Compile Data Set for Download or QSAR
maximum 50k data
Found 8 with Last Name = 'utata' and Initial = 'r'
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50059889((staurosporine)3-methoxy-2-methyl-4-methylamino-(2...)
Affinity DataIC50:  37nMAssay Description:Inhibition of ASK1 (unknown origin) by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM7491((4Z)-4-(2-amino-5-oxo-3,5-dihydro-4H-imidazol-4-yl...)
Affinity DataIC50:  150nMAssay Description:Inhibition of ASK1 (unknown origin) by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50059889((staurosporine)3-methoxy-2-methyl-4-methylamino-(2...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of ASK1 (unknown origin) by fluorescence correlation spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM7491((4Z)-4-(2-amino-5-oxo-3,5-dihydro-4H-imidazol-4-yl...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of ASK1 (unknown origin) by fluorescence correlation spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50243715(3-((1-methyl-1H-indol-3-yl)methylene)indolin-2-one...)
Affinity DataIC50:  8.27E+4nMAssay Description:Inhibition of ASK1 (unknown origin) by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50243715(3-((1-methyl-1H-indol-3-yl)methylene)indolin-2-one...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of ASK1 (unknown origin) by fluorescence correlation spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50059889((staurosporine)3-methoxy-2-methyl-4-methylamino-(2...)
Affinity DataKd:  110nMAssay Description:Binding affinity to ASK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50243867(CHEMBL478889 | STS-PEG-TAMRA)
Affinity DataKd:  8.00E+3nMAssay Description:Binding affinity to ASK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed