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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetHistone deacetylase 2(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research (Niper) - Ahmedabad

Curated by ChEMBL
LigandPNGBDBM50591647(CHEMBL5191354)
Affinity DataIC50:  750nMAssay Description:Inhibition of recombinant human HDAC2 expressed in baculovirus infected Hi-5 insect cells using Ac-Lys-Tyr-Lys (epsilon-acetyl)-AMC as substrate incu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research (Niper) - Ahmedabad

Curated by ChEMBL
LigandPNGBDBM50591647(CHEMBL5191354)
Affinity DataIC50:  5.30E+3nMAssay Description:Inhibition of recombinant human HDAC3 expressed in baculovirus infected Hi-5 insect cells using Ac-Lys-Tyr-Lys (epsilon-acetyl)-AMC as substrate incu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research (Niper) - Ahmedabad

Curated by ChEMBL
LigandPNGBDBM50591647(CHEMBL5191354)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of recombinant human HDAC1 expressed in baculovirus infected Hi-5 insect cells using Ac-Lys-Tyr-Lys (epsilon-acetyl)-AMC as substrate incu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed