Affinity DataIC50: 2.40nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca
Curated by ChEMBL
Astrazeneca
Curated by ChEMBL
Affinity DataIC50: 2.51nMAssay Description:Displacement of [3H]dofetilide from human recombinant ERG expressed in HEK293 cells by patch clamp methodMore data for this Ligand-Target Pair
Affinity DataIC50: 2.63nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
Affinity DataIC50: 2.63nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
Affinity DataIC50: 2.82nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
Affinity DataIC50: 4.90nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
Affinity DataIC50: 5.62nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca
Curated by ChEMBL
Astrazeneca
Curated by ChEMBL
Affinity DataIC50: 6.46nMAssay Description:Displacement of [3H]dofetilide from human recombinant ERG expressed in HEK293 cells by patch clamp methodMore data for this Ligand-Target Pair
Affinity DataIC50: 6.61nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
Affinity DataIC50: 8.13nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
Affinity DataIC50: 11.5nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
Affinity DataIC50: 14.8nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
Affinity DataIC50: 17.4nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
Affinity DataIC50: 19.1nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
Affinity DataIC50: 22.4nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
Affinity DataIC50: 22.4nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
Affinity DataIC50: 27.5nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
Affinity DataIC50: 29nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca
Curated by ChEMBL
Astrazeneca
Curated by ChEMBL
Affinity DataIC50: 30.2nMAssay Description:Displacement of [3H]dofetilide from human recombinant ERG expressed in HEK293 cells by patch clamp methodMore data for this Ligand-Target Pair
Affinity DataIC50: 30.9nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
Affinity DataIC50: 32.4nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
Affinity DataIC50: 34.7nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca
Curated by ChEMBL
Astrazeneca
Curated by ChEMBL
Affinity DataIC50: 45.7nMAssay Description:Inhibition of wild type human ERG expressed in CHOK1 cells by whole-cell plate-based electrophysiologyMore data for this Ligand-Target Pair
Affinity DataIC50: 55.0nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca
Curated by ChEMBL
Astrazeneca
Curated by ChEMBL
Affinity DataIC50: 70.8nMAssay Description:Inhibition of wild type human ERG expressed in CHOK1 cells by whole-cell plate-based electrophysiologyMore data for this Ligand-Target Pair