Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 15 hits for monomerid = 50017893,50444525,50444526,50444527,50444528,50017893,50444525,50444526,50444527,50444528   

TargetSuppressor of tumorigenicity 14 protein(Human)
Aurigene Discovery Technologies

Curated by ChEMBL
LigandPNGBDBM50444526(CHEMBL3099812)
Affinity DataKi:  40nMAssay Description:Inhibition of matriptase-SP1 (615 to 855) (unknown origin) expressed in Escherichia coli BL21(DE3) using Boc-Gln-Ala-Arg-7-amido-4-methyl coumarin hy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSuppressor of tumorigenicity 14 protein(Human)
Aurigene Discovery Technologies

Curated by ChEMBL
LigandPNGBDBM50444525(CHEMBL3099813)
Affinity DataKi:  200nMAssay Description:Inhibition of matriptase-SP1 (615 to 855) (unknown origin) expressed in Escherichia coli BL21(DE3) using Boc-Gln-Ala-Arg-7-amido-4-methyl coumarin hy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Aurigene Discovery Technologies

Curated by ChEMBL
LigandPNGBDBM50444528(CHEMBL3099589)
Affinity DataKi:  200nMAssay Description:Inhibition of matriptase-SP1 (615 to 855) (unknown origin) expressed in Escherichia coli BL21(DE3) using Boc-Gln-Ala-Arg-7-amido-4-methyl coumarin hy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCoagulation factor X(Human)
Aurigene Discovery Technologies

Curated by ChEMBL
LigandPNGBDBM50444528(CHEMBL3099589)
Affinity DataKi:  300nMAssay Description:Inhibition of factor 10a (unknown origin) using CH3OCO-D-CHA-Gly-Arg-pNA.AcoH as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Aurigene Discovery Technologies

Curated by ChEMBL
LigandPNGBDBM50444526(CHEMBL3099812)
Affinity DataKi:  300nMAssay Description:Inhibition of factor 10a (unknown origin) using CH3OCO-D-CHA-Gly-Arg-pNA.AcoH as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetCoagulation factor X(Bovine)
Aurigene Discovery Technologies

Curated by ChEMBL
LigandPNGBDBM50017893(CHEMBL3289036)
Affinity DataKi:  1.16E+3nMAssay Description:Inhibition of bovine plasma factor 10a using CH3OCO-D-CHA-Gly-Arg-pNA.AcoH substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Aurigene Discovery Technologies

Curated by ChEMBL
LigandPNGBDBM50444527(CHEMBL3099811)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of matriptase-SP1 (615 to 855) (unknown origin) expressed in Escherichia coli BL21(DE3) using Boc-Gln-Ala-Arg-7-amido-4-methyl coumarin hy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
Aurigene Discovery Technologies

Curated by ChEMBL
LigandPNGBDBM50017893(CHEMBL3289036)
Affinity DataKi:  1.98E+3nMAssay Description:Inhibition of recombinant matriptase (unknown origin) using Boc-Gln-Ala-Arg-7-amido-4-methyl coumarin hydrobromideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetProthrombin(Human)
Aurigene Discovery Technologies

Curated by ChEMBL
LigandPNGBDBM50444528(CHEMBL3099589)
Affinity DataKi:  4.10E+3nMAssay Description:Inhibition of thrombin (unknown origin) by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetProthrombin(Human)
Aurigene Discovery Technologies

Curated by ChEMBL
LigandPNGBDBM50017893(CHEMBL3289036)
Affinity DataKi:  4.85E+3nMAssay Description:Inhibition of human thrombin using Boc-Gln-Ala-Arg-7-amido-4-methyl coumarin hydrobromideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetProthrombin(Human)
Aurigene Discovery Technologies

Curated by ChEMBL
LigandPNGBDBM50444526(CHEMBL3099812)
Affinity DataKi:  5.80E+3nMAssay Description:Inhibition of thrombin (unknown origin) by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Aurigene Discovery Technologies

Curated by ChEMBL
LigandPNGBDBM50444527(CHEMBL3099811)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of uPA (unknown origin) using L-PyroGlu-Gly-Arg-pNA.HCl as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Aurigene Discovery Technologies

Curated by ChEMBL
LigandPNGBDBM50444525(CHEMBL3099813)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of uPA (unknown origin) using L-PyroGlu-Gly-Arg-pNA.HCl as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Aurigene Discovery Technologies

Curated by ChEMBL
LigandPNGBDBM50444526(CHEMBL3099812)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of uPA (unknown origin) using L-PyroGlu-Gly-Arg-pNA.HCl as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Aurigene Discovery Technologies

Curated by ChEMBL
LigandPNGBDBM50444528(CHEMBL3099589)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of uPA (unknown origin) using L-PyroGlu-Gly-Arg-pNA.HCl as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed