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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 9 hits in this display   

TargetCoagulation factor VII(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50228753((S)-N*1*-[(S)-4-Guanidino-1-(thiazole-2-carbonyl)-...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human factor 7aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50228753((S)-N*1*-[(S)-4-Guanidino-1-(thiazole-2-carbonyl)-...)
Affinity DataIC50:  1.03E+3nMAssay Description:Inhibitory activity against tissue coagulation factor VII.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50228753((S)-N*1*-[(S)-4-Guanidino-1-(thiazole-2-carbonyl)-...)
Affinity DataIC50:  1.03E+3nMAssay Description:Inhibition of tissue coagulation factor VIIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50228753((S)-N*1*-[(S)-4-Guanidino-1-(thiazole-2-carbonyl)-...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibitory activity against coagulation factor X.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50228753((S)-N*1*-[(S)-4-Guanidino-1-(thiazole-2-carbonyl)-...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50228753((S)-N*1*-[(S)-4-Guanidino-1-(thiazole-2-carbonyl)-...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50228753((S)-N*1*-[(S)-4-Guanidino-1-(thiazole-2-carbonyl)-...)
Affinity DataIC50:  6.00E+4nMAssay Description:Inhibitory activity against thrombin (IIa).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50228753((S)-N*1*-[(S)-4-Guanidino-1-(thiazole-2-carbonyl)-...)
Affinity DataIC50:  6.00E+4nMAssay Description:Inhibition of human alpha-thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50228753((S)-N*1*-[(S)-4-Guanidino-1-(thiazole-2-carbonyl)-...)
Affinity DataIC50:  6.00E+4nMAssay Description:Inhibitory activity against thrombin (IIa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed