TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Cardiome Pharma
Curated by ChEMBL
Cardiome Pharma
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human potassium channel Kv1.5 by patch-clamp methodMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily D member 2(Rattus norvegicus)
Cardiome Pharma
Curated by ChEMBL
Cardiome Pharma
Curated by ChEMBL
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of rat potassium channel Kv4.2 by patch-clamp methodMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily B member 1(Rattus norvegicus)
Cardiome Pharma
Curated by ChEMBL
Cardiome Pharma
Curated by ChEMBL
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of rat potassium channel Kv2.1 by patch-clamp methodMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily B member 1(Rattus norvegicus)
Cardiome Pharma
Curated by ChEMBL
Cardiome Pharma
Curated by ChEMBL
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of rat potassium channel Kv2.1 by patch-clamp methodMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Cardiome Pharma
Curated by ChEMBL
Cardiome Pharma
Curated by ChEMBL
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of human potassium channel Kv1.5 by patch-clamp methodMore data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Cardiome Pharma
Curated by ChEMBL
Cardiome Pharma
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of human heart sodium channel Nav1.5 by patch-clamp methodMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Cardiome Pharma
Curated by ChEMBL
Cardiome Pharma
Curated by ChEMBL
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of human potassium channel Kv1.5 by patch-clamp methodMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Cardiome Pharma
Curated by ChEMBL
Cardiome Pharma
Curated by ChEMBL
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of human potassium channel Kv1.5 by patch-clamp methodMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily B member 1(Rattus norvegicus)
Cardiome Pharma
Curated by ChEMBL
Cardiome Pharma
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of rat potassium channel Kv2.1 by patch-clamp methodMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily B member 1(Rattus norvegicus)
Cardiome Pharma
Curated by ChEMBL
Cardiome Pharma
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of rat potassium channel Kv2.1 by patch-clamp methodMore data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Cardiome Pharma
Curated by ChEMBL
Cardiome Pharma
Curated by ChEMBL
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibition of human heart sodium channel Nav1.5 by patch-clamp methodMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Cardiome Pharma
Curated by ChEMBL
Cardiome Pharma
Curated by ChEMBL
Affinity DataIC50: 7.70E+3nMAssay Description:Inhibition of human potassium channel Kv1.5 by patch-clamp methodMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily B member 1(Rattus norvegicus)
Cardiome Pharma
Curated by ChEMBL
Cardiome Pharma
Curated by ChEMBL
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of rat potassium channel Kv2.1 by patch-clamp methodMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily D member 2(Rattus norvegicus)
Cardiome Pharma
Curated by ChEMBL
Cardiome Pharma
Curated by ChEMBL
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of rat potassium channel Kv4.2 by patch-clamp methodMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily D member 2(Rattus norvegicus)
Cardiome Pharma
Curated by ChEMBL
Cardiome Pharma
Curated by ChEMBL
Affinity DataIC50: 1.01E+4nMAssay Description:Inhibition of rat potassium channel Kv4.2 by patch-clamp methodMore data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Cardiome Pharma
Curated by ChEMBL
Cardiome Pharma
Curated by ChEMBL
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of human heart sodium channel Nav1.5 by patch-clamp methodMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily D member 2(Rattus norvegicus)
Cardiome Pharma
Curated by ChEMBL
Cardiome Pharma
Curated by ChEMBL
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of rat potassium channel Kv4.2 by patch-clamp methodMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily D member 2(Rattus norvegicus)
Cardiome Pharma
Curated by ChEMBL
Cardiome Pharma
Curated by ChEMBL
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of rat potassium channel Kv4.2 by patch-clamp methodMore data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Cardiome Pharma
Curated by ChEMBL
Cardiome Pharma
Curated by ChEMBL
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of human heart sodium channel Nav1.5 by patch-clamp methodMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily D member 2(Rattus norvegicus)
Cardiome Pharma
Curated by ChEMBL
Cardiome Pharma
Curated by ChEMBL
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of rat potassium channel Kv4.2 by patch-clamp methodMore data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Cardiome Pharma
Curated by ChEMBL
Cardiome Pharma
Curated by ChEMBL
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of human heart sodium channel Nav1.5 by patch-clamp methodMore data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Cardiome Pharma
Curated by ChEMBL
Cardiome Pharma
Curated by ChEMBL
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of human heart sodium channel Nav1.5 by patch-clamp methodMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily D member 2(Rattus norvegicus)
Cardiome Pharma
Curated by ChEMBL
Cardiome Pharma
Curated by ChEMBL
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of rat potassium channel Kv4.2 by patch-clamp methodMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Cardiome Pharma
Curated by ChEMBL
Cardiome Pharma
Curated by ChEMBL
Affinity DataIC50: 5.10E+4nMAssay Description:Inhibition of human potassium channel Kv1.5 by patch-clamp methodMore data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Cardiome Pharma
Curated by ChEMBL
Cardiome Pharma
Curated by ChEMBL
Affinity DataIC50: 1.08E+5nMAssay Description:Inhibition of human heart sodium channel Nav1.5 by patch-clamp methodMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily D member 2(Rattus norvegicus)
Cardiome Pharma
Curated by ChEMBL
Cardiome Pharma
Curated by ChEMBL
Affinity DataIC50: 1.21E+6nMAssay Description:Inhibition of rat potassium channel Kv4.2 by patch-clamp methodMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Cardiome Pharma
Curated by ChEMBL
Cardiome Pharma
Curated by ChEMBL
Affinity DataIC50: 2.19E+6nMAssay Description:Inhibition of human potassium channel Kv1.5 by patch-clamp methodMore data for this Ligand-Target Pair