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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
21
hits in this display
Target
Carbonic anhydrase 7
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM50027536
((phosphonoformate)Trisodium phosphonoformate | Ant...)
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Affinity Data
Ki: 5.60E+5nM
Assay Description:
Inhibition of human recombinant CA7 by CO2 hydration assay
More data for this Ligand-Target Pair
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Target
Carbonic anhydrase 4
(Homo sapiens (Human))
Università
Curated by
ChEMBL
Ligand
BDBM50027536
((phosphonoformate)Trisodium phosphonoformate | Ant...)
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Affinity Data
Ki: 8.20E+5nM
Assay Description:
Inhibition constant of anion against human carbonic anhydrase isozyme hCA IV
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Target
Carbonic anhydrase 4
(Homo sapiens (Human))
Università
Curated by
ChEMBL
Ligand
BDBM50027536
((phosphonoformate)Trisodium phosphonoformate | Ant...)
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Affinity Data
Ki: 8.20E+5nM
Assay Description:
Inhibition of human recombinant CA4 by CO2 hydration assay
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Target
Carbonic anhydrase 13
(Mus musculus (mouse))
Universit£
Curated by
ChEMBL
Ligand
BDBM50027536
((phosphonoformate)Trisodium phosphonoformate | Ant...)
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Affinity Data
Ki: 8.70E+5nM
Assay Description:
Inhibition of mouse recombinant CA13 by CO2 hydration assay
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Target
Carbonic anhydrase 12
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM50027536
((phosphonoformate)Trisodium phosphonoformate | Ant...)
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Affinity Data
Ki: 1.29E+6nM
Assay Description:
Inhibition of human recombinant CA12 by CO2 hydration assay
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Target
Carbonic anhydrase 6
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM50027536
((phosphonoformate)Trisodium phosphonoformate | Ant...)
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Affinity Data
Ki: 1.81E+6nM
Assay Description:
Inhibition of human recombinant CA6 by CO2 hydration assay
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Target
Carbonic anhydrase 9
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM50027536
((phosphonoformate)Trisodium phosphonoformate | Ant...)
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Affinity Data
Ki: 2.21E+6nM
Assay Description:
Inhibition of human recombinant CA9 by CO2 hydration assay
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Target
Carbonic anhydrase 9
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM50027536
((phosphonoformate)Trisodium phosphonoformate | Ant...)
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Affinity Data
Ki: 2.21E+6nM
Assay Description:
Inhibition constant of anion against human carbonic anhydrase isozyme hCA IX
More data for this Ligand-Target Pair
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Target
Carbonic anhydrase 14
(Homo sapiens (Human))
Universit£
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ChEMBL
Ligand
BDBM50027536
((phosphonoformate)Trisodium phosphonoformate | Ant...)
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Affinity Data
Ki: 3.60E+6nM
Assay Description:
Inhibition of human recombinant CA14 by CO2 hydration assay
More data for this Ligand-Target Pair
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Target
Carbonic anhydrase 5B, mitochondrial
(Homo sapiens (Human))
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Curated by
ChEMBL
Ligand
BDBM50027536
((phosphonoformate)Trisodium phosphonoformate | Ant...)
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Affinity Data
Ki: 1.18E+7nM
Assay Description:
Inhibition of human recombinant CA5B by CO2 hydration assay
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Target
Carbonic anhydrase 2
(Homo sapiens (Human))
Università
Curated by
ChEMBL
Ligand
BDBM50027536
((phosphonoformate)Trisodium phosphonoformate | Ant...)
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Affinity Data
Ki: 1.42E+7nM
Assay Description:
Inhibition constant of anion against human carbonic anhydrase isozyme hCA II
More data for this Ligand-Target Pair
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Target
Carbonic anhydrase 2
(Homo sapiens (Human))
Università
Curated by
ChEMBL
Ligand
BDBM50027536
((phosphonoformate)Trisodium phosphonoformate | Ant...)
