent noradrenaline transporter(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL

BDBM35229(3-(10,11-dihydro-5H-dibenzo[b,f]azepin-5-yl)-N-met...)

Ki: 2.5nMAssay Description:Displacement of [3H]nisoxetine from human NET expressed in HEK293 cells measured after 30 minsMore data for this Ligand-Target Pair

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Sodium-dependent noradrenaline transporter(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL

BDBM35229(3-(10,11-dihydro-5H-dibenzo[b,f]azepin-5-yl)-N-met...)

Ki: 2.5nMAssay Description:Displacement of [3H]nisoxetine from human NET expressed in HEK293 cells measured after 30 minsMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532516(CHEMBL4460187)

Ki: 2.60nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532516(CHEMBL4460187)

Ki: 2.60nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
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Alpha-1D adrenergic receptor(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL

BDBM50164739(CHEMBL3800305)

Ki: 2.60nMAssay Description:Displacement of 7-methoxy-[3H]-prazosin from human alpha1D adrenergic receptor expressed in CHO-K1 cell membranes incubated for 60 mins by liquid sci...More data for this Ligand-Target Pair

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Displayed 1 to 50 (of 1501 total ) | Next | Last >>

Filter my 1501 hits

Targets 73▿
- Collagenase 3 127
- Sigma non-opioid intracellular receptor 1 105
- Sigma intracellular receptor 2 94
- Sphingosine 1-phosphate receptor 1 66
- Sphingosine 1-phosphate receptor 3 61
- Alpha-1D adrenergic receptor 55
- Alpha-ketoglutarate-dependent dioxygenase alkB homolog 3 49
- C-C chemokine receptor type 6 48
- Cannabinoid receptor 2 46
- 5-hydroxytryptamine receptor 2C 42
- Neuronal acetylcholine receptor subunit alpha-4/beta-2 39
- Neutrophil collagenase 38
- 72 kDa type IV collagenase 38
- Stromelysin-2 38
- Progesterone receptor 37
- Fibroblast growth factor receptor 2 36
- Vitamin D3 receptor 33
- 5-hydroxytryptamine receptor 2B 31
- Glycogen synthase kinase-3 beta 31
- Lysine-specific histone demethylase 1A 30
- Coagulation factor X 21
- Matrix metalloproteinase-9 20
- Matrix metalloproteinase-14 20
- Stromelysin-1 20
- Interstitial collagenase 20
- Epidermal growth factor receptor 20
- Matrilysin 20
- Disintegrin and metalloproteinase domain-containing protein 17 19
- 5-hydroxytryptamine receptor 2A 17
- Vascular endothelial growth factor receptor 2 16
- STE20/SPS1-related proline-alanine-rich protein kinase 16
- Sodium-dependent noradrenaline transporter 14
- Sodium-dependent dopamine transporter 14
- Acetylcholine receptor subunit alpha/beta/delta/gamma 14
- Cannabinoid receptor 1 13
- Alpha-1B adrenergic receptor 13
- Alpha-1A adrenergic receptor 13
- Sodium-dependent serotonin transporter 12
- Lysine-specific histone demethylase 2 11
- Neuronal acetylcholine receptor subunit alpha-3/beta-2 11
- Neuronal acetylcholine receptor subunit alpha-2/beta-2 11
- Neuronal acetylcholine receptor subunit alpha-4/beta-4 11
- P2X purinoceptor 7 10
- Amine oxidase [flavin-containing] B 10
- Amine oxidase [flavin-containing] A 10
- Macrophage metalloelastase 8
- Neuronal acetylcholine receptor subunit alpha-3/beta-4 7
- Neuronal acetylcholine receptor subunit alpha-2/beta-4 7
- C-C chemokine receptor type 1 6
- Prothrombin 6
- C-C chemokine receptor type 7 6
- Sphingosine 1-phosphate receptor 5 5
- Polyunsaturated fatty acid 5-lipoxygenase 3
- Potassium voltage-gated channel subfamily H member 2 3
- Sphingosine 1-phosphate receptor 2 3
- Neuronal acetylcholine receptor; alpha2/beta4 2
- Glucocorticoid receptor 2
- Androgen receptor 2
- Fibroblast growth factor receptor 4 2
- 5-hydroxytryptamine receptor 1A 2
- 5-hydroxytryptamine receptor 6 2
- Fibroblast growth factor receptor 1 2
- Alpha-2A adrenergic receptor 2
- Fibroblast growth factor receptor 3 2
- Sphingosine 1-phosphate receptor 4 1
- Alpha-2C adrenergic receptor 1
- D(3) dopamine receptor 1
- Alpha-2B adrenergic receptor 1
- Histamine H1 receptor 1
- 5-hydroxytryptamine receptor 7 1
- Acetylcholinesterase 1
- Beta-2 adrenergic receptor 1
- Histamine H2 receptor 1
- ...
Publications 30▿
- J Med Chem 59: 6329-43 (2016) 224
- Bioorg Med Chem 24: 6149-6165 (2016) 152
- J Med Chem 58: 1992-2002 (2015) 96
- Eur J Med Chem 124: 689-697 (2016) 88
- J Med Chem 60: 608-626 (2017) 86
- Bioorg Med Chem 22: 5487-505 (2014) 66
- J Med Chem 57: 8886-902 (2014) 64
- Eur J Med Chem 141: 101-112 (2017) 61
- Bioorg Med Chem Lett 28: 3067-3072 (2018) 60
- J Med Chem 60: 9508-9530 (2017) 58
- J Med Chem 60: 7067-7083 (2017) 55
- Bioorg Med Chem Lett 24: 1071-4 (2014) 49
- Eur J Med Chem 139: 114-127 (2017) 44
- J Med Chem 54: 7055-65 (2011) 41
- J Med Chem 59: 2989-3002 (2016) 38
- ACS Med Chem Lett 3: 1054-1058 (2012) 38
- J Med Chem 56: 5115-29 (2013) 31
- Bioorg Med Chem Lett 21: 3885-9 (2011) 28
- Bioorg Med Chem Lett 18: 4682-7 (2008) 27
- Bioorg Med Chem Lett 22: 144-8 (2011) 26
- Bioorg Med Chem Lett 21: 1390-3 (2011) 24
- Bioorg Med Chem 25: 3845-3852 (2017) 16
- Bioorg Med Chem 16: 6949-64 (2008) 16
- J Med Chem 64: 516-526 (2021) 12
- Bioorg Med Chem 17: 4861-5 (2009) 10
- Bioorg Med Chem 15: 1475-82 (2007) 4
- RSC Med Chem 12: 1910-1925 (2021) 4
- J Med Chem 32: 583-93 (1989) 3
- Bioorg Med Chem Lett 23: 1544-7 (2013) 1
- Bioorg Med Chem 27: 3674-3681 (2019) 1
Institutions 14▿
- Takeda Pharmaceutical 424
- East China Normal University 340
- University Of Illinois At Chicago 216
- Ono Pharmaceutical 136
- Pharmaceutical 86
- Ochanomizu University 53
- Hyogo University Of Health Science 49
- TBA 38
- Kissei Pharmaceutical 27
- Tokyo Medical And Dental University 21
- Tokyo Medical And Dental University (Tmdu) 16
- University Of Sydney 10
- Curtin University 4
- Dainippon Pharmaceutical 3
Affinity: 0.0021 to 2.0E+6 nM▿
- Ki 432
- IC50 745
- EC50 324
- Affinity ≤ nM
Xtal structures: 15
Docked structures: 0
Catalog Cmpds: 56