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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Prolyl endopeptidase
(Sus scrofa)
University Of Antwerp
Curated by
ChEMBL
Ligand
BDBM50399743
(CHEMBL2178978)
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Affinity Data
IC50: 142nM
Assay Description:
Inhibition of pig PREP expressed in Escherichia coli using Z-Gly-Pro-p-nitroanilide substrate
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
DrugBank
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Prolyl endopeptidase FAP
(Mus musculus (Mouse))
University Of Antwerp
Curated by
ChEMBL
Ligand
BDBM50399743
(CHEMBL2178978)
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Affinity Data
IC50: >1.00E+5nM
Assay Description:
Inhibition of mouse recombinant FAP expressed in HEK293 cells assessed as pNA release from Ala-Pro-p-nitroanilide pre-incubated with enzyme for 15 mi...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Dipeptidyl peptidase 4
(Homo sapiens (Human))
University Of Antwerp
Curated by
ChEMBL
Ligand
BDBM50399743
(CHEMBL2178978)
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Affinity Data
IC50: >1.00E+5nM
Assay Description:
Inhibition of human seminal plasma DPP4 assessed as pNA release from Gly-Pro-p-nitroanilide substrate pre-incubated with enzyme for 15 min prior to s...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Dipeptidyl peptidase 2
(Homo sapiens (Human))
University Of Antwerp
Curated by
ChEMBL
Ligand
BDBM50399743
(CHEMBL2178978)
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Copy InChI
Affinity Data
IC50: >1.00E+5nM
Assay Description:
Inhibition of human seminal plasma DPP2 assessed as pNA release from Lys-Ala-p-nitroanilide substrate pre-incubated with enzyme for 15 min prior to s...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI