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Found 580 with Last Name = 'xu' and Initial = 'yz'

Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

Ki: 0.300nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532486(CHEMBL4564992)

Ki: 0.300nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532506(CHEMBL4536431)

Ki: 0.5nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532506(CHEMBL4536431)

Ki: 0.5nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532508(CHEMBL4471576)

Ki: 0.5nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532518(CHEMBL4440420)

Ki: 0.5nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532518(CHEMBL4440420)

Ki: 0.5nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532508(CHEMBL4471576)

Ki: 0.5nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532502(CHEMBL4538923)

Ki: 0.700nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532502(CHEMBL4538923)

Ki: 0.700nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532512(CHEMBL4539105)

Ki: 0.800nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532512(CHEMBL4539105)

Ki: 0.800nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532507(CHEMBL4593797)

Ki: 0.900nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532507(CHEMBL4593797)

Ki: 0.900nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532489(CHEMBL4434692)

Ki: 1.10nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532489(CHEMBL4434692)

Ki: 1.10nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532521(CHEMBL4524740)

Ki: 1.40nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532503(CHEMBL4458060)

Ki: 1.40nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532503(CHEMBL4458060)

Ki: 1.40nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532521(CHEMBL4524740)

Ki: 1.40nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532505(CHEMBL4535404)

Ki: 1.80nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532505(CHEMBL4535404)

Ki: 1.80nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sodium-dependent noradrenaline transporter(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL

BDBM35229(3-(10,11-dihydro-5H-dibenzo[b,f]azepin-5-yl)-N-met...)

Ki: 2.5nMAssay Description:Displacement of [3H]nisoxetine from human NET expressed in HEK293 cells measured after 30 minsMore data for this Ligand-Target Pair

Reactome pathway KEGG
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Sodium-dependent noradrenaline transporter(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL

BDBM35229(3-(10,11-dihydro-5H-dibenzo[b,f]azepin-5-yl)-N-met...)

Ki: 2.5nMAssay Description:Displacement of [3H]nisoxetine from human NET expressed in HEK293 cells measured after 30 minsMore data for this Ligand-Target Pair

Reactome pathway KEGG
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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532516(CHEMBL4460187)

Ki: 2.60nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532516(CHEMBL4460187)

Ki: 2.60nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532493(CHEMBL4533250)

Ki: 2.70nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532493(CHEMBL4533250)

Ki: 2.70nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532515(CHEMBL4470605)

Ki: 3.20nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532515(CHEMBL4470605)

Ki: 3.20nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532513(CHEMBL4579980)

Ki: 3.40nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532513(CHEMBL4579980)

Ki: 3.40nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532501(CHEMBL4452090)

Ki: 3.70nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532501(CHEMBL4452090)

Ki: 3.70nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532497(CHEMBL4447015)

Ki: 4nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532497(CHEMBL4447015)

Ki: 4nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532517(CHEMBL4454404)

Ki: 4.40nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532517(CHEMBL4454404)

Ki: 4.40nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532509(CHEMBL4549596)

Ki: 5.30nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532509(CHEMBL4549596)

Ki: 5.30nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sodium-dependent serotonin transporter(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL

BDBM50020712(10,11-dihydro-5-(gamma-dimethylaminopropylidene)-5...)

Ki: 5.40nMAssay Description:Displacement of [3H]citalopram from human SERT expressed in HEK293 cells measured after 30 minsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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Sodium-dependent serotonin transporter(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL

BDBM50020712(10,11-dihydro-5-(gamma-dimethylaminopropylidene)-5...)

Ki: 5.40nMAssay Description:Displacement of [3H]citalopram from human SERT expressed in HEK293 cells measured after 30 minsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532490(CHEMBL4563018)

Ki: 6nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532490(CHEMBL4563018)

Ki: 6nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532494(CHEMBL4581357)

Ki: 6.60nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532494(CHEMBL4581357)

Ki: 6.60nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sodium-dependent dopamine transporter(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL

BDBM22165(1-{2-[bis(4-fluorophenyl)methoxy]ethyl}-4-(3-pheny...)

Ki: 8.80nMAssay Description:Displacement of [3H]-WIN35428 from human DAT expressed in HEK293 cells measured after 30 minsMore data for this Ligand-Target Pair

NCI pathway Reactome pathway KEGG
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Sodium-dependent dopamine transporter(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL

BDBM22165(1-{2-[bis(4-fluorophenyl)methoxy]ethyl}-4-(3-pheny...)

Ki: 8.80nMAssay Description:Displacement of [3H]-WIN35428 from human DAT expressed in HEK293 cells measured after 30 minsMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532482(CHEMBL4586113)

Ki: 13nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
East China Normal University

Curated by ChEMBL

BDBM50532495(CHEMBL4466675)

Ki: 13nMAssay Description:Displacement of [3H]-pentazocine from rat brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair

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Displayed 1 to 50 (of 580 total ) | Next | Last >>

Filter my 580 hits

Targets 14▿
- Presenilin-1 109
- Integrin alpha-4/beta-1 98
- Sigma non-opioid intracellular receptor 1 94
- Sigma intracellular receptor 2 94
- Beta-secretase 1 61
- Cathepsin D 45
- Integrin alpha-4/beta-7 38
- Sodium-dependent serotonin transporter 12
- Sodium-dependent noradrenaline transporter 12
- Sodium-dependent dopamine transporter 12
- Peroxisome proliferator-activated receptor alpha/delta/gamma 2
- Integrin alpha-V/beta-1 1
- Integrin alpha-L/beta-2 1
- Integrin alpha-5/beta-1 1
- ...
Publications 10▿
- J Med Chem 59: 6329-43 (2016) 224
- Bioorg Med Chem Lett 23: 4370-3 (2013) 107
- Bioorg Med Chem Lett 20: 6034-9 (2010) 87
- Bioorg Med Chem Lett 20: 2195-9 (2010) 71
- Bioorg Med Chem Lett 23: 996-1000 (2013) 38
- Bioorg Med Chem Lett 21: 1741-3 (2011) 28
- Bioorg Med Chem Lett 23: 2181-6 (2013) 17
- Bioorg Med Chem Lett 23: 3070-4 (2013) 4
- Bioorg Med Chem Lett 26: 338-42 (2016) 2
- Bioorg Med Chem Lett 23: 3075-80 (2013) 2
Institutions 3▿
- Elan Pharmaceuticals 354
- East China Normal University 224
- Northwest A & F University 2
Affinity: 0.13 to 6.4E+5 nM▿
- Ki 224
- IC50 354
- EC50 2
- Affinity ≤ nM
Xtal structures: 6
Docked structures: 0
Catalog Cmpds: 11