Affinity DataKi: 12nMAssay Description:Binding affinity towards rat Adenosine A1 receptor using [3H]-DPCPXMore data for this Ligand-Target Pair
Affinity DataKi: 230nMAssay Description:Binding affinity towards rat Adenosine A1 receptor using [3H]-DPCPXMore data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Vrije Universiteit Amsterdam
Curated by ChEMBL
Vrije Universiteit Amsterdam
Curated by ChEMBL
Affinity DataIC50: 930nMAssay Description:Inhibitory concentration against CX3C chemokine receptor 3 expressed in human HEK-293 cells using [125I]-CXCL10 as radioligandMore data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Vrije Universiteit Amsterdam
Curated by ChEMBL
Vrije Universiteit Amsterdam
Curated by ChEMBL
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibitory concentration against CX3C chemokine receptor 3 expressed in human HEK-293 cells using [125I]-CXCL10 as radioligandMore data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Vrije Universiteit Amsterdam
Curated by ChEMBL
Vrije Universiteit Amsterdam
Curated by ChEMBL
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibitory concentration against CX3C chemokine receptor 3 expressed in human HEK-293 cells using [125I]-CXCL10 as radioligandMore data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Vrije Universiteit Amsterdam
Curated by ChEMBL
Vrije Universiteit Amsterdam
Curated by ChEMBL
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibitory concentration against CX3C chemokine receptor 3 expressed in human HEK-293 cells using [125I]-CXCL10 as radioligandMore data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Vrije Universiteit Amsterdam
Curated by ChEMBL
Vrije Universiteit Amsterdam
Curated by ChEMBL
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibitory concentration against CX3C chemokine receptor 3 expressed in human HEK-293 cells using [125I]-CXCL10 as radioligandMore data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Vrije Universiteit Amsterdam
Curated by ChEMBL
Vrije Universiteit Amsterdam
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against CX3C chemokine receptor 3 expressed in human HEK-293 cells using [125I]-CXCL10 as radioligandMore data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Vrije Universiteit Amsterdam
Curated by ChEMBL
Vrije Universiteit Amsterdam
Curated by ChEMBL
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibitory concentration against CX3C chemokine receptor 3 expressed in human HEK-293 cells using [125I]-CXCL10 as radioligandMore data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Vrije Universiteit Amsterdam
Curated by ChEMBL
Vrije Universiteit Amsterdam
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against CX3C chemokine receptor 3 expressed in human HEK-293 cells using [125I]-CXCL10 as radioligandMore data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Vrije Universiteit Amsterdam
Curated by ChEMBL
Vrije Universiteit Amsterdam
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against CX3C chemokine receptor 3 expressed in human HEK-293 cells using [125I]-CXCL10 as radioligandMore data for this Ligand-Target Pair
Affinity DataKd: 1.13E+3nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
Affinity DataKd: 526nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
Affinity DataKd: 5.50E+4nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
Affinity DataKd: 382nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
Affinity DataKd: 307nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
Affinity DataKd: 210nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
Affinity DataKd: 12nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
Affinity DataKd: 79nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
Affinity DataKd: 270nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
Affinity DataKd: 127nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
Affinity DataKd: 504nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
Affinity DataKd: 17nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
Affinity DataKd: 1.10E+4nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
Affinity DataKd: 11nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
Affinity DataKd: 17nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
Affinity DataKd: 1.73E+3nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
Affinity DataKd: 31nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
Affinity DataKd: 1.75E+3nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
Affinity DataKd: 17nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
Affinity DataKd: 408nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
Affinity DataKd: 101nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
Affinity DataKd: 13nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair
Affinity DataKd: 1.10E+3nMAssay Description:In vitro affinity for CysLT1 receptors on guinea pig lung membranes, measured by displacement of [3H]-LTD4.More data for this Ligand-Target Pair