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Found 51 with Last Name = 'yoo' and Initial = 'yj'
TargetProthrombin(Homo sapiens (Human))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069294((S)-3-[4-(carbohydrazonamidol)-phenyl]-N-cyclopent...)
Affinity DataKi:  0.380nMAssay Description:Binding affinity towards human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069294((S)-3-[4-(carbohydrazonamidol)-phenyl]-N-cyclopent...)
Affinity DataKi:  0.380nMAssay Description:Compound was tested for inhibitory activity against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069294((S)-3-[4-(carbohydrazonamidol)-phenyl]-N-cyclopent...)
Affinity DataKi:  1.10nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50071729(CHEMBL313826 | Naphthalene-2-sulfonic acid [(S)-1-...)
Affinity DataKi:  3.10nMAssay Description:Binding affinity towards human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50071723((S)-3-(4-Aminomethyl-phenyl)-N-cyclopentyl-N-methy...)
Affinity DataKi:  3.30nMAssay Description:Binding affinity towards human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069292(CHEMBL156082 | N-ethyl-N-cyclopentyl-3-(4-hydrazon...)
Affinity DataKi:  4nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50071725((S)-3-(4-Aminomethyl-phenyl)-2-(anthracene-2-sulfo...)
Affinity DataKi:  5.70nMAssay Description:Binding affinity towards human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50071722((S)-3-(4-Aminomethyl-phenyl)-N-cyclopentyl-2-(6-me...)
Affinity DataKi:  6.60nMAssay Description:Binding affinity towards human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50070783((S)-3-(4-Carbamimidoyl-phenyl)-N-cyclopentyl-N-met...)
Affinity DataKi:  6.80nMAssay Description:Binding affinity towards human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069055((S)-3-(4-Aminomethyl-phenyl)-N-cyclopentyl-N-methy...)
Affinity DataKi:  9.60nMAssay Description:Binding affinity towards human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50071726((S)-3-(4-Aminomethyl-phenyl)-N-cyclopentyl-N-methy...)
Affinity DataKi:  10nMAssay Description:Binding affinity towards human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50071724((S)-3-(4-Aminomethyl-phenyl)-N-cyclopentyl-2-(5-di...)
Affinity DataKi:  11nMAssay Description:Binding affinity towards human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069053((S)-3-(4-Aminomethyl-phenyl)-N-cyclopentyl-N-methy...)
Affinity DataKi:  18nMAssay Description:Binding affinity towards human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50071721((S)-3-(4-Aminomethyl-phenyl)-2-(4-cyclohexyl-benze...)
Affinity DataKi:  20nMAssay Description:Binding affinity towards human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069293(CHEMBL440188 | N-methyl-N-n-butyl-3-(4-hydrazonofo...)
Affinity DataKi:  41nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50071728((S)-3-(4-Aminomethyl-phenyl)-2-(biphenyl-4-sulfony...)
Affinity DataKi:  61nMAssay Description:Binding affinity towards human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069296(CHEMBL347371 | N-(n-propyl)-N-cyclopentyl-3-(4-hyd...)
Affinity DataKi:  93nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50071727((S)-3-(4-Aminomethyl-phenyl)-N-cyclopentyl-N-methy...)
Affinity DataKi:  107nMAssay Description:Binding affinity towards human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069298(CHEMBL434678 | N-methyl-N-cyclohexyl-3-(4-hydrazon...)
Affinity DataKi:  152nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069299(CHEMBL155317 | N-(n-butyl)-N-cyclopentyl-3-(4-hydr...)
Affinity DataKi:  231nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069295(CHEMBL348175 | N-methyl-N-cyclopropyl-3-(4-hydrazo...)
Affinity DataKi:  247nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069300(CHEMBL350901 | N-hydroxy-N-cyclopentyl-3-(4-hydraz...)
Affinity DataKi:  367nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069294((S)-3-[4-(carbohydrazonamidol)-phenyl]-N-cyclopent...)
Affinity DataKi:  1.10E+3nMAssay Description:The compound was tested for inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069297(1-[3-[4-amino(amineimino)methylphenyl]-2-(2-naphth...)
Affinity DataKi:  1.47E+3nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069294((S)-3-[4-(carbohydrazonamidol)-phenyl]-N-cyclopent...)
Affinity DataKi:  3.29E+3nMAssay Description:Compound was tested for inhibitory activity against bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50071725((S)-3-(4-Aminomethyl-phenyl)-2-(anthracene-2-sulfo...)
Affinity DataKi:  3.30E+3nMAssay Description:Binding affinity of the compound towards bovine trypsin was evaluated in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50071721((S)-3-(4-Aminomethyl-phenyl)-2-(4-cyclohexyl-benze...)
Affinity DataKi:  4.80E+3nMAssay Description:Binding affinity of the compound towards bovine trypsin was evaluated in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50071723((S)-3-(4-Aminomethyl-phenyl)-N-cyclopentyl-N-methy...)
Affinity DataKi:  6.30E+3nMAssay Description:Binding affinity of the compound towards bovine trypsin was evaluated in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069301(CHEMBL155311 | N-hydroxyethyl-N-cyclopentyl-3-(4-h...)
Affinity DataKi:  7.04E+3nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069055((S)-3-(4-Aminomethyl-phenyl)-N-cyclopentyl-N-methy...)
Affinity DataKi:  9.04E+3nMAssay Description:Binding affinity of the compound towards bovine trypsin was evaluated in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50071726((S)-3-(4-Aminomethyl-phenyl)-N-cyclopentyl-N-methy...)
Affinity DataKi:  9.80E+3nMAssay Description:Binding affinity of the compound towards bovine trypsin was evaluated in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069053((S)-3-(4-Aminomethyl-phenyl)-N-cyclopentyl-N-methy...)
Affinity DataKi:  1.36E+4nMAssay Description:Binding affinity of the compound towards bovine trypsin was evaluated in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50071722((S)-3-(4-Aminomethyl-phenyl)-N-cyclopentyl-2-(6-me...)
Affinity DataKi:  1.42E+4nMAssay Description:Binding affinity of the compound towards bovine trypsin was evaluated in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50071724((S)-3-(4-Aminomethyl-phenyl)-N-cyclopentyl-2-(5-di...)
Affinity DataKi:  1.71E+4nMAssay Description:Binding affinity of the compound towards bovine trypsin was evaluated in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069294((S)-3-[4-(carbohydrazonamidol)-phenyl]-N-cyclopent...)
Affinity DataKi:  2.72E+4nMAssay Description:The compound was tested for inhibitory activity against tissue plasminogen activatorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069294((S)-3-[4-(carbohydrazonamidol)-phenyl]-N-cyclopent...)
Affinity DataKi:  4.79E+4nMAssay Description:The compound was tested for inhibitory activity against human plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
College Of Pharmacy Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50167706((S)-N-(4-amino-3,4-dioxo-1-phenylbutan-2-yl)-3-met...)
Affinity DataIC50:  70nMAssay Description:Inhibition of human erythrocytes mu-calpain using Suc-Leu-Tyr-AMC fluorogenic substrate after 30 mins by spectrofluorimeteryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
College Of Pharmacy Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50343071((S)-2-(3,4-dihydroxybenzylidene)-N-(4-(4-methoxyph...)
Affinity DataIC50:  130nMAssay Description:Inhibition of human erythrocytes mu-calpain using Suc-Leu-Tyr-AMC fluorogenic substrate after 30 mins by spectrofluorimeteryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
College Of Pharmacy Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50343074((S)-N-(4-(benzylamino)-3,4-dioxo-1-phenylbutan-2-y...)
Affinity DataIC50:  320nMAssay Description:Inhibition of human erythrocytes mu-calpain using Suc-Leu-Tyr-AMC fluorogenic substrate after 30 mins by spectrofluorimeteryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
College Of Pharmacy Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50343070((S)-N-(4-(benzylamino)-3,4-dioxo-1-phenylbutan-2-y...)
Affinity DataIC50:  360nMAssay Description:Inhibition of human erythrocytes mu-calpain using Suc-Leu-Tyr-AMC fluorogenic substrate after 30 mins by spectrofluorimeteryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
College Of Pharmacy Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50343069((S)-3-(2-(3,4-dihydroxybenzylidene)butanamido)-N-(...)
Affinity DataIC50:  460nMAssay Description:Inhibition of human erythrocytes mu-calpain using Suc-Leu-Tyr-AMC fluorogenic substrate after 30 mins by spectrofluorimeteryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
College Of Pharmacy Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50343073((S)-2-(3,4-dihydroxybenzylidene)-N-(4-(4-methoxyph...)
Affinity DataIC50:  500nMAssay Description:Inhibition of human erythrocytes mu-calpain using Suc-Leu-Tyr-AMC fluorogenic substrate after 30 mins by spectrofluorimeteryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
College Of Pharmacy Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50265975((S)-N-(4-amino-3,4-dioxo-1-phenylbutan-2-yl)-4-(2,...)
Affinity DataIC50:  520nMAssay Description:Inhibition of human erythrocytes mu-calpain using Suc-Leu-Tyr-AMC fluorogenic substrate after 30 mins by spectrofluorimeteryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
College Of Pharmacy Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50343068((S)-N-benzyl-3-(2-(3,4-dihydroxybenzylidene)butana...)
Affinity DataIC50:  610nMAssay Description:Inhibition of human erythrocytes mu-calpain using Suc-Leu-Tyr-AMC fluorogenic substrate after 30 mins by spectrofluorimeteryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
College Of Pharmacy Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50343075((S)-2-(4-hydroxy-3-methoxybenzylidene)-N-(4-(4-met...)
Affinity DataIC50:  630nMAssay Description:Inhibition of human erythrocytes mu-calpain using Suc-Leu-Tyr-AMC fluorogenic substrate after 30 mins by spectrofluorimeteryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
College Of Pharmacy Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50343072((S)-N-(4-(benzylamino)-3,4-dioxo-1-phenylbutan-2-y...)
Affinity DataIC50:  670nMAssay Description:Inhibition of human erythrocytes mu-calpain using Suc-Leu-Tyr-AMC fluorogenic substrate after 30 mins by spectrofluorimeteryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
College Of Pharmacy Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50343076((S)-2-(3,4-dimethoxybenzylidene)-N-(4-(4-methoxyph...)
Affinity DataIC50:  1.38E+3nMAssay Description:Inhibition of human erythrocytes mu-calpain using Suc-Leu-Tyr-AMC fluorogenic substrate after 30 mins by spectrofluorimeteryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
College Of Pharmacy Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50343067((S)-N-benzyl-3-(3-(3,4-dihydroxyphenyl)acrylamido)...)
Affinity DataIC50:  6.07E+3nMAssay Description:Inhibition of human erythrocytes mu-calpain using Suc-Leu-Tyr-AMC fluorogenic substrate after 30 mins by spectrofluorimeteryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50462013(CHEBI:8241 | Piplartine)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of STAT3 phosphorylation at Tyr705 residues in human DU145 cells after 24 hrs by Western blot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50462012(CHEMBL4227152)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of STAT3 (unknown origin) expressed in human HCT116 cells after 24 hrs by dual-luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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