Affinity DataKi: 0.148nMAssay Description:Compounds can be screened for their ability to inhibit ATR kinase using a radioactive-phosphate incorporation assay. Assays are carried out in a mixt...More data for this Ligand-Target Pair
Affinity DataKi: 0.148nMAssay Description:Compounds can be screened for their ability to inhibit ATR kinase using a radioactive-phosphate incorporation assay. Assays are carried out in a mixt...More data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Compounds can be screened for their ability to inhibit ATR kinase using a radioactive-phosphate incorporation assay. Assays are carried out in a mixt...More data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Compounds can be screened for their ability to inhibit ATR kinase using a radioactive-phosphate incorporation assay. Assays are carried out in a mixt...More data for this Ligand-Target Pair
Affinity DataKi: <1nMAssay Description:Compounds can be screened for their ability to inhibit ATR kinase using a radioactive-phosphate incorporation assay. Assays are carried out in a mixt...More data for this Ligand-Target Pair
Affinity DataKi: <1nMAssay Description:Compounds can be screened for their ability to inhibit ATR kinase using a radioactive-phosphate incorporation assay. Assays are carried out in a mixt...More data for this Ligand-Target Pair
Affinity DataKi: <1nMAssay Description:Compounds can be screened for their ability to inhibit ATR kinase using a radioactive-phosphate incorporation assay. Assays are carried out in a mixt...More data for this Ligand-Target Pair
Affinity DataKi: <1nMAssay Description:Compounds can be screened for their ability to inhibit ATR kinase using a radioactive-phosphate incorporation assay. Assays are carried out in a mixt...More data for this Ligand-Target Pair
Affinity DataKi: 62nMAssay Description:Inhibition of Trypanosoma cruzi squalene synthaseMore data for this Ligand-Target Pair
TargetPhosphotransferase(Trypanosoma cruzi)
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Affinity DataKi: 400nMAssay Description:Inhibition of Trypanosoma cruzi hexokinase in presence of D-glucose, 1 mM ATP and 3 mM MgCl2 by competitive inhibition assayMore data for this Ligand-Target Pair
TargetPhosphotransferase(Trypanosoma cruzi)
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Affinity DataKi: 500nMAssay Description:Inhibition of Trypanosoma cruzi hexokinase in presence of D-glucose, 1 mM ATP and 3 mM MgCl2 by competitive inhibition assayMore data for this Ligand-Target Pair
TargetPhosphotransferase(Trypanosoma cruzi)
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Affinity DataKi: 600nMAssay Description:Inhibition of Trypanosoma cruzi hexokinase in presence of ATP, 2 mM D-glucose and 3 mM MgCl2 by competitive inhibition assayMore data for this Ligand-Target Pair
TargetPhosphotransferase(Trypanosoma cruzi)
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Affinity DataKi: 1.20E+3nMAssay Description:Inhibition of glycosomal Trypanosoma cruzi hexokinase in presence of ATP, 2 mM D-glucose and 3 mM MgCl2 by competitive inhibition assayMore data for this Ligand-Target Pair
TargetPhosphotransferase(Trypanosoma cruzi)
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Affinity DataKi: 1.20E+3nMAssay Description:Inhibition of Trypanosoma cruzi hexokinase in presence of ATP, 2 mM D-glucose and 3 mM MgCl2More data for this Ligand-Target Pair
TargetPhosphotransferase(Trypanosoma cruzi)
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Affinity DataKi: 1.70E+3nMAssay Description:Inhibition of glycosomal Trypanosoma cruzi hexokinase in presence of ATP, 2 mM D-glucose and 3 mM MgCl2More data for this Ligand-Target Pair
TargetPhosphotransferase(Trypanosoma cruzi)
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Affinity DataKi: 1.70E+3nMAssay Description:Inhibition of Trypanosoma cruzi hexokinase in presence of ATP, 2 mM D-glucose and 3 mM MgCl2 by competitive inhibition assayMore data for this Ligand-Target Pair
TargetPhosphotransferase(Trypanosoma cruzi)
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Affinity DataKi: 2.40E+3nMAssay Description:Inhibition of glycosomal Trypanosoma cruzi hexokinase in presence of D-glucose, 1 mM ATP and 3 mM MgCl2 by competitive inhibition assayMore data for this Ligand-Target Pair
TargetPhosphotransferase(Trypanosoma cruzi)
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Affinity DataKi: 2.60E+3nMAssay Description:Inhibition of glycosomal Trypanosoma cruzi hexokinase in presence of ATP, 2 mM D-glucose and 3 mM MgCl2 by competitive inhibition assayMore data for this Ligand-Target Pair
TargetPhosphotransferase(Trypanosoma cruzi)
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Affinity DataKi: 2.80E+3nMAssay Description:Inhibition of Trypanosoma cruzi hexokinase in presence of ATP, 2 mM D-glucose and 3 mM MgCl2More data for this Ligand-Target Pair
TargetPhosphotransferase(Trypanosoma cruzi)
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Affinity DataKi: 2.80E+3nMAssay Description:Inhibition of Trypanosoma cruzi hexokinase in presence of ATP, 2 mM D-glucose and 3 mM MgCl2 by competitive inhibition assayMore data for this Ligand-Target Pair
TargetPhosphotransferase(Trypanosoma cruzi)
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Affinity DataKi: 2.90E+3nMAssay Description:Inhibition of glycosomal Trypanosoma cruzi hexokinase in presence of D-glucose, 1 mM ATP and 3 mM MgCl2 by competitive inhibition assayMore data for this Ligand-Target Pair
TargetPhosphotransferase(Trypanosoma cruzi)
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Affinity DataKi: 3.30E+3nMAssay Description:Inhibition of Trypanosoma cruzi hexokinase in presence of D-glucose, 1 mM ATP and 3 mM MgCl2 by competitive inhibition assayMore data for this Ligand-Target Pair
TargetPhosphotransferase(Trypanosoma cruzi)
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Affinity DataKi: 3.40E+3nMAssay Description:Inhibition of glycosomal Trypanosoma cruzi hexokinase in presence of D-glucose, 1 mM ATP and 3 mM MgCl2 by competitive inhibition assayMore data for this Ligand-Target Pair
TargetPhosphotransferase(Trypanosoma cruzi)
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Affinity DataKi: 4.30E+3nMAssay Description:Inhibition of Trypanosoma cruzi hexokinase in presence of ATP, 2 mM D-glucose and 3 mM MgCl2More data for this Ligand-Target Pair
TargetPhosphotransferase(Trypanosoma cruzi)
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Affinity DataKi: 4.30E+3nMAssay Description:Inhibition of glycosomal Trypanosoma cruzi hexokinase in presence of D-glucose, 1 mM ATP and 3 mM MgCl2More data for this Ligand-Target Pair
TargetPhosphotransferase(Trypanosoma cruzi)
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Affinity DataKi: 6.00E+3nMAssay Description:Inhibition of Trypanosoma cruzi hexokinase in presence of D-glucose, 1 mM ATP and 3 mM MgCl2More data for this Ligand-Target Pair
TargetPhosphotransferase(Trypanosoma cruzi)
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Affinity DataKi: 1.05E+4nMAssay Description:Inhibition of glycosomal Trypanosoma cruzi hexokinase in presence of ATP, 2 mM D-glucose and 3 mM MgCl2More data for this Ligand-Target Pair
TargetPhosphotransferase(Trypanosoma cruzi)
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Affinity DataKi: 1.06E+4nMAssay Description:Inhibition of glycosomal Trypanosoma cruzi hexokinase in presence of D-glucose, 1 mM ATP and 3 mM MgCl2More data for this Ligand-Target Pair
TargetPhosphotransferase(Trypanosoma cruzi)
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Affinity DataKi: 1.14E+4nMAssay Description:Inhibition of glycosomal Trypanosoma cruzi hexokinase in presence of ATP, 2 mM D-glucose and 3 mM MgCl2 by competitive inhibition assayMore data for this Ligand-Target Pair
TargetPhosphotransferase(Trypanosoma cruzi)
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Affinity DataKi: 4.39E+4nMAssay Description:Inhibition of glycosomal Trypanosoma cruzi hexokinase in presence of D-glucose, 1 mM ATP and 3 mM MgCl2More data for this Ligand-Target Pair
TargetSqualene synthase(Homo sapiens (Human))
Instituto De Parasitolog£A Y Biomedicina&Quot;L£Pez-Neyra
Curated by ChEMBL
Instituto De Parasitolog£A Y Biomedicina&Quot;L£Pez-Neyra
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Inhibition of human recombinant squalene synthaseMore data for this Ligand-Target Pair
TargetSqualene synthase(Homo sapiens (Human))
Instituto De Parasitolog£A Y Biomedicina&Quot;L£Pez-Neyra
Curated by ChEMBL
Instituto De Parasitolog£A Y Biomedicina&Quot;L£Pez-Neyra
