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Found 45 with Last Name = 'zeltser' and Initial = 'i'
TargetNeuromedin-K receptor(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50030211((S)-2-{2-[(2R,5S,8R)-5,8-Dibenzyl-2-(3-guanidino-p...)
Affinity DataEC50: >1.00E+4nMAssay Description:Tested for the biological activity and selectivity against NK-3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50052525((S)-2-{2-[(2S,5R,8S)-5,8-Dibenzyl-2-(3-guanidino-p...)
Affinity DataEC50:  5nMAssay Description:Effective concentration to activate Tachykinin receptor 1 in guinea pig ileum(GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50030211((S)-2-{2-[(2R,5S,8R)-5,8-Dibenzyl-2-(3-guanidino-p...)
Affinity DataEC50: >5.00E+4nMAssay Description:Tested for the biological activity and selectivity against NK-2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50030212((S)-2-{2-[(2R,5S,8R)-5,8-Dibenzyl-2-(3-guanidino-p...)
Affinity DataEC50: >1.00E+4nMAssay Description:Tested for the biological activity and selectivity against NK-3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50030211((S)-2-{2-[(2R,5S,8R)-5,8-Dibenzyl-2-(3-guanidino-p...)
Affinity DataEC50:  5nMAssay Description:Tested for the biological activity and selectivity against NK-1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50030213((S)-2-{2-[(2R,5S,8R)-5,8-Dibenzyl-2-(3-guanidino-p...)
Affinity DataEC50: >5.00E+4nMAssay Description:Tested for the biological activity and selectivity against NK-2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50030212((S)-2-{2-[(2R,5S,8R)-5,8-Dibenzyl-2-(3-guanidino-p...)
Affinity DataEC50: >5.00E+4nMAssay Description:Tested for the biological activity and selectivity against NK-2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50030213((S)-2-{2-[(2R,5S,8R)-5,8-Dibenzyl-2-(3-guanidino-p...)
Affinity DataEC50:  11nMAssay Description:Tested for the biological activity and selectivity against NK-1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50030214((S)-2-{2-[(6R,9S,12R)-6,9-Dibenzyl-12-(3-guanidino...)
Affinity DataEC50: >1.00E+4nMAssay Description:Tested for the biological activity and selectivity against NK-3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50030213((S)-2-{2-[(2R,5S,8R)-5,8-Dibenzyl-2-(3-guanidino-p...)
Affinity DataEC50: >1.00E+4nMAssay Description:Tested for the biological activity and selectivity against NK-3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50030214((S)-2-{2-[(6R,9S,12R)-6,9-Dibenzyl-12-(3-guanidino...)
Affinity DataEC50: >1.00E+4nMAssay Description:Tested for the biological activity and selectivity against NK-1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50030214((S)-2-{2-[(6R,9S,12R)-6,9-Dibenzyl-12-(3-guanidino...)
Affinity DataEC50: >5.00E+4nMAssay Description:Tested for the biological activity and selectivity against NK-2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50052515((S)-2-{2-[(2S,5R,8S)-5,8-Dibenzyl-2-(3-guanidino-p...)
Affinity DataEC50:  11nMAssay Description:Effective concentration to activate Tachykinin receptor 1 in guinea pig ileum(GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50052516((S)-2-{2-[(3S,6R,9S)-3,6-Dibenzyl-9-(3-guanidino-p...)
Affinity DataEC50:  60nMAssay Description:Effective concentration to activate Tachykinin receptor 1 in guinea pig ileum(GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50052517((S)-2-{2-[(6S,9R,12S)-6,9-Dibenzyl-12-(3-guanidino...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 1 in guinea pig ileum(GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50052518((S)-2-{2-[(6S,9R,12S)-6,9-Dibenzyl-12-(3-guanidino...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 3 in rat portal vein (RPV)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50052519(CHEMBL265115 | Hexanedioic acid (1-{1-[1-((3-acety...)
Affinity DataEC50: >1.00E+5nMAssay Description:Effective concentration to activate Tachykinin receptor 2 in rat vas deferens(RVD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50052520((S)-2-{2-[(3S,6R,9S)-3,6-Dibenzyl-9-(3-guanidino-p...)
Affinity DataEC50:  1.00E+3nMAssay Description:Effective concentration to activate Tachykinin receptor 3 in rat portal vein (RPV)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50052518((S)-2-{2-[(6S,9R,12S)-6,9-Dibenzyl-12-(3-guanidino...)
Affinity DataEC50:  4.00E+3nMAssay Description:Effective concentration to activate Tachykinin receptor 1 in guinea pig ileum(GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50052519(CHEMBL265115 | Hexanedioic acid (1-{1-[1-((3-acety...)
Affinity DataEC50:  2.00E+3nMAssay Description:Effective concentration to activate Tachykinin receptor 3 in rat portal vein(RPV).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50052521((S)-2-{2-[{(S)-2-[(S)-2-((S)-2-Acetylamino-5-guani...)
Affinity DataEC50:  2.00E+3nMAssay Description:Effective concentration to activate Tachykinin receptor 3 in rat portal vein (RPV)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50052522((S)-2-{2-[(2S,5R,8S)-5,8-Dibenzyl-2-(3-guanidino-p...)
Affinity DataEC50: >5.00E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 2 in rat vas deferens (RVD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50052524((S)-N-((S)-1-{[(S)-1-({[(S)-1-((S)-1-Carbamoyl-3-m...)
Affinity DataEC50:  3.50E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 1 in guinea pig ileum(GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50052523((R)-1-{(S)-2-[(S)-2-((S)-2-Acetylamino-5-guanidino...)
Affinity DataEC50: >5.00E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 3 in rat portal vein(RPV).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50052516((S)-2-{2-[(3S,6R,9S)-3,6-Dibenzyl-9-(3-guanidino-p...)
Affinity DataEC50: >5.00E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 2 in rat vas deferens (RVD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50052522((S)-2-{2-[(2S,5R,8S)-5,8-Dibenzyl-2-(3-guanidino-p...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 3 in rat portal vein (RPV)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50052519(CHEMBL265115 | Hexanedioic acid (1-{1-[1-((3-acety...)
Affinity DataEC50:  400nMAssay Description:Effective concentration to activate Tachykinin receptor 1 in guinea pig ileum(GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50052525((S)-2-{2-[(2S,5R,8S)-5,8-Dibenzyl-2-(3-guanidino-p...)
Affinity DataEC50: >5.00E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 2 in rat vas deferens (RVD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50052523((R)-1-{(S)-2-[(S)-2-((S)-2-Acetylamino-5-guanidino...)
Affinity DataEC50: >2.00E+5nMAssay Description:Effective concentration to activate Tachykinin receptor 2 in rat vas deferens (RVD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50052524((S)-N-((S)-1-{[(S)-1-({[(S)-1-((S)-1-Carbamoyl-3-m...)
Affinity DataEC50: >2.00E+5nMAssay Description:Effective concentration to activate Tachykinin receptor 2 in rat vas deferens (RVD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50052524((S)-N-((S)-1-{[(S)-1-({[(S)-1-((S)-1-Carbamoyl-3-m...)
Affinity DataEC50:  0.5nMAssay Description:Effective concentration to activate Tachykinin receptor 3 in rat portal vein (RPV)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50052523((R)-1-{(S)-2-[(S)-2-((S)-2-Acetylamino-5-guanidino...)
Affinity DataEC50:  3nMAssay Description:Effective concentration to activate Tachykinin receptor 1 in guinea pig ileum(GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50052520((S)-2-{2-[(3S,6R,9S)-3,6-Dibenzyl-9-(3-guanidino-p...)
Affinity DataEC50:  160nMAssay Description:Effective concentration to activate Tachykinin receptor 1 in guinea pig ileum(GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50052517((S)-2-{2-[(6S,9R,12S)-6,9-Dibenzyl-12-(3-guanidino...)
Affinity DataEC50: >5.00E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 2 in rat vas deferens (RVD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50052521((S)-2-{2-[{(S)-2-[(S)-2-((S)-2-Acetylamino-5-guani...)
Affinity DataEC50:  300nMAssay Description:Effective concentration to activate Tachykinin receptor 1 in guinea pig ileum(GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50052518((S)-2-{2-[(6S,9R,12S)-6,9-Dibenzyl-12-(3-guanidino...)
Affinity DataEC50: >5.00E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 2 in rat vas deferens (RVD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50052521((S)-2-{2-[{(S)-2-[(S)-2-((S)-2-Acetylamino-5-guani...)
Affinity DataEC50: >1.00E+5nMAssay Description:Effective concentration to activate Tachykinin receptor 2 in rat vas deferens (RVD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50052517((S)-2-{2-[(6S,9R,12S)-6,9-Dibenzyl-12-(3-guanidino...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 3 in rat portal vein (RPV)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50052525((S)-2-{2-[(2S,5R,8S)-5,8-Dibenzyl-2-(3-guanidino-p...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 3 in rat portal vein (RPV)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50052515((S)-2-{2-[(2S,5R,8S)-5,8-Dibenzyl-2-(3-guanidino-p...)
Affinity DataEC50: >5.00E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 2 in rat vas deferens (RVD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50052515((S)-2-{2-[(2S,5R,8S)-5,8-Dibenzyl-2-(3-guanidino-p...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 3 in rat portal vein (RPV)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50052522((S)-2-{2-[(2S,5R,8S)-5,8-Dibenzyl-2-(3-guanidino-p...)
Affinity DataEC50:  180nMAssay Description:Effective concentration to activate Tachykinin receptor 1 in guinea pig ileum(GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50052520((S)-2-{2-[(3S,6R,9S)-3,6-Dibenzyl-9-(3-guanidino-p...)
Affinity DataEC50: >5.00E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 2 in rat vas deferens (RVD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50052516((S)-2-{2-[(3S,6R,9S)-3,6-Dibenzyl-9-(3-guanidino-p...)
Affinity DataEC50:  1.00E+3nMAssay Description:Effective concentration to activate Tachykinin receptor 3 in rat portal vein (RPV)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50030212((S)-2-{2-[(2R,5S,8R)-5,8-Dibenzyl-2-(3-guanidino-p...)
Affinity DataEC50:  180nMAssay Description:Tested for the biological activity and selectivity against NK-1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed