Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 12 hits in this display
BDBM50434169(CHEMBL2385300 | US9346814, Cmpd No 22 Example 26)
BDBM50434169(CHEMBL2385300 | US9346814, Cmpd No 22 Example 26)
BDBM50434169(CHEMBL2385300 | US9346814, Cmpd No 22 Example 26)
IC50: 11nMAssay Description:Inhibition of recombinant mouse FAP purified from HEK293 cell supernatant using Ala-Pro-p-nitroanilide as substrate by spectrophotometryMore data for this Ligand-Target Pair
BDBM50434169(CHEMBL2385300 | US9346814, Cmpd No 22 Example 26)
IC50: 11nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
BDBM50434169(CHEMBL2385300 | US9346814, Cmpd No 22 Example 26)
BDBM50434169(CHEMBL2385300 | US9346814, Cmpd No 22 Example 26)
IC50: >5.00E+4nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
BDBM50434169(CHEMBL2385300 | US9346814, Cmpd No 22 Example 26)
IC50: >5.00E+4nMAssay Description:Inhibition of recombinant human PREP purified from Escherichia coli using Z-Gly-Pro-p-nitroanilide as substrate by spectrophotometryMore data for this Ligand-Target Pair
BDBM50434169(CHEMBL2385300 | US9346814, Cmpd No 22 Example 26)
IC50: >1.00E+5nMAssay Description:Inhibition of DPP4 purified from human seminal plasma using Gly-Pro-p-nitroanilide as substrate by spectrophotometryMore data for this Ligand-Target Pair
BDBM50434169(CHEMBL2385300 | US9346814, Cmpd No 22 Example 26)
IC50: >1.00E+5nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
BDBM50434169(CHEMBL2385300 | US9346814, Cmpd No 22 Example 26)
IC50: >1.00E+5nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
BDBM50434169(CHEMBL2385300 | US9346814, Cmpd No 22 Example 26)
IC50: >1.00E+5nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
BDBM50434169(CHEMBL2385300 | US9346814, Cmpd No 22 Example 26)
IC50: >1.00E+5nMAssay Description:Inhibition of DPP2 purified from human seminal plasma using Lys-Ala-p-nitroanilide as substrate by spectrophotometryMore data for this Ligand-Target Pair