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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50330179(CHEMBL4169168)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP level after 30 mins by LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Mus musculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50330179(CHEMBL4169168)
Affinity DataEC50:  113nMAssay Description:Agonist activity at mouse GPR119 assessed as increase in cAMP levelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed