Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50071108,50432489,50432490,50432491,50432492,50432493,50071108,50432489,50432490,50432491,50432492,50432493   

TargetBromodomain-containing protein 4(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50432490(CHEMBL2349344)Copy SMILESCopy InChI

Affinity DataIC50: 2.38E+4nMAssay Description:Displacement of FITC-labeled (+)-JQ1 from bromodomain BRD4(1) (unknown origin) expressed in Escherichia coli BL21(DE3) after 4 hrs by fluorescence an...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
9/24/2013
Entry Details Article
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TargetBromodomain-containing protein 4(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50432493(CHEMBL2349341)Copy SMILESCopy InChI

Affinity DataIC50: 2.40E+4nMAssay Description:Displacement of FITC-labeled (+)-JQ1 from bromodomain BRD4(1) (unknown origin) expressed in Escherichia coli BL21(DE3) after 4 hrs by fluorescence an...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPurchaseCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
9/24/2013
Entry Details Article
Copy BDB DOIPubMed
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TargetBromodomain-containing protein 4(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50432492(CHEMBL2349342)Copy SMILESCopy InChI

Affinity DataIC50: 4.20E+4nMAssay Description:Displacement of FITC-labeled (+)-JQ1 from bromodomain BRD4(1) (unknown origin) expressed in Escherichia coli BL21(DE3) after 4 hrs by fluorescence an...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPurchaseCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
9/24/2013
Entry Details Article
Copy BDB DOIPubMed
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TargetBromodomain-containing protein 4(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50432489(CHEMBL2349345)Copy SMILESCopy InChI

Affinity DataIC50: 5.07E+4nMAssay Description:Displacement of FITC-labeled (+)-JQ1 from bromodomain BRD4(1) (unknown origin) expressed in Escherichia coli BL21(DE3) after 4 hrs by fluorescence an...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
9/24/2013
Entry Details Article
Copy BDB DOIPubMed
Copy reaction URL

TargetBromodomain-containing protein 4(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50432491(CHEMBL2349343)Copy SMILESCopy InChI

Affinity DataIC50: 5.10E+4nMAssay Description:Displacement of FITC-labeled (+)-JQ1 from bromodomain BRD4(1) (unknown origin) expressed in Escherichia coli BL21(DE3) after 4 hrs by fluorescence an...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPurchaseCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
9/24/2013
Entry Details Article
Copy BDB DOIPubMed
Copy reaction URL

TargetBromodomain-containing protein 4(Human)
Chinese Academy of Sciences

Curated by ChEMBL

LigandBDBM50071108(CHEMBL3409981)Copy SMILESCopy InChI

Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of BRD4(1) (unknown origin) incubated for 4 hrs by (+)-JQ1 fluorescent ligand based fluorescence anisotrophyMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPurchaseCHEMBLPC cidPC sidPDBSimilars

In Depth
Date in BDB:
4/21/2016
Entry Details Article
Copy BDB DOIPubMed
Copy reaction URL