Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 13 hits for monomerid = 50327038,50377442,50377443,50377444,50377445,50327038,50377442,50377443,50377444,50377445   

TargetProtein O-GlcNAcase(Human)
Daegu University

Curated by ChEMBL
LigandPNGBDBM50327038((3aR,5R,6S,7R,7aR)-5-(hydroxymethyl)-2-methyl-5,6,...)
Affinity DataKi:  10nMAssay Description:Inhibition of human O-GlcNAcase after 5 mins by Lineweaver-Burke plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetProtein O-GlcNAcase(Human)
Daegu University

Curated by ChEMBL
LigandPNGBDBM50327038((3aR,5R,6S,7R,7aR)-5-(hydroxymethyl)-2-methyl-5,6,...)
Affinity DataKi:  70nMAssay Description:Inhibition of human OGAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetProtein O-GlcNAcase(Human)
Daegu University

Curated by ChEMBL
LigandPNGBDBM50327038((3aR,5R,6S,7R,7aR)-5-(hydroxymethyl)-2-methyl-5,6,...)
Affinity DataKi:  180nMAssay Description:Inhibition of recombinant human OGA expressed in Escherichia coli BL21 (DE3) using varying levels of pNP-beta-GlcNAc as substrate by Lineweaver-burk ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetBeta-hexosaminidase subunit beta(Human)
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50327038((3aR,5R,6S,7R,7aR)-5-(hydroxymethyl)-2-methyl-5,6,...)
Affinity DataKi:  190nMAssay Description:Inhibition of human HexBMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetBeta-hexosaminidase subunit alpha(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50327038((3aR,5R,6S,7R,7aR)-5-(hydroxymethyl)-2-methyl-5,6,...)
Affinity DataKi:  270nMAssay Description:Competitive inhibition of human beta-N-acetyl-D-hexosaminidase-A using 4-Methylumbelliferyl N-acetyl-beta-D-glucosaminide as substrate assessed as re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetBeta-hexosaminidase subunit beta(Human)
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50327038((3aR,5R,6S,7R,7aR)-5-(hydroxymethyl)-2-methyl-5,6,...)
Affinity DataKi:  290nMAssay Description:Competitive inhibition of human beta-N-acetyl-D-hexosaminidase-B using 4-Methylumbelliferyl N-acetyl-beta-D-glucosaminide as substrate assessed as re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetBeta-N-acetylhexosaminidase(Streptomyces plicatus)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50327038((3aR,5R,6S,7R,7aR)-5-(hydroxymethyl)-2-methyl-5,6,...)
Affinity DataKi:  2.00E+4nMAssay Description:Inhibition of Streptomyces plicatus N-acetyl-hexosaminidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetBeta-N-acetylhexosaminidase(Streptomyces plicatus)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50377445(CHEMBL403756)
Affinity DataKi:  1.00E+5nMAssay Description:Inhibition of Streptomyces plicatus N-acetyl-hexosaminidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetBeta-N-acetylhexosaminidase(Streptomyces plicatus)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50377444(CHEMBL404356)
Affinity DataKi:  2.00E+5nMAssay Description:Inhibition of Streptomyces plicatus N-acetyl-hexosaminidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetBeta-hexosaminidase subunit beta(Human)
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50327038((3aR,5R,6S,7R,7aR)-5-(hydroxymethyl)-2-methyl-5,6,...)
Affinity DataKi:  2.70E+5nMAssay Description:Inhibition of human beta hexosaminidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetBeta-hexosaminidase subunit beta(Human)
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50377445(CHEMBL403756)
Affinity DataKi:  8.20E+5nMAssay Description:Inhibition of human beta hexosaminidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetBeta-N-acetylhexosaminidase(Streptomyces plicatus)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50377442(CHEMBL255693)
Affinity DataKi: >2.00E+6nMAssay Description:Inhibition of Streptomyces plicatus N-acetyl-hexosaminidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetBeta-N-acetylhexosaminidase(Streptomyces plicatus)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50377443(CHEMBL403748)
Affinity DataKi: >2.00E+6nMAssay Description:Inhibition of Streptomyces plicatus N-acetyl-hexosaminidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed