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Found 222 with Last Name = 'upton' and Initial = 'a'
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50537192(CHEMBL4563167)
Affinity DataIC50:  240nMAssay Description:Inhibition of human ERG by manual patch clamp electrophysiology assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50537183(CHEMBL4575859)
Affinity DataIC50:  300nMAssay Description:Inhibition of human ERG by manual patch clamp electrophysiology assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50460275(CHEMBL4228918)
Affinity DataIC50:  300nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50063995(Bedaquiline | CHEBI:72292 | TMC207)
Affinity DataIC50:  370nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50063995(Bedaquiline | CHEBI:72292 | TMC207)
Affinity DataIC50:  370nMAssay Description:Inhibition of human ERG assessed as prolongation of QT intervalMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50460282(CHEMBL4226478)
Affinity DataIC50:  400nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50537180(CHEMBL4535649)
Affinity DataIC50:  450nMAssay Description:Inhibition of human ERG by manual patch clamp electrophysiology assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50452142(CHEMBL4212501)
Affinity DataIC50:  460nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50460274(CHEMBL4225434)
Affinity DataIC50:  500nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50452135(CHEMBL4213428)
Affinity DataIC50:  530nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50460276(CHEMBL4226743)
Affinity DataIC50:  600nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50460280(CHEMBL4229114)
Affinity DataIC50:  600nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50460279(CHEMBL4224771)
Affinity DataIC50:  800nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50460283(CHEMBL4226688)
Affinity DataIC50:  800nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50452136(CHEMBL4206467)
Affinity DataIC50:  880nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50452140(CHEMBL4204414)
Affinity DataIC50:  890nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50460288(CHEMBL4227540)
Affinity DataIC50:  900nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50460281(CHEMBL4228130)
Affinity DataIC50:  900nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50460295(CHEMBL4227762)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Sanofi R & D

Curated by ChEMBL
LigandPNGBDBM50192998(CHEMBL3933716)
Affinity DataIC50: <1.00E+3nMAssay Description:Inhibition of CYP3A4 in human liver microsomes assessed as 1'-hydroxymidazolam metabolite formation using midazolam as substrate incubated for 10 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50460286(CHEMBL4228555)
Affinity DataIC50: <1.00E+3nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Sanofi R & D

Curated by ChEMBL
LigandPNGBDBM50192920(CHEMBL3975000)
Affinity DataIC50: <1.00E+3nMAssay Description:Inhibition of CYP3A4 in human liver microsomes assessed as 1'-hydroxymidazolam metabolite formation using midazolam as substrate incubated for 10 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50460300(CHEMBL4225899)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Sanofi R & D

Curated by ChEMBL
LigandPNGBDBM50192916(CHEMBL3941754)
Affinity DataIC50: <1.00E+3nMAssay Description:Inhibition of CYP3A4 in human liver microsomes assessed as 1'-hydroxymidazolam metabolite formation using midazolam as substrate incubated for 10 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50460291(CHEMBL4227161)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Sanofi R & D

Curated by ChEMBL
LigandPNGBDBM50193008(CHEMBL3976702)
Affinity DataIC50: <1.00E+3nMAssay Description:Inhibition of CYP3A4 in human liver microsomes assessed as 1'-hydroxymidazolam metabolite formation using midazolam as substrate incubated for 10 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50460289(CHEMBL4225217)
Affinity DataIC50: <1.00E+3nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50460293(CHEMBL4225886)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50537194(CHEMBL4528706)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of human ERG by manual patch clamp electrophysiology assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50460299(CHEMBL4228122)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50539082(CHEMBL4638334)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50063995(Bedaquiline | CHEBI:72292 | TMC207)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50537226(CHEMBL4543900)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50063995(Bedaquiline | CHEBI:72292 | TMC207)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50063995(Bedaquiline | CHEBI:72292 | TMC207)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50279196(CHEMBL4162672)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50063995(Bedaquiline | CHEBI:72292 | TMC207)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50063995(Bedaquiline | CHEBI:72292 | TMC207)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of human ERG by manual patch clamp electrophysiology assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50537222(CHEMBL4574425)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50537181(CHEMBL4522192)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of human ERG by manual patch clamp electrophysiology assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50279217(CHEMBL4177019)
Affinity DataIC50:  1.70E+3nMAssay Description:Effective concentration on alkaline phosphatase activity in human T47D breast carcinoma cell line.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50539065(CHEMBL4646329)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50452143(CHEMBL4218132)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50460296(CHEMBL4227994)
Affinity DataIC50: >2.00E+3nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50537215(CHEMBL4593713)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50279222(CHEMBL4176516)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50537217(CHEMBL4519972)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50537241(CHEMBL4570895)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50537231(CHEMBL4578975)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50537185(CHEMBL4483435)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of human ERG by manual patch clamp electrophysiology assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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