Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Troms£

Curated by ChEMBL

LigandBDBM50398993(CHEMBL2180085)Copy SMILESCopy InChI

Affinity DataEC50:  661nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Troms£

Curated by ChEMBL

LigandBDBM50398993(CHEMBL2180085)Copy SMILESCopy InChI

Affinity DataEC50:  660nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI