Affinity DataKi: 0.00500nMAssay Description:Inhibition against Opioid receptor mu 1 using [3H]- DAMGO radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 0.0600nMAssay Description:Inhibition against Opioid receptor mu 1 using [3H]- DAMGO radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 0.0800nMAssay Description:Inhibition against Opioid receptor mu 1 using [3H]- DAMGO radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 0.130nMAssay Description:Inhibition against Opioid receptor mu 1 using [3H]- DAMGO radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 0.150nMAssay Description:Inhibition against Opioid receptor mu 1 using [3H]- DAMGO radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 0.150nMAssay Description:Inhibition against Opioid receptor mu 1 using [3H]- DAMGO radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 2.89nMAssay Description:Inhibition against Opioid receptor mu 1 using [3H]- DAMGO radioligand.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 3.10nMAssay Description:Displacement of bound [3H]-diprenorphine in cloned rat Opioid receptor kappa 1 expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 5.70nMAssay Description:Displacement of bound [3H]-diprenorphine in cloned rat Opioid receptor kappa 1 expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.85nMAssay Description:Inhibition against Opioid receptor mu 1 using [3H]- DAMGO radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 114nMAssay Description:Inhibition against delta-opioid receptor using [3H]-DPDPE radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 150nMAssay Description:Inhibition against Opioid receptor delta 1 using [3H]-DPDPE radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Inhibition against delta-opioid receptor using [3H]-DPDPE radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 230nMAssay Description:Inhibition against delta-opioid receptor using [3H]-DPDPE radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 230nMAssay Description:Inhibition against delta-opioid receptor using [3H]-DPDPE radioligand.More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition against delta-opioid receptor using [3H]-DPDPE radioligand.More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition against delta-opioid receptor using [3H]-DPDPE radioligand.More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition against delta-opioid receptor using [3H]-DPDPE radioligand.More data for this Ligand-Target Pair