Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50237233,50400040,50400041,50400042,50400043,50237233,50400040,50400041,50400042,50400043   

TargetTyrosine-protein kinase SYK(Human)
Second Military Medical University

Curated by ChEMBL

LigandBDBM50237233(CHEMBL4104392)Copy SMILESCopy InChI

Affinity DataIC50: 47nMAssay Description:Inhibition of SYK (unknown origin) using FAM-labeled peptide as substrate preincubated for 10 mins followed by substrate addition measured after 25 m...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidPDBSimilars

In Depth
Date in BDB:
8/12/2019
Entry Details Article
Copy BDB DOIPubMedPDB3D Structure (crystal)
Copy reaction URL

TargetTyrosine-protein kinase SYK(Human)
Second Military Medical University

Curated by ChEMBL

LigandBDBM50400040(CHEMBL2177730)Copy SMILESCopy InChI

Affinity DataIC50: 47nMAssay Description:Inhibition of human recombinant spleen tyrosine kinase (360 to 635 amino acid residues) after 10 mins by scintillation counting analysisMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidPDBSimilars

In Depth
Date in BDB:
5/17/2013
Entry Details Article
Copy BDB DOIPubMedPDB3D Structure (crystal)
Copy reaction URL

TargetTyrosine-protein kinase SYK(Human)
Second Military Medical University

Curated by ChEMBL

LigandBDBM50400043(CHEMBL2177727)Copy SMILESCopy InChI

Affinity DataIC50: 50nMAssay Description:Inhibition of human recombinant spleen tyrosine kinase (360 to 635 amino acid residues) after 10 mins by scintillation counting analysisMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
5/17/2013
Entry Details Article
Copy BDB DOIPubMed
Copy reaction URL

TargetTyrosine-protein kinase SYK(Human)
Second Military Medical University

Curated by ChEMBL

LigandBDBM50400042(CHEMBL2177728)Copy SMILESCopy InChI

Affinity DataIC50: 93nMAssay Description:Inhibition of human recombinant spleen tyrosine kinase (360 to 635 amino acid residues) after 10 mins by scintillation counting analysisMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
5/17/2013
Entry Details Article
Copy BDB DOIPubMed
Copy reaction URL

TargetTyrosine-protein kinase SYK(Human)
Second Military Medical University

Curated by ChEMBL

LigandBDBM50400041(CHEMBL2177729)Copy SMILESCopy InChI

Affinity DataIC50: 423nMAssay Description:Inhibition of human recombinant spleen tyrosine kinase (360 to 635 amino acid residues) after 10 mins by scintillation counting analysisMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
5/17/2013
Entry Details Article
Copy BDB DOIPubMed
Copy reaction URL