Affinity DataIC50: 0.160nMAssay Description:Binding affinity to estrogen receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 0.170nMAssay Description:Binding affinity to estrogen receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 0.170nMAssay Description:Binding affinity to estrogen receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 0.170nMAssay Description:Binding affinity to estrogen receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 0.180nMAssay Description:Induction of estrogen receptor degradation in human MCF7 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.210nMAssay Description:Binding affinity to estrogen receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 0.220nMAssay Description:Binding affinity to estrogen receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 0.240nMAssay Description:Binding affinity to estrogen receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 0.280nMAssay Description:Binding affinity to estrogen receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 0.440nMAssay Description:Binding affinity to estrogen receptor (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using PIP2:3PS peptide as substrate preincubated for 15 mins followed by ATP addition at Km concentration an...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using PIP2:3PS peptide as substrate preincubated for 15 mins followed by ATP addition at Km concentration an...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Affinity DataIC50: 0.600nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using PIP2:3PS peptide as substrate preincubated for 15 mins followed by ATP addition at Km concentration an...More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
German University In Cairo
Curated by ChEMBL
German University In Cairo
Curated by ChEMBL
Affinity DataIC50: 0.670nMAssay Description:Inhibition of N-terminal FLAG-tagged human Clk1 using myelin basic protein as substrate preincubated for 10 mins followed by ATP addition measured af...More data for this Ligand-Target Pair
Affinity DataIC50: 0.760nMAssay Description:Binding affinity to estrogen receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 0.870nMAssay Description:Binding affinity to estrogen receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 0.980nMAssay Description:Binding affinity to estrogen receptor (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Affinity DataIC50: 1.10nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using PIP2:3PS peptide as substrate preincubated for 15 mins followed by ATP addition at Km concentration an...More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
German University In Cairo
Curated by ChEMBL
German University In Cairo
Curated by ChEMBL
Affinity DataIC50: 1.10nMAssay Description:Inhibition of human recombinant GST-tagged Clk1 (129 to 484 residues) expressed in Escherichia coli expression system using GRSRSRSRSRSRSRSR peptide ...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Affinity DataIC50: 1.10nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using PIP2:3PS peptide as substrate preincubated for 15 mins followed by ATP addition at Km concentration an...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Affinity DataIC50: 1.20nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using PIP2:3PS peptide as substrate preincubated for 15 mins followed by ATP addition at Km concentration an...More data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Binding affinity to estrogen receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Binding affinity to estrogen receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Binding affinity to estrogen receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Binding affinity to estrogen receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Binding affinity to estrogen receptor (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Affinity DataIC50: 1.70nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using PIP2:3PS peptide as substrate preincubated for 15 mins followed by ATP addition at Km concentration an...More data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:Binding affinity to estrogen receptor (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Affinity DataIC50: 1.80nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using PIP2:3PS peptide as substrate preincubated for 15 mins followed by ATP addition at Km concentration an...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using PIP2:3PS peptide as substrate preincubated for 15 mins followed by ATP addition at Km concentration an...More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Induction of estrogen receptor degradation in human MCF7 cellsMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Affinity DataIC50: 2.10nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using PIP2:3PS peptide as substrate preincubated for 15 mins followed by ATP addition at Km concentration an...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Affinity DataIC50: 2.10nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using PIP2:3PS peptide as substrate preincubated for 15 mins followed by ATP addition at Km concentration an...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Affinity DataIC50: 2.30nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using PIP2:3PS peptide as substrate preincubated for 15 mins followed by ATP addition at Km concentration an...More data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:Binding affinity to estrogen receptor (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
German University In Cairo
Curated by ChEMBL
German University In Cairo
Curated by ChEMBL
Affinity DataIC50: 2.40nMAssay Description:Inhibition of human recombinant GST-tagged Clk2 expressed in Baculovirus expression system using GRSRSRSRSRSRSRSR peptide as substrate preincubated f...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Affinity DataIC50: 2.5nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using PIP2:3PS peptide as substrate preincubated for 15 mins followed by ATP addition at Km concentration an...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Affinity DataIC50: 2.70nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using PIP2:3PS peptide as substrate preincubated for 15 mins followed by ATP addition at Km concentration an...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Affinity DataIC50: 2.70nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using PIP2:3PS peptide as substrate preincubated for 15 mins followed by ATP addition at Km concentration an...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using PIP2:3PS peptide as substrate preincubated for 15 mins followed by ATP addition at Km concentration an...More data for this Ligand-Target Pair
Affinity DataIC50: 3.20nMAssay Description:Binding affinity to estrogen receptor (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Affinity DataIC50: 3.40nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using PIP2:3PS peptide as substrate preincubated for 15 mins followed by ATP addition at Km concentration an...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Affinity DataIC50: 3.5nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using PIP2:3PS peptide as substrate preincubated for 15 mins followed by ATP addition at Km concentration an...More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Induction of estrogen receptor degradation in human MCF7 cellsMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
German University In Cairo
Curated by ChEMBL
German University In Cairo
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of human recombinant GST-tagged Clk1 (129 to 484 residues) expressed in Escherichia coli expression system using GRSRSRSRSRSRSRS peptide a...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Affinity DataIC50: 4.10nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using PIP2:3PS peptide as substrate preincubated for 15 mins followed by ATP addition at Km concentration an...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Affinity DataIC50: 4.30nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using PIP2:3PS peptide as substrate preincubated for 15 mins followed by ATP addition at Km concentration an...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Affinity DataIC50: 4.40nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using PIP2:3PS peptide as substrate preincubated for 15 mins followed by ATP addition at Km concentration an...More data for this Ligand-Target Pair
Affinity DataIC50: 4.70nMAssay Description:Binding affinity to estrogen receptor (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Luoxin Pharmaceutical (Shanghai) Co.
Curated by ChEMBL
Affinity DataIC50: 4.90nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using PIP2:3PS peptide as substrate preincubated for 15 mins followed by ATP addition at Km concentration an...More data for this Ligand-Target Pair