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Found 138 with Last Name = 'van heertum' and Initial = 'rl'
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50182020(2-(4-(4-(3-methoxyphenyl)piperazin-1-yl)butyl)-4-m...)
Affinity DataKi:  1.10nMAssay Description:Agonist activity assessed by stimulation of [35S]GTP-gamma-S binding to human 5HT1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50180054(CHEMBL199824 | [O-methyl-11C]2-{4-[4-(7-methoxynap...)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 1(BOVINE)
Columbia University

Curated by PDSP Ki Database
LigandPNGBDBM86757(CAS_0 | NSC_11603174 | [11C]MMP)
Affinity DataKi:  6.75nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50180054(CHEMBL199824 | [O-methyl-11C]2-{4-[4-(7-methoxynap...)
Affinity DataKi:  8.5nMAssay Description:Binding affinity to dopamine D4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50180054(CHEMBL199824 | [O-methyl-11C]2-{4-[4-(7-methoxynap...)
Affinity DataKi:  9.10nMAssay Description:Binding affinity to human 5HT7 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(BOVINE)
Columbia University

Curated by PDSP Ki Database
LigandPNGBDBM86757(CAS_0 | NSC_11603174 | [11C]MMP)
Affinity DataKi:  12.9nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(BOVINE)
Columbia University

Curated by PDSP Ki Database
LigandPNGBDBM86757(CAS_0 | NSC_11603174 | [11C]MMP)
Affinity DataKi:  15.4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDopamine receptor D4(BOVINE)
Columbia University

Curated by PDSP Ki Database
LigandPNGBDBM86757(CAS_0 | NSC_11603174 | [11C]MMP)
Affinity DataKi:  21.8nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50180054(CHEMBL199824 | [O-methyl-11C]2-{4-[4-(7-methoxynap...)
Affinity DataKi:  22nMAssay Description:Binding affinity to dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50180054(CHEMBL199824 | [O-methyl-11C]2-{4-[4-(7-methoxynap...)
Affinity DataKi:  24nMAssay Description:Binding affinity to adrenergic alpha-2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50180054(CHEMBL199824 | [O-methyl-11C]2-{4-[4-(7-methoxynap...)
Affinity DataKi:  32nMAssay Description:Binding affinity to adrenergic alpha-1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50182020(2-(4-(4-(3-methoxyphenyl)piperazin-1-yl)butyl)-4-m...)
Affinity DataKi:  34nMAssay Description:Binding affinity to 5HT2B receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50180054(CHEMBL199824 | [O-methyl-11C]2-{4-[4-(7-methoxynap...)
Affinity DataKi:  42nMAssay Description:Binding affinity to human 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAP-4 complex subunit sigma-1(BOVINE)
Columbia University

Curated by PDSP Ki Database
LigandPNGBDBM86757(CAS_0 | NSC_11603174 | [11C]MMP)
Affinity DataKi:  59.1nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50180054(CHEMBL199824 | [O-methyl-11C]2-{4-[4-(7-methoxynap...)
Affinity DataKi:  61nMAssay Description:Binding affinity to adrenergic beta-2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50180054(CHEMBL199824 | [O-methyl-11C]2-{4-[4-(7-methoxynap...)
Affinity DataKi:  63nMAssay Description:Binding affinity to dopamine D3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(BOVINE)
Columbia University

Curated by PDSP Ki Database
LigandPNGBDBM86757(CAS_0 | NSC_11603174 | [11C]MMP)
Affinity DataKi:  73.6nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine 1D receptor(Bos taurus (Bovine))
Columbia University

Curated by PDSP Ki Database
LigandPNGBDBM86757(CAS_0 | NSC_11603174 | [11C]MMP)
Affinity DataKi:  88.3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(BOVINE)
Columbia University

Curated by PDSP Ki Database
LigandPNGBDBM86757(CAS_0 | NSC_11603174 | [11C]MMP)
Affinity DataKi:  96nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50180054(CHEMBL199824 | [O-methyl-11C]2-{4-[4-(7-methoxynap...)
Affinity DataKi:  100nMAssay Description:Binding affinity to human 5HT2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50182020(2-(4-(4-(3-methoxyphenyl)piperazin-1-yl)butyl)-4-m...)
Affinity DataKi:  109nMAssay Description:Binding affinity to alpha 2C adrenergic receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50180054(CHEMBL199824 | [O-methyl-11C]2-{4-[4-(7-methoxynap...)
Affinity DataKi:  120nMAssay Description:Binding affinity to human 5HT6 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAP-3 complex subunit sigma-2(BOVINE)
Columbia University

Curated by PDSP Ki Database
LigandPNGBDBM86757(CAS_0 | NSC_11603174 | [11C]MMP)
Affinity DataKi:  123nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50180054(CHEMBL199824 | [O-methyl-11C]2-{4-[4-(7-methoxynap...)
Affinity DataKi:  150nMAssay Description:Binding affinity to histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50182020(2-(4-(4-(3-methoxyphenyl)piperazin-1-yl)butyl)-4-m...)
Affinity DataKi:  180nMAssay Description:Binding affinity to sigma1 opioid receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50182020(2-(4-(4-(3-methoxyphenyl)piperazin-1-yl)butyl)-4-m...)
Affinity DataKi:  228nMAssay Description:Binding affinity to 5HT1B receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50180054(CHEMBL199824 | [O-methyl-11C]2-{4-[4-(7-methoxynap...)
Affinity DataKi:  229nMAssay Description:Binding affinity to human 5HT5A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(BOVINE)
Columbia University

Curated by PDSP Ki Database
LigandPNGBDBM86757(CAS_0 | NSC_11603174 | [11C]MMP)
Affinity DataKi:  238nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50182020(2-(4-(4-(3-methoxyphenyl)piperazin-1-yl)butyl)-4-m...)
Affinity DataKi:  250nMAssay Description:Binding affinity to alpha 2A adrenergic receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50180054(CHEMBL199824 | [O-methyl-11C]2-{4-[4-(7-methoxynap...)
Affinity DataKi:  302nMAssay Description:Binding affinity to histamine H2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50180054(CHEMBL199824 | [O-methyl-11C]2-{4-[4-(7-methoxynap...)
Affinity DataKi:  316nMAssay Description:Binding affinity to adrenergic alpha-2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50182020(2-(4-(4-(3-methoxyphenyl)piperazin-1-yl)butyl)-4-m...)
Affinity DataKi:  328nMAssay Description:Binding affinity to 5HT7 receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50182020(2-(4-(4-(3-methoxyphenyl)piperazin-1-yl)butyl)-4-m...)
Affinity DataKi:  378nMAssay Description:Binding affinity to alpha 1B adrenergic receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50180054(CHEMBL199824 | [O-methyl-11C]2-{4-[4-(7-methoxynap...)
Affinity DataKi:  407nMAssay Description:Binding affinity to DATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50182020(2-(4-(4-(3-methoxyphenyl)piperazin-1-yl)butyl)-4-m...)
Affinity DataKi:  413nMAssay Description:Binding affinity to alpha 1A adrenergic receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50180054(CHEMBL199824 | [O-methyl-11C]2-{4-[4-(7-methoxynap...)
Affinity DataKi:  476nMAssay Description:Binding affinity to adrenergic beta-1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50180054(CHEMBL199824 | [O-methyl-11C]2-{4-[4-(7-methoxynap...)
Affinity DataKi:  480nMAssay Description:Binding affinity to sigma1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(BOVINE)
Columbia University

Curated by PDSP Ki Database
LigandPNGBDBM86757(CAS_0 | NSC_11603174 | [11C]MMP)
Affinity DataKi:  643nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50182020(2-(4-(4-(3-methoxyphenyl)piperazin-1-yl)butyl)-4-m...)
Affinity DataKi:  839nMAssay Description:Binding affinity to histamine H1 receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50180054(CHEMBL199824 | [O-methyl-11C]2-{4-[4-(7-methoxynap...)
Affinity DataKi:  1.01E+3nMAssay Description:Binding affinity to adrenergic alpha-2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(BOVINE)
Columbia University

Curated by PDSP Ki Database
LigandPNGBDBM86757(CAS_0 | NSC_11603174 | [11C]MMP)
Affinity DataKi:  1.03E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50182020(2-(4-(4-(3-methoxyphenyl)piperazin-1-yl)butyl)-4-m...)
Affinity DataKi:  2.10E+3nMAssay Description:Binding affinity to 5HT2A receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(BOVINE)
Columbia University

Curated by PDSP Ki Database
LigandPNGBDBM86757(CAS_0 | NSC_11603174 | [11C]MMP)
Affinity DataKi:  2.13E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50182020(2-(4-(4-(3-methoxyphenyl)piperazin-1-yl)butyl)-4-m...)
Affinity DataKi:  2.13E+3nMAssay Description:Binding affinity to histamine H2 receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50182020(2-(4-(4-(3-methoxyphenyl)piperazin-1-yl)butyl)-4-m...)
Affinity DataKi:  2.58E+3nMAssay Description:Binding affinity to D2 dopamine receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(BOVINE)
Columbia University

Curated by PDSP Ki Database
LigandPNGBDBM86757(CAS_0 | NSC_11603174 | [11C]MMP)
Affinity DataKi:  4.98E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50180054(CHEMBL199824 | [O-methyl-11C]2-{4-[4-(7-methoxynap...)
Affinity DataKi:  6.14E+3nMAssay Description:Binding affinity to SERTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50180054(CHEMBL199824 | [O-methyl-11C]2-{4-[4-(7-methoxynap...)
Affinity DataKi:  6.98E+3nMAssay Description:Binding affinity to NETMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons

Curated by ChEMBL
LigandPNGBDBM50180054(CHEMBL199824 | [O-methyl-11C]2-{4-[4-(7-methoxynap...)
Affinity DataKi:  7.40E+3nMAssay Description:Binding affinity to dopamine D1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1E(BOVINE)
Columbia University

Curated by PDSP Ki Database
LigandPNGBDBM86757(CAS_0 | NSC_11603174 | [11C]MMP)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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