Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 14 hits for monomerid = 50295045,50295046,50295047,50295048,50295049,50295045,50295046,50295047,50295048,50295049   

TargetPeroxisome proliferator-activated receptor gamma(Human)
Wake Forest University

Curated by ChEMBL
LigandPNGBDBM50295045((9Z,12E)-12-nitrooctadeca-9,12-dienoic acid | CHEM...)
Affinity DataEC50:  45nMAssay Description:Activation of PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Wake Forest University

Curated by ChEMBL
LigandPNGBDBM50295045((9Z,12E)-12-nitrooctadeca-9,12-dienoic acid | CHEM...)
Affinity DataEC50:  70nMAssay Description:Activation of human PPAR-gamma-dependent transcription expressed in human MCF7 cells assessed as induction of PPRE-reporter gene expression after 24 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Wake Forest University

Curated by ChEMBL
LigandPNGBDBM50295045((9Z,12E)-12-nitrooctadeca-9,12-dienoic acid | CHEM...)
Affinity DataIC50: 410nMAssay Description:Displacement of [3H2]nTZD3 from GST-tagged human recombinant PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Wake Forest University

Curated by ChEMBL
LigandPNGBDBM50295046((E)-10-Nitrohexadec-9-enoic Acid | CHEMBL564368)
Affinity DataIC50: 630nMAssay Description:Displacement of [3H2]nTZD3 from GST-tagged human recombinant PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Wake Forest University

Curated by ChEMBL
LigandPNGBDBM50295047((E)-9-Nitrohexadec-9-enoicAcid | CHEMBL560513)
Affinity DataIC50: 830nMAssay Description:Displacement of [3H2]nTZD3 from GST-tagged human recombinant PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Wake Forest University

Curated by ChEMBL
LigandPNGBDBM50295048((E)-9-nitrooctadec-9-enoic acid | Nitroleic acid |...)
Affinity DataIC50: 980nMAssay Description:Displacement of [3H2]nTZD3 from GST-tagged human recombinant PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
LigandPNGBDBM50295048((E)-9-nitrooctadec-9-enoic acid | Nitroleic acid |...)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human TRPA1 channel in HEK293 cells assessed as increase in intracellular calcium influx by radiometric Ca2+ imagingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Wake Forest University

Curated by ChEMBL
LigandPNGBDBM50295049((E)-10-nitrooctadec-9-enoic acid | CHEMBL561371)
Affinity DataIC50: 1.61E+3nMAssay Description:Displacement of [3H2]nTZD3 from GST-tagged human recombinant PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Wake Forest University

Curated by ChEMBL
LigandPNGBDBM50295045((9Z,12E)-12-nitrooctadeca-9,12-dienoic acid | CHEM...)
Affinity DataIC50: 9.60E+3nMAssay Description:Displacement of [3H2]nTZD3 from GST-tagged human recombinant PPARalpha by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Wake Forest University

Curated by ChEMBL
LigandPNGBDBM50295048((E)-9-nitrooctadec-9-enoic acid | Nitroleic acid |...)
Affinity DataIC50: 1.50E+4nMAssay Description:Displacement of [3H2]nTZD3 from GST-tagged human recombinant PPARalpha by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Wake Forest University

Curated by ChEMBL
LigandPNGBDBM50295046((E)-10-Nitrohexadec-9-enoic Acid | CHEMBL564368)
Affinity DataIC50: 1.50E+4nMAssay Description:Displacement of [3H2]nTZD3 from GST-tagged human recombinant PPARalpha by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Wake Forest University

Curated by ChEMBL
LigandPNGBDBM50295049((E)-10-nitrooctadec-9-enoic acid | CHEMBL561371)
Affinity DataIC50: 1.50E+4nMAssay Description:Displacement of [3H2]nTZD3 from GST-tagged human recombinant PPARalpha by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Wake Forest University

Curated by ChEMBL
LigandPNGBDBM50295047((E)-9-Nitrohexadec-9-enoicAcid | CHEMBL560513)
Affinity DataIC50: 1.50E+4nMAssay Description:Displacement of [3H2]nTZD3 from GST-tagged human recombinant PPARalpha by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetFructose-1,6-bisphosphatase 1(Human)
International Cooperation Base of Pesticide and Green Synthesis (Hubei)

Curated by ChEMBL
LigandPNGBDBM50295048((E)-9-nitrooctadec-9-enoic acid | Nitroleic acid |...)
Affinity DataIC50: 5.80E+4nMAssay Description:Inhibition of human FBPase expressed in Escherichia coli BL21 (DE3) using FBP as substrate incubated for 5 mins by malachite green dye based spectrop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed