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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 26 hits in this display   

TargetArginase-2, mitochondrial(Homo sapiens (Human))
Drexel University

Curated by ChEMBL
LigandPNGBDBM50350311(CHEMBL1812661)
Affinity DataKi:  8.5nMAssay Description:Binding affinity to human arginase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArginase-2, mitochondrial(Homo sapiens (Human))
Drexel University

Curated by ChEMBL
LigandPNGBDBM50350311(CHEMBL1812661)
Affinity DataKi:  8.5nMAssay Description:Inhibition of human Arg2 at pH 7.5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArginase(Plasmodium falciparum)
Drexel University

Curated by ChEMBL
LigandPNGBDBM50350311(CHEMBL1812661)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibition of Plasmodium falciparum arginase using L-arginine as substrate by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50350311(CHEMBL1812661)
Affinity DataIC50:  5nMMore data for this Ligand-Target Pair
In DepthDetails
TargetArginase-2, mitochondrial(Homo sapiens (Human))
Drexel University

Curated by ChEMBL
LigandPNGBDBM50350311(CHEMBL1812661)
Affinity DataIC50:  8.5nMMore data for this Ligand-Target Pair
In DepthDetails
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50350311(CHEMBL1812661)
Affinity DataIC50:  311nMAssay Description:Inhibition of human recombinant ARG1 expressed in Escherichia coli using thioarginine as a substrate preincubated for 30 mins followed by substrate a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50350311(CHEMBL1812661)
Affinity DataIC50:  311nMAssay Description:Inhibition of human arginase1 in presence of DNTB by thio ornithine generation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50350311(CHEMBL1812661)
Affinity DataIC50:  800nMAssay Description:Inhibition of human Arg1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArginase-1(Rattus norvegicus)TBA
LigandPNGBDBM50350311(CHEMBL1812661)
Affinity DataIC50:  800nMMore data for this Ligand-Target Pair
In DepthDetails
TargetArginase-1(Rattus norvegicus)TBA
LigandPNGBDBM50350311(CHEMBL1812661)
Affinity DataIC50:  800nMAssay Description:Inhibition of rat Arg1 at pH 7.4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArginase-1(Rattus norvegicus)TBA
LigandPNGBDBM50350311(CHEMBL1812661)
Affinity DataIC50:  800nMMore data for this Ligand-Target Pair
In DepthDetails
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50350311(CHEMBL1812661)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of recombinant human arginase 1 using L-arginine as substrate measured after 60 mins in presence of manganese chloride by o-phthaldialdehy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50350311(CHEMBL1812661)
Affinity DataIC50:  1.45E+3nMAssay Description:Inhibition of human recombinant full length Arg1 using L-arginine as substrate assessed as urea level after 1 hr by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50350311(CHEMBL1812661)
Affinity DataIC50:  1.45E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50350311(CHEMBL1812661)
Affinity DataIC50:  1.47E+3nMAssay Description:Inhibition of human arginase-1 assessed as L-arginine conversion to L-ornithine measured as urea level after 1 hr by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50350311(CHEMBL1812661)
Affinity DataIC50:  1.55E+3nMAssay Description:Inhibition of human recombinant arginase 1 expressed in Escherichia coli BL21 (DE3) assessed as reduction in urea production using L-arginine as subs...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArginase-2, mitochondrial(Homo sapiens (Human))
Drexel University

Curated by ChEMBL
LigandPNGBDBM50350311(CHEMBL1812661)
Affinity DataIC50:  1.92E+3nMAssay Description:Inhibition of human Arg2 by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArginase-2, mitochondrial(Homo sapiens (Human))
Drexel University

Curated by ChEMBL
LigandPNGBDBM50350311(CHEMBL1812661)
Affinity DataIC50:  2.15E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetArginase-2, mitochondrial(Homo sapiens (Human))
Drexel University

Curated by ChEMBL
LigandPNGBDBM50350311(CHEMBL1812661)
Affinity DataIC50:  2.15E+3nMAssay Description:Inhibition of human arginase-2 assessed as L-arginine conversion to L-ornithine measured as urea level after 1 hr by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50350311(CHEMBL1812661)
Affinity DataIC50:  1.68E+4nMAssay Description:Inhibition of recombinant human ARG1 expressed in CHO-K1 cells assessed as reduction in urea level incubated for 24 hrs by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50350311(CHEMBL1812661)
Affinity DataKd:  18nMAssay Description:Binding affinity to human arginase 1 using L-arginine as substrate by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArginase(Plasmodium falciparum)
Drexel University

Curated by ChEMBL
LigandPNGBDBM50350311(CHEMBL1812661)
Affinity DataKd:  1.10E+4nMAssay Description:Binding affinity to Plasmodium falciparum arginaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50350311(CHEMBL1812661)
Affinity DataKd:  5nMAssay Description:Binding affinity to human arginase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50350311(CHEMBL1812661)
In DepthDetails
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50350311(CHEMBL1812661)
In DepthDetails
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50350311(CHEMBL1812661)
Affinity DataKd:  5nMAssay Description:Binding affinity to human Arg1 at pH 8.5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed