Affinity DataKi: 1nMAssay Description:Radioligand binding assay using CRTH2.More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Radioligand binding assay using CRTH2.More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Radioligand binding assay using CRTH2.More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Radioligand binding assay using CRTH2.More data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Radioligand binding assay using CRTH2.More data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Radioligand binding assay using CRTH2.More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of [3H]WIN-55212-2 from human CB2R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Displacement of [3H]WIN-55212-2 from human CB2R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Displacement of [3H]WIN-55212-2 from human CB2R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 61nMAssay Description:Displacement of [3H]CP55940 from human CB1R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 155nMAssay Description:Displacement of [3H]WIN-55212-2 from human CB2R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 215nMAssay Description:Displacement of [3H]WIN-55212-2 from human CB2R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 235nMAssay Description:Displacement of [3H]WIN-55212-2 from human CB2R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 258nMAssay Description:Radioligand binding assay using CRTH2.More data for this Ligand-Target Pair
Affinity DataKi: 275nMAssay Description:Displacement of [3H]CP55940 from human CB1R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 290nMAssay Description:Displacement of [3H]WIN-55212-2 from human CB2R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Displacement of [3H]WIN-55212-2 from human CB2R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 320nMAssay Description:Displacement of [3H]WIN-55212-2 from human CB2R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 355nMAssay Description:Displacement of [3H]WIN-55212-2 from human CB2R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 360nMAssay Description:Displacement of [3H]WIN-55212-2 from human CB2R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 380nMAssay Description:Displacement of [3H]WIN-55212-2 from human CB2R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 450nMAssay Description:Displacement of [3H]WIN-55212-2 from human CB2R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 490nMAssay Description:Displacement of [3H]WIN-55212-2 from human CB2R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 979nMAssay Description:Radioligand binding assay using CRTH2.More data for this Ligand-Target Pair
Affinity DataKi: 3.20E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55940 from human CB1R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55940 from human CB1R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: >6.00E+4nMAssay Description:Displacement of [3H]CP55940 from human CB1R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: >6.00E+4nMAssay Description:Displacement of [3H]CP55940 from human CB1R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: >6.00E+4nMAssay Description:Displacement of [3H]CP55940 from human CB1R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: >6.00E+4nMAssay Description:Displacement of [3H]CP55940 from human CB1R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: >6.00E+4nMAssay Description:Displacement of [3H]CP55940 from human CB1R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: >6.00E+4nMAssay Description:Displacement of [3H]CP55940 from human CB1R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: >6.00E+4nMAssay Description:Displacement of [3H]CP55940 from human CB1R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: >6.00E+4nMAssay Description:Displacement of [3H]CP55940 from human CB1R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: >6.00E+4nMAssay Description:Displacement of [3H]CP55940 from human CB1R expressed in CHO cellsMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
University Of Oxford
Curated by ChEMBL
University Of Oxford
Curated by ChEMBL
Affinity DataIC50: 0.00600nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
University Of Oxford
Curated by ChEMBL
University Of Oxford
Curated by ChEMBL
Affinity DataIC50: 0.00900nMAssay Description:Inhibition of PIM3 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-2(Homo sapiens (Human))
University Of Oxford
Curated by ChEMBL
University Of Oxford
Curated by ChEMBL
Affinity DataIC50: 0.0180nMAssay Description:Inhibition of PIM2 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
University Of Oxford
Curated by ChEMBL
University Of Oxford
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Inhibition of human PIM1 using full-length BAD as substrateMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
University Of Oxford
Curated by ChEMBL
University Of Oxford
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Inhibition of human PIM1 using full length BAD peptide substrate in presence of ATP at Km concentrationMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
University Of Oxford
Curated by ChEMBL
University Of Oxford
Curated by ChEMBL
Affinity DataIC50: 1.40nMAssay Description:Inhibition of recombinant PIM1 (unknown origin) by pyruvate kinase/lactate dehydrogenase-coupled assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
University Of Oxford
Curated by ChEMBL
University Of Oxford
Curated by ChEMBL
Affinity DataIC50: 1.90nMAssay Description:Inhibition of human PIM3 using full length BAD peptide substrate in presence of ATP at Km concentrationMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
University Of Oxford
Curated by ChEMBL
University Of Oxford
Curated by ChEMBL
Affinity DataIC50: 1.90nMAssay Description:Inhibition of human PIM3 using full-length BAD as substrateMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
University Of Oxford
Curated by ChEMBL
University Of Oxford
Curated by ChEMBL
Affinity DataIC50: 2.20nMAssay Description:Inhibition of recombinant PIM1 (unknown origin) by pyruvate kinase/lactate dehydrogenase-coupled assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
University Of Oxford
Curated by ChEMBL
University Of Oxford
Curated by ChEMBL
Affinity DataIC50: 2.40nMAssay Description:Inhibition of recombinant PIM1 (unknown origin) by pyruvate kinase/lactate dehydrogenase-coupled assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
University Of Oxford
Curated by ChEMBL
University Of Oxford
Curated by ChEMBL
Affinity DataIC50: 2.90nMAssay Description:Inhibition of recombinant PIM1 (unknown origin) by pyruvate kinase/lactate dehydrogenase-coupled assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
University Of Oxford
Curated by ChEMBL
University Of Oxford
Curated by ChEMBL
Affinity DataIC50: 3.60nMAssay Description:Inhibition of recombinant PIM1 (unknown origin) by pyruvate kinase/lactate dehydrogenase-coupled assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
University Of Oxford
Curated by ChEMBL
University Of Oxford
Curated by ChEMBL
Affinity DataIC50: 4.90nMAssay Description:Inhibition of PIM1 (unknown origin) by coupled kinetic assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
University of Oxford
Curated by ChEMBL
University of Oxford
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of P13Kalpha (unknown origin)More data for this Ligand-Target Pair