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Found 34 with Last Name = 'van de stolpe' and Initial = 'ac'
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50039676(4-Fluorosulfonyl-benzoic acid 3-(8-cyclopentyl-2,6...)
Affinity DataKi:  12nMAssay Description:Binding affinity towards rat Adenosine A1 receptor using [3H]-DPCPXMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM25400((2R,3R,4S,5R)-2-[6-(cyclopentylamino)-9H-purin-9-y...)
Affinity DataKi:  230nMAssay Description:Binding affinity towards rat Adenosine A1 receptor using [3H]-DPCPXMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50167783(CHEMBL196885 | Decanoic acid {1-[3-(4-cyano-phenyl...)
Affinity DataIC50:  930nMAssay Description:Inhibitory concentration against CX3C chemokine receptor 3 expressed in human HEK-293 cells using [125I]-CXCL10 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50167781(CHEMBL193448 | Decanoic acid (2-dimethylamino-ethy...)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibitory concentration against CX3C chemokine receptor 3 expressed in human HEK-293 cells using [125I]-CXCL10 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50167778(CHEMBL194494 | Decanoic acid (2-dimethylamino-ethy...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibitory concentration against CX3C chemokine receptor 3 expressed in human HEK-293 cells using [125I]-CXCL10 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50167782(CHEMBL383346 | Decanoic acid (2-dimethylamino-ethy...)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibitory concentration against CX3C chemokine receptor 3 expressed in human HEK-293 cells using [125I]-CXCL10 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50167784(CHEMBL197368 | Decanoic acid {1-[3-(3-cyano-phenyl...)
Affinity DataIC50:  5.80E+3nMAssay Description:Inhibitory concentration against CX3C chemokine receptor 3 expressed in human HEK-293 cells using [125I]-CXCL10 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50167780(CHEMBL370482 | Decanoic acid {1-[3-(2-cyano-phenyl...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory concentration against CX3C chemokine receptor 3 expressed in human HEK-293 cells using [125I]-CXCL10 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50167785(CHEMBL196248 | Decanoic acid (2-dimethylamino-ethy...)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibitory concentration against CX3C chemokine receptor 3 expressed in human HEK-293 cells using [125I]-CXCL10 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50167779(CHEMBL371577 | Decanoic acid (2-dimethylamino-ethy...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against CX3C chemokine receptor 3 expressed in human HEK-293 cells using [125I]-CXCL10 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50167786(CHEMBL371154 | Decanoic acid (2-dimethylamino-ethy...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against CX3C chemokine receptor 3 expressed in human HEK-293 cells using [125I]-CXCL10 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50064081(6-Bromo-2-[3-(naphthalen-2-ylmethoxy)-phenyl]-4-ox...)
Affinity DataKd:  1.13E+3nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50064071(4-Oxo-2-[4-(quinolin-2-ylmethoxy)-phenyl]-4H-chrom...)
Affinity DataKd:  526nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50064065(2-(4-Benzyloxy-phenyl)-4-oxo-4H-chromene-8-carboxy...)
Affinity DataKd:  5.50E+4nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50064076(6-bromo-4-oxo-N-(phenylsulfonyl)-2-(4-(quinolin-2-...)
Affinity DataKd:  382nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50064080(2-[3-((E)-2-Quinolin-2-yl-vinyl)-phenyl]-6-(1H-tet...)
Affinity DataKd:  307nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50064070(6-Bromo-2-[3-(1-methyl-1H-benzoimidazol-2-ylmethox...)
Affinity DataKd:  210nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50064078(6-Bromo-2-[3-(7-chloro-quinolin-2-ylmethoxy)-pheny...)
Affinity DataKd:  12nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50064066(2-[3-(Benzothiazol-2-ylmethoxy)-phenyl]-6-bromo-4-...)
Affinity DataKd:  79nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50064077(4-Oxo-2-[4-((E)-2-quinolin-2-yl-vinyl)-phenyl]-4H-...)
Affinity DataKd:  270nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50064075(6-Fluoro-4-oxo-2-[3-((E)-2-quinolin-2-yl-vinyl)-ph...)
Affinity DataKd:  127nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50064067(6-Bromo-4-oxo-2-[4-(quinolin-2-ylmethoxy)-phenyl]-...)
Affinity DataKd:  504nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50064072(4-Oxo-2-[3-(quinolin-2-ylmethoxy)-phenyl]-4H-chrom...)
Affinity DataKd:  17nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50064063(6-Chloro-2-[3-((E)-2-quinolin-2-yl-vinyl)-phenyl]-...)
Affinity DataKd:  1.10E+4nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50064062(6-Chloro-4-oxo-2-[3-((E)-2-quinolin-2-yl-vinyl)-ph...)
Affinity DataKd:  11nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50064068(6-Bromo-4-oxo-2-[3-((E)-2-quinolin-2-yl-vinyl)-phe...)
Affinity DataKd:  17nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50064073(4-Oxo-2-[3-((E)-2-quinolin-2-yl-vinyl)-phenyl]-4H-...)
Affinity DataKd:  1.73E+3nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50064064(6-Bromo-4-oxo-2-[3-(quinolin-2-ylmethoxy)-phenyl]-...)
Affinity DataKd:  31nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50064082(4-Oxo-2-[3-((E)-2-quinolin-2-yl-vinyl)-phenyl]-4H-...)
Affinity DataKd:  1.75E+3nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50064074(4-Oxo-2-[3-((E)-2-quinolin-2-yl-vinyl)-phenyl]-4H-...)
Affinity DataKd:  17nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50064079(4-Oxo-2-[3-((E)-2-quinolin-2-yl-vinyl)-phenyl]-4H-...)
Affinity DataKd:  408nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50064061(6-Bromo-4-oxo-2-[3-(quinazolin-2-ylmethoxy)-phenyl...)
Affinity DataKd:  101nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50064060(6-Methyl-4-oxo-2-[3-((E)-2-quinolin-2-yl-vinyl)-ph...)
Affinity DataKd:  13nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50064069(4-Oxo-2-[4-(quinazolin-2-ylmethoxy)-phenyl]-4H-chr...)
Affinity DataKd:  1.10E+3nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed