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Found 114 with Last Name = 'wapenaar' and Initial = 'h'
TargetC-C motif chemokine 2(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50440552(CHEMBL2426340)
Affinity DataKi:  3.60nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C motif chemokine 2(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50440556(CHEMBL2426334)
Affinity DataKi:  3.90nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C motif chemokine 2(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50440549(CHEMBL2426351)
Affinity DataKi:  6.10nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C motif chemokine 2(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50440557(CHEMBL2426335)
Affinity DataKi:  6.30nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C motif chemokine 2(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257898((1S,3R)-N-(3,5-bis(trifluoromethyl)benzyl)-1-isopr...)
Affinity DataKi:  6.80nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C motif chemokine 2(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50440552(CHEMBL2426340)
Affinity DataKi:  7.20nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C motif chemokine 2(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50440552(CHEMBL2426340)
Affinity DataKi:  7.20nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT8(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM43339(4-amino-1-naphthalenol;hydrochloride | 4-amino-1-n...)
Affinity DataKi:  17nMAssay Description:Inhibition of N-terminal His6-tagged KAT8 catalytic domain (125 to 458 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) assessed as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C motif chemokine 2(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50440551(CHEMBL2426354)
Affinity DataKi:  18nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C motif chemokine 2(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50440558(CHEMBL2426336)
Affinity DataKi:  27nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C motif chemokine 2(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50440550(CHEMBL2426352)
Affinity DataKi:  29nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C motif chemokine 2(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257900((1S,3R)-N-(3,5-bis(trifluoromethyl)benzyl)-1-isopr...)
Affinity DataKi:  31nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C motif chemokine 2(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50440545(CHEMBL2426345)
Affinity DataKi:  33nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C motif chemokine 2(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50440559(CHEMBL2426337)
Affinity DataKi:  35nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C motif chemokine 2(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50440546(CHEMBL2426346)
Affinity DataKi:  43nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C motif chemokine 2(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257992((1S,3R)-N-(3,5-bis(trifluoromethyl)benzyl)-3-(2,3-...)
Affinity DataKi:  50nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C motif chemokine 2(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50440554(CHEMBL2426357)
Affinity DataKi:  54nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C motif chemokine 2(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50440553(CHEMBL2426356)
Affinity DataKi:  55nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C motif chemokine 2(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50440548(CHEMBL2426348)
Affinity DataKi:  70nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C motif chemokine 2(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50440547(CHEMBL2426347)
Affinity DataKi:  86nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C motif chemokine 2(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257792((1S,3R)-N-(3,5-bis(trifluoromethyl)benzyl)-3-(cycl...)
Affinity DataKi:  110nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C motif chemokine 2(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50440555(CHEMBL2426333)
Affinity DataKi:  130nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C motif chemokine 2(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50440544(CHEMBL2426344)
Affinity DataKi:  134nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C motif chemokine 2(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50440542(CHEMBL2426342)
Affinity DataKi:  437nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C motif chemokine 2(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50440543(CHEMBL2426343)
Affinity DataKi:  2.40E+3nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT8(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM43339(4-amino-1-naphthalenol;hydrochloride | 4-amino-1-n...)
Affinity DataKi:  2.60E+3nMAssay Description:Inhibition of N-terminal His6-tagged KAT8 catalytic domain (125 to 458 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) assessed as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT8(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50469667(6-Decylsalicylic Acid | CHEMBL416038)
Affinity DataKi:  3.70E+4nMAssay Description:Inhibition of recombinant N-terminal His6-tagged KAT8 (unknown origin) expressed in Escherichia Coli BL21 DE3 cells assessed as reduction of Co A lev...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT8(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50499159(CHEMBL3735604)
Affinity DataKi:  5.70E+4nMAssay Description:Inhibition of recombinant N-terminal His6-tagged KAT8 (unknown origin) expressed in Escherichia Coli BL21 DE3 cells assessed as reduction of Co A lev...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT8(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50240436(2-Hydroxy-6-pentadecyl-benzoic acid | 2-hydroxy-6-...)
Affinity DataKi:  6.40E+4nMAssay Description:Inhibition of recombinant N-terminal His6-tagged KAT8 (unknown origin) expressed in Escherichia Coli BL21 DE3 cells assessed as reduction of Co A lev...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT8(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50499157(CHEMBL3735420)
Affinity DataKi:  7.90E+4nMAssay Description:Inhibition of recombinant N-terminal His6-tagged KAT8 (unknown origin) expressed in Escherichia Coli BL21 DE3 cells assessed as reduction of Co A lev...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT8(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50499160(CHEMBL3736378)
Affinity DataKi:  1.57E+5nMAssay Description:Inhibition of recombinant N-terminal His6-tagged KAT8 (unknown origin) expressed in Escherichia Coli BL21 DE3 cells assessed as reduction of Co A lev...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50456444(CHEMBL3734823)
Affinity DataIC50:  320nMAssay Description:Inhibition of human recombinant Histone acetyltransferase p300 catalytic domain (1284-1672 residues) using [3H]Acetyl-CoA and histone H3 substrate at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50282619(CHEMBL4159902)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of KAT3B catalytic domain (1284 to 1673 residues) (unknown origin) using SGRGKGGKGLGKGGAKRHRK-NH2 as substrate after 5 mins in presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT8(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM43339(4-amino-1-naphthalenol;hydrochloride | 4-amino-1-n...)
Affinity DataIC50:  1.10E+3nMAssay Description:Tested for antagonist activity against NK1 receptor in rabbit vena cava by using substance P (SP) as agonistMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM43339(4-amino-1-naphthalenol;hydrochloride | 4-amino-1-n...)
Affinity DataIC50:  1.40E+3nMAssay Description:Tested for antagonist activity against NK1 receptor in rabbit vena cava by using substance P (SP) as agonistMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT8(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM43339(4-amino-1-naphthalenol;hydrochloride | 4-amino-1-n...)
Affinity DataIC50:  1.60E+3nMAssay Description:Tested for antagonist activity against NK-3 receptor in rat portal vein by using Neurokinin B as agonistMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT8(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM43339(4-amino-1-naphthalenol;hydrochloride | 4-amino-1-n...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of N-terminal His6-tagged KAT8 catalytic domain (125 to 458 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM43307(4-methyl-N-(4-oxidanylnaphthalen-1-yl)benzenesulfo...)
Affinity DataIC50:  2.60E+3nMAssay Description:Tested for antagonist activity against NK-3 receptor in rat portal vein by using Neurokinin B as agonistMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50282490(CHEMBL4172065)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of KAT3B catalytic domain (1284 to 1673 residues) (unknown origin) using SGRGKGGKGLGKGGAKRHRK-NH2 as substrate after 5 mins in presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM43339(4-amino-1-naphthalenol;hydrochloride | 4-amino-1-n...)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of KAT2B catalytic domain (492 to 658 residues) (unknown origin) using H-ARTKQTARKSTGGKAPRKQL-OH as substrate after 5 mins in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50303931(4-(dimethylamino)naphthalen-1-ol | CHEMBL571241)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of KAT3B catalytic domain (1284 to 1673 residues) (unknown origin) using SGRGKGGKGLGKGGAKRHRK-NH2 as substrate after 5 mins in presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50282490(CHEMBL4172065)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of KAT2B catalytic domain (492 to 658 residues) (unknown origin) using H-ARTKQTARKSTGGKAPRKQL-OH as substrate after 5 mins in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50303931(4-(dimethylamino)naphthalen-1-ol | CHEMBL571241)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of KAT2B catalytic domain (492 to 658 residues) (unknown origin) using H-ARTKQTARKSTGGKAPRKQL-OH as substrate after 5 mins in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage migration inhibitory factor(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50455046(CHEMBL4207747)
Affinity DataIC50:  6.20E+3nMAssay Description:Inhibition of recombinant His-tagged MIF tautomerase activity (unknown origin) using 4-HPP as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMacrophage migration inhibitory factor(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50455042(CHEMBL4209531)
Affinity DataIC50:  7.10E+3nMAssay Description:Inhibition of recombinant His-tagged MIF tautomerase activity (unknown origin) using 4-HPP as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50282619(CHEMBL4159902)
Affinity DataIC50:  7.10E+3nMAssay Description:Inhibition of KAT2B catalytic domain (492 to 658 residues) (unknown origin) using H-ARTKQTARKSTGGKAPRKQL-OH as substrate after 5 mins in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT8(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50282619(CHEMBL4159902)
Affinity DataIC50:  7.60E+3nMAssay Description:Inhibition of N-terminal His6-tagged KAT8 catalytic domain (125 to 458 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage migration inhibitory factor(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50455047(CHEMBL4217822)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of recombinant His-tagged MIF tautomerase activity (unknown origin) using 4-HPP as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT8(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM43339(4-amino-1-naphthalenol;hydrochloride | 4-amino-1-n...)
Affinity DataIC50:  9.70E+3nMAssay Description:Inhibition of N-terminal His6-tagged KAT8 catalytic domain (125 to 458 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM43307(4-methyl-N-(4-oxidanylnaphthalen-1-yl)benzenesulfo...)
Affinity DataIC50:  1.20E+4nMAssay Description:Tested for antagonist activity against NK-3 receptor in rat portal vein by using Neurokinin B as agonistMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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