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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetCoagulation factor VII(Homo sapiens (Human))
Technical University Of Denmark

Curated by ChEMBL
LigandPNGBDBM50347170(CHEMBL1797524)
Affinity DataKi:  4.30E+4nMAssay Description:Inhibition of recombinant F7a using S-2288 as substrate after 15 mins by linear fitting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII(Homo sapiens (Human))
Technical University Of Denmark

Curated by ChEMBL
LigandPNGBDBM50347170(CHEMBL1797524)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of recombinant F7a using S-2288 as substrate after 15 mins by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Technical University Of Denmark

Curated by ChEMBL
LigandPNGBDBM50347170(CHEMBL1797524)
Affinity DataIC50: >5.90E+5nMAssay Description:Inhibition of thrombin using S-2288 as substrate after 15 mins by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Technical University Of Denmark

Curated by ChEMBL
LigandPNGBDBM50347170(CHEMBL1797524)
Affinity DataIC50: >5.90E+5nMAssay Description:Inhibition of F10a using S-2288 as substrate after 15 mins by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed