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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 9 hits in this display   

TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50525098(CHEMBL1160694)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]-CGP-12177 from human beta2-adrenergic receptor expressed in CHO cells after 60 mins by radioligand competition binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50525098(CHEMBL1160694)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]-CGP-12177 from murine beta1-adrenergic receptor expressed in HEK293T cells after 60 mins by radioligand competition binding assa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50525098(CHEMBL1160694)
Affinity DataEC50:  316nMAssay Description:Agonist activity at beta1-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50525098(CHEMBL1160694)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at beta1-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50525098(CHEMBL1160694)
Affinity DataEC50:  794nMAssay Description:Agonist activity at beta2-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring Rluc2-117-GalphaS/GFP10-Ggamma/Gbeta1 assessed as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50525098(CHEMBL1160694)
Affinity DataEC50:  631nMAssay Description:Agonist activity at beta1-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring Rluc2-117-GalphaS/GFP10-Ggamma/Gbeta1 assessed as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50525098(CHEMBL1160694)
Affinity DataEC50:  251nMAssay Description:Agonist activity at beta2-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50525098(CHEMBL1160694)
Affinity DataEC50:  316nMAssay Description:Agonist activity at beta2-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)

Curated by ChEMBL
LigandPNGBDBM50525098(CHEMBL1160694)
Affinity DataEC50:  631nMAssay Description:Agonist activity at beta1-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed