TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.110nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.160nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.260nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.290nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.350nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.360nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.380nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.380nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Mixed-type inhibition of AChE in mouse cerebral cortex using acetylthiocholine iodide as substrate by double reciprocal Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.410nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.450nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.460nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.590nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.991nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Binding affinity at endothelin receptor subtype AMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 3.80nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 6.5nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 9.10nMAssay Description:Inhibition of human factor 9a using CH3SO2-DCHG-Gly-Arg-AFC.AcOH as substrate preinubated for 30 mins followed by substrate addition measured after 1...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 9.10nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 9.80nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Binding affinity at type 1 angiotensin 2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibition of human factor 9a using CH3SO2-DCHG-Gly-Arg-AFC.AcOH as substrate preinubated for 30 mins followed by substrate addition measured after 1...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 26nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 32nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 33nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 37nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 41nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 42nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 57nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 60nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 61nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 68nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 74nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 96nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Ability to inhibit the hydrolysis of chromogenic 4-phenylazophenyl ester from the peptide fragment Ac- DTEDVVP(Nva)-O-4-PAP in a HCV protease continu...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 117nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 145nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor expressed in HEK293 cells by liquid scintillation spectrophotometryMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 150nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor expressed in HEK293 cells by liquid scintillation spectrophotometryMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 153nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor expressed in HEK293 cells by liquid scintillation spectrophotometryMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 153nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor expressed in HEK293 cells by liquid scintillation spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: 160nMAssay Description:Ability to inhibit the hydrolysis of chromogenic 4-phenylazophenyl ester from the peptide fragment Ac- DTEDVVP(Nva)-O-4-PAP in a HCV protease continu...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 256nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor expressed in HEK293 cells by liquid scintillation spectrophotometryMore data for this Ligand-Target Pair