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Affinity Data
Ki: 1.42E+7nM
Assay Description:
Inhibition of human recombinant CA2 by CO2 hydration assay
More data for this Ligand-Target Pair
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Target
Carbonic anhydrase 1
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM50027536
((phosphonoformate)Trisodium phosphonoformate | Ant...)
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Affinity Data
Ki: 2.41E+7nM
Assay Description:
Inhibition of cloned human CA1 by CO2 hydration assay
More data for this Ligand-Target Pair
Target Info
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Target
Carbonic anhydrase 5A, mitochondrial
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM50027536
((phosphonoformate)Trisodium phosphonoformate | Ant...)
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Affinity Data
Ki: 4.17E+7nM
Assay Description:
Inhibition of human recombinant CA5A by CO2 hydration assay
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Target
Reverse transcriptase/RNaseH
(Human immunodeficiency virus 1)
Life Science Research Center
Curated by
ChEMBL
Ligand
BDBM50027536
((phosphonoformate)Trisodium phosphonoformate | Ant...)
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Affinity Data
IC50: 2.03E+3nM
Assay Description:
Inhibitory activity against HIV-1 reverse transcriptase
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Target
Reverse transcriptase/RNaseH
(Human immunodeficiency virus 1)
Life Science Research Center
Curated by
ChEMBL
Ligand
BDBM50027536
((phosphonoformate)Trisodium phosphonoformate | Ant...)
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Affinity Data
IC50: 1.76E+4nM
Assay Description:
Inhibitory effect of the compound on Molony Murine Leukemia virus (mo-MuLv) Recombiannt Reverse transcriptase
More data for this Ligand-Target Pair
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Target
DNA polymerase catalytic subunit
(Human herpesvirus 1 (strain 17) (HHV-1) (Human her...)
TBA
Curated by
ChEMBL
Ligand
BDBM50027536
((phosphonoformate)Trisodium phosphonoformate | Ant...)
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Affinity Data
IC50: 7.40E+4nM
Assay Description:
Inhibition of HSV-1 DNA polymerase in HSV-1 C42 plaque reduction assay
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Target
ATP-binding cassette sub-family C member 2
(Homo sapiens (Human))
Amgen
Curated by
ChEMBL
Ligand
BDBM50027536
((phosphonoformate)Trisodium phosphonoformate | Ant...)
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Affinity Data
IC50: >1.33E+5nM
Assay Description:
Inhibition of human MRP2 overexpressed in Sf9 cell membrane vesicles assessed as uptake of [3H]-estradiol-17beta-D-glucuronide in presence of ATP and...
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Target
ATP-binding cassette sub-family C member 3
(Homo sapiens (Human))
Amgen
Curated by
ChEMBL
Ligand
BDBM50027536
((phosphonoformate)Trisodium phosphonoformate | Ant...)
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Affinity Data
IC50: >1.33E+5nM
Assay Description:
Inhibition of human MRP3 overexpressed in Sf9 insect cell membrane vesicles assessed as uptake of [3H]-estradiol-17beta-D-glucuronide in presence of ...
More data for this Ligand-Target Pair
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Target
ATP-binding cassette sub-family C member 4
(Homo sapiens (Human))
Amgen
Curated by
ChEMBL
Ligand
BDBM50027536
((phosphonoformate)Trisodium phosphonoformate | Ant...)
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Affinity Data
IC50: >1.33E+5nM
Assay Description:
Inhibition of human MRP4 overexpressed in Sf9 cell membrane vesicles assessed as uptake of [3H]-estradiol-17beta-D-glucuronide in presence of ATP and...
More data for this Ligand-Target Pair
Target Info
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Target
Bile salt export pump
(Homo sapiens (Human))
Amgen
Curated by
ChEMBL
Ligand
BDBM50027536
((phosphonoformate)Trisodium phosphonoformate | Ant...)
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Affinity Data
IC50: >1.33E+5nM
Assay Description:
Inhibition of human BSEP overexpressed in Sf9 cell membrane vesicles assessed as uptake of [3H]-taurocholate in presence of ATP measured after 15 to ...
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