Affinity DataKi: 16nMAssay Description:Displacement of [3H]DPCPX from human A2B receptor expressed in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Displacement of [3H]DPCPX from human A2B receptor expressed in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Displacement of [3H]DPCPX from human A2B receptor expressed in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Displacement of [3H]DPCPX from human A2B receptor expressed in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Displacement of [3H]DPCPX from human A2B receptor expressed in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Displacement of [3H]DPCPX from human A2B receptor expressed in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 69nMAssay Description:Displacement of [3H]DPCPX from human A2B receptor expressed in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 115nMAssay Description:Displacement of [3H]DPCPX from human A2B receptor expressed in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 116nMAssay Description:Displacement of [3H]DPCPX from human A2B receptor expressed in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 119nMAssay Description:Displacement of [3H]DPCPX from human A2B receptor expressed in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
Celltech R&D
Curated by ChEMBL
Celltech R&D
Curated by ChEMBL
Affinity DataKi: 423nMAssay Description:Inhibition of human recombinant phosphodiesterase 4AMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [2H]NECA from human A3 receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [2H]NECA from human A3 receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [2H]NECA from human A3 receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [2H]NECA from human A3 receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [2H]NECA from human A3 receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [2H]NECA from human A3 receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [2H]NECA from human A3 receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [2H]NECA from human A3 receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [2H]NECA from human A3 receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [2H]NECA from human A3 receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
Celltech R&D
Curated by ChEMBL
Celltech R&D
Curated by ChEMBL
Affinity DataKi: 1.17E+3nMAssay Description:Inhibition of human recombinant phosphodiesterase 4AMore data for this Ligand-Target Pair
Affinity DataKi: >2.50E+3nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: >2.50E+3nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: >2.50E+3nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: >2.50E+3nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: >2.50E+3nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: >2.50E+3nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: >2.50E+3nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: >2.50E+3nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: >2.50E+3nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: >2.50E+3nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HeLa cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
Celltech R&D
Curated by ChEMBL
Celltech R&D
Curated by ChEMBL
Affinity DataKi: >8.00E+3nMAssay Description:Inhibition of human recombinant phosphodiesterase 4AMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0500nMAssay Description:Inhibition of VLA-4 to VCAM-1 bindingMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of binding of Very late antigen 4/vascular cell adhesion molecule 1 in a protein-based ligand binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of binding of Very late antigen 4/vascular cell adhesion molecule 1 in a protein-based ligand binding assayMore data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
Celltech R&D
Curated by ChEMBL
Celltech R&D
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Inhibition of human recombinant phosphodiesterase 4AMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Inhibition of binding of Very late antigen 4/vascular cell adhesion molecule 1 in a cell based ligand binding assay (Jurkat cells)More data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibition of binding of Very late antigen 4/vascular cell adhesion molecule 1 in a protein-based ligand binding assayMore data for this Ligand-Target Pair