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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
5
hits in this display
Target
Mast/stem cell growth factor receptor Kit
(Human)
Vertex Pharmaceuticals
Curated by
ChEMBL
Ligand
BDBM50355465
(CHEMBL1835741)
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Affinity Data
Ki: 12nM
Assay Description:
Displacement of [33P]ATP from human recombinant c-KIT domain after 20 mins by scintillation counting
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
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Target
Receptor-type tyrosine-protein kinase FLT3
(Human)
Vertex Pharmaceuticals
Curated by
ChEMBL
Ligand
BDBM50355465
(CHEMBL1835741)
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Affinity Data
Ki: 15nM
Assay Description:
Displacement of [33P]ATP from human recombinant FLT3 domain after 20 mins by scintillation counting
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
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Target
Interleukin-1 receptor-associated kinase 4
(Human)
Vertex Pharmaceuticals
Curated by
ChEMBL
Ligand
BDBM50355465
(CHEMBL1835741)
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Affinity Data
Ki: 420nM
Assay Description:
Inhibition of IRAK4 by spectrophotometry
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
UniProtKB/TrEMBL
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
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Target
Tyrosine-protein kinase JAK2
(Human)
Vertex Pharmaceuticals
Curated by
ChEMBL
Ligand
BDBM50355465
(CHEMBL1835741)
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Affinity Data
Ki: >4.00E+3nM
Assay Description:
Inhibition of JAK2 by spectrophotometry
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Aurora kinase A
(Human)
Vertex Pharmaceuticals
Curated by
ChEMBL
Ligand
BDBM50355465
(CHEMBL1835741)
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Copy InChI
Affinity Data
Ki: >7.00E+3nM
Assay Description:
Inhibition of Aurora A by spectrophotometry
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI