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Found 16 with Last Name = 'varela' and Initial = 'cl'
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50398447(Aromasin | EXEMESTANE)
Affinity DataIC50:  50nMAssay Description:Inhibition of human placental microsome aromatase using [1beta-3H] androstenedione as substrate after 15 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50069753(CHEMBL3407538)
Affinity DataIC50:  100nMAssay Description:Inhibition of human placental microsome aromatase using [1beta-3H] androstenedione as substrate after 15 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50168058(CHEMBL3798461)
Affinity DataIC50:  110nMAssay Description:Inhibition of aromatase in human placental microsomes using [1beta-3H]-androstenedione as substrate assessed as tritiated H2O release after 15 mins b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50069753(CHEMBL3407538)
Affinity DataIC50:  250nMAssay Description:Inhibition of human placental microsome aromatase expressed in human MCF7 cells using [1beta-3H] androstenedione as substrate after 1 hr by liquid sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50168056(CHEMBL3799363)
Affinity DataIC50:  250nMAssay Description:Inhibition of aromatase in human placental microsomes using [1beta-3H]-androstenedione as substrate assessed as tritiated H2O release after 15 mins b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50123151(CHEMBL3623223)
Affinity DataIC50:  470nMAssay Description:Inhibition of aromatase in human placental microsomes using [1beta-3H]-androstenedione as substrate assessed as tritiated H2O release after 15 mins b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50168057(CHEMBL3800417)
Affinity DataIC50:  530nMAssay Description:Inhibition of aromatase in human placental microsomes using [1beta-3H]-androstenedione as substrate assessed as tritiated H2O release after 15 mins b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50069755(CHEMBL3407536)
Affinity DataIC50:  620nMAssay Description:Inhibition of human placental microsome aromatase using [1beta-3H] androstenedione as substrate after 15 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50069752(CHEMBL3407539)
Affinity DataIC50:  670nMAssay Description:Inhibition of human placental microsome aromatase using [1beta-3H] androstenedione as substrate after 15 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50069755(CHEMBL3407536)
Affinity DataIC50:  730nMAssay Description:Inhibition of human placental microsome aromatase expressed in human MCF7 cells using [1beta-3H] androstenedione as substrate after 1 hr by liquid sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50069754(CHEMBL3407537)
Affinity DataIC50:  810nMAssay Description:Inhibition of human placental microsome aromatase using [1beta-3H] androstenedione as substrate after 15 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50398447(Aromasin | EXEMESTANE)
Affinity DataIC50:  900nMAssay Description:Inhibition of human placental microsome aromatase expressed in human MCF7 cells using [1beta-3H] androstenedione as substrate after 1 hr by liquid sc...More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50069752(CHEMBL3407539)
Affinity DataIC50:  980nMAssay Description:Inhibition of human placental microsome aromatase expressed in human MCF7 cells using [1beta-3H] androstenedione as substrate after 1 hr by liquid sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50069754(CHEMBL3407537)
Affinity DataIC50:  1.18E+3nMAssay Description:Inhibition of human placental microsome aromatase expressed in human MCF7 cells using [1beta-3H] androstenedione as substrate after 1 hr by liquid sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50388393(CHEMBL2058266)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of aromatase in disrupted human MCF-7aro cells using [1beta-3H] androstenedione as substrate incubated for 1 hrs in the presence of NADPHMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50388393(CHEMBL2058266)
Affinity DataIC50:  8.50E+3nMAssay Description:Inhibition of aromatase in human MCF-7aro cells using [1beta-3H] androstenedione as substrate incubated for 1 hrsMore data for this Ligand-Target Pair
In DepthDetails PubMed