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Found 126 with Last Name = 'vogtherr' and Initial = 'm'
TargetThymidylate kinase(Mycobacterium tuberculosis)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498068(CHEMBL3394234)
Affinity DataIC50:  1nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498069(CHEMBL3394233)
Affinity DataIC50:  2nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetThymidylate kinase(Mycobacterium tuberculosis)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498093(CHEMBL3394236)
Affinity DataIC50:  2nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498070(CHEMBL3394163)
Affinity DataIC50:  3nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498096(CHEMBL3394232)
Affinity DataIC50:  5nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498082(CHEMBL3394237)
Affinity DataIC50:  5nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498089(CHEMBL3394162)
Affinity DataIC50:  6nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498090(CHEMBL3394161)
Affinity DataIC50:  6nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498057(CHEMBL3394235)
Affinity DataIC50:  17nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498060(CHEMBL3394249)
Affinity DataIC50:  22nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498059(CHEMBL3394250)
Affinity DataIC50:  32nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498061(CHEMBL3394247)
Affinity DataIC50:  100nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498062(CHEMBL3394246)
Affinity DataIC50:  140nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498056(CHEMBL3394242)
Affinity DataIC50:  200nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetThymidylate kinase(Mycobacterium tuberculosis)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498080(CHEMBL3394245)
Affinity DataIC50:  240nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498074(CHEMBL3394155)
Affinity DataIC50:  250nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86138(LDHA Inhibitor, 34)
Affinity DataIC50:  270nMpH: 7.5 T: 2°CAssay Description:Enzyme assay using lactate dehydrogenase A (LDHA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86135(LDHA Inhibitor, 31)
Affinity DataIC50:  290nMpH: 7.5 T: 2°CAssay Description:Enzyme assay using lactate dehydrogenase A (LDHA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498079(CHEMBL3394248)
Affinity DataIC50:  330nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498088(CHEMBL3394240)
Affinity DataIC50:  350nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498085(CHEMBL3394151)
Affinity DataIC50:  420nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetThymidylate kinase(Mycobacterium tuberculosis)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498073(CHEMBL3394157)
Affinity DataIC50:  430nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86137(LDHA Inhibitor, 33)
Affinity DataIC50:  500nMpH: 7.5 T: 2°CAssay Description:Enzyme assay using lactate dehydrogenase A (LDHA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498063(CHEMBL3394244)
Affinity DataIC50:  820nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498065(CHEMBL3394241)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498058(CHEMBL3394153)
Affinity DataIC50:  1.01E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498091(CHEMBL3394160)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498094(CHEMBL3394154)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498077(CHEMBL3394148)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498054(CHEMBL1477426)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86133(LDHA Inhibitor, 29)
Affinity DataIC50:  1.90E+3nMpH: 7.5 T: 2°CAssay Description:Enzyme assay using lactate dehydrogenase A (LDHA).More data for this Ligand-Target Pair
TargetThymidylate kinase(Mycobacterium tuberculosis)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498078(CHEMBL3394146)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498064(CHEMBL3394243)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498084(CHEMBL3394156)
Affinity DataIC50:  2.63E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498095(CHEMBL3394152)
Affinity DataIC50:  2.73E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86131(LDHA Inhibitor, 27)
Affinity DataIC50:  3.10E+3nMpH: 7.5 T: 2°CAssay Description:Enzyme assay using lactate dehydrogenase A (LDHA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498055(CHEMBL3394145)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86130(LDHA Inhibitor, 26)
Affinity DataIC50:  4.20E+3nMpH: 7.5 T: 2°CAssay Description:Enzyme assay using lactate dehydrogenase A (LDHA).More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86136(LDHA Inhibitor, 32)
Affinity DataIC50:  7.40E+3nMpH: 7.5 T: 2°CAssay Description:Enzyme assay using lactate dehydrogenase A (LDHA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498076(CHEMBL3394149)
Affinity DataIC50:  7.70E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
Astrazeneca

LigandPNGBDBM23251(1,2,5-Thiadiazole, TDA1 | 4-hydroxy-1,2,5-thiadiaz...)
Affinity DataIC50:  7.80E+3nMpH: 7.5 T: 2°CAssay Description:Enzyme assay using lactate dehydrogenase A (LDHA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498072(CHEMBL3394158)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
Astrazeneca

LigandPNGBDBM86114(LDHA Inhibitor, 8)
Affinity DataIC50:  9.40E+3nMpH: 7.5 T: 2°CAssay Description:Enzyme assay using lactate dehydrogenase A (LDHA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498083(CHEMBL3394159)
Affinity DataIC50:  1.43E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498075(CHEMBL3394150)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498087(CHEMBL3394251)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86134(LDHA Inhibitor, 30)
Affinity DataIC50:  2.95E+4nMpH: 7.5 T: 2°CAssay Description:Enzyme assay using lactate dehydrogenase A (LDHA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498092(CHEMBL3394252)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498086(CHEMBL3394147)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498071(CHEMBL110569)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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