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of human recombinant squalene synthaseMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of Leishmania major recombinant squalene synthase expressed in Escherichia coli by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of Leishmania major recombinant squalene synthase expressed in Escherichia coli by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Inhibition of Leishmania major recombinant squalene synthase expressed in Escherichia coli by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of Leishmania major recombinant squalene synthase expressed in Escherichia coli by liquid scintillation counterMore data for this Ligand-Target Pair
TargetPolyprenyl synthetase family protein(Plasmodium falciparum (isolate 3D7))
University Of Illinois At Urbana-Champaign
Curated by ChEMBL
University Of Illinois At Urbana-Champaign
Curated by ChEMBL
Affinity DataIC50: 112nMAssay Description:Inhibitory activity against FPPS in Leishmania majorMore data for this Ligand-Target Pair
TargetPolyprenyl synthetase family protein(Plasmodium falciparum (isolate 3D7))
University Of Illinois At Urbana-Champaign
Curated by ChEMBL
University Of Illinois At Urbana-Champaign
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:Inhibitory activity against FPPS in Leishmania majorMore data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Inhibition of Leishmania major recombinant squalene synthase expressed in Escherichia coli by liquid scintillation counterMore data for this Ligand-Target Pair
TargetPolyprenyl synthetase family protein(Plasmodium falciparum (isolate 3D7))
University Of Illinois At Urbana-Champaign
Curated by ChEMBL
University Of Illinois At Urbana-Champaign
Curated by ChEMBL
Affinity DataIC50: 228nMAssay Description:Inhibitory activity against FPPS in Leishmania majorMore data for this Ligand-Target Pair
TargetSqualene synthase(Homo sapiens (Human))
Instituto De Parasitolog£A Y Biomedicina&Quot;L£Pez-Neyra
Curated by ChEMBL
Instituto De Parasitolog£A Y Biomedicina&Quot;L£Pez-Neyra
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Inhibition of human recombinant squalene synthaseMore data for this Ligand-Target Pair
TargetSqualene synthase(Homo sapiens (Human))
Instituto De Parasitolog£A Y Biomedicina&Quot;L£Pez-Neyra
Curated by ChEMBL
Instituto De Parasitolog£A Y Biomedicina&Quot;L£Pez-Neyra
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Inhibition of human recombinant squalene synthase expressed in Escherichia coli BL21(DE3 pLysS) by liquid scintillation counterMore data for this Ligand-Target Pair
TargetPolyprenyl synthetase family protein(Plasmodium falciparum (isolate 3D7))
University Of Illinois At Urbana-Champaign
Curated by ChEMBL
University Of Illinois At Urbana-Champaign
Curated by ChEMBL
Affinity DataIC50: 420nMAssay Description:Inhibitory activity against FPPS in Leishmania majorMore data for this Ligand-Target Pair
Affinity DataIC50: 490nMAssay Description:Inhibition of Leishmania major recombinant squalene synthase expressed in Escherichia coli by liquid scintillation counterMore data for this Ligand-Target Pair
TargetSqualene synthase(Homo sapiens (Human))
Instituto De Parasitolog£A Y Biomedicina&Quot;L£Pez-Neyra
Curated by ChEMBL
Instituto De Parasitolog£A Y Biomedicina&Quot;L£Pez-Neyra
Curated by ChEMBL
Affinity DataIC50: 660nMAssay Description:Inhibition of human recombinant squalene synthase expressed in Escherichia coli BL21(DE3 pLysS) by liquid scintillation counterMore data for this Ligand-Target Pair
TargetPhosphotransferase(Trypanosoma cruzi)
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Affinity DataIC50: 810nMAssay Description:Inhibitory activity against Trypanosoma cruzi hexokinaseMore data for this Ligand-Target Pair
TargetPhosphotransferase(Trypanosoma cruzi)
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Affinity DataIC50: 810nMAssay Description:Inhibition of Trypanosoma cruzi hexokinaseMore data for this Ligand-Target Pair
TargetPhosphotransferase(Trypanosoma cruzi)
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Affinity DataIC50: 810nMAssay Description:Inhibition of Trypanosoma cruzi hexokinaseMore data for this Ligand-Target Pair
TargetPhosphotransferase(Trypanosoma cruzi)
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Affinity DataIC50: 810nMAssay Description:Inhibition of Trypanosoma cruzi hexokinaseMore data for this Ligand-Target Pair
TargetPhosphotransferase(Trypanosoma cruzi)
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Instituto Venezolano De Investigaciones Cient£Ficas
Curated by ChEMBL
Affinity DataIC50: 810nMAssay Description:Inhibition of Trypanosoma cruzi hexokinaseMore data for this Ligand-Target Pair