Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 4 hits in this display
DNA ligase A(Mycobacterium tuberculosis)India Central Drug Research Institute
BDBM22986(18-[6-(piperidin-1-yl)hexyl]-8-thia-18-azatetracyc...)
DNA ligase A(Mycobacterium tuberculosis)India Central Drug Research Institute
BDBM22986(18-[6-(piperidin-1-yl)hexyl]-8-thia-18-azatetracyc...)
IC50: 1.35E+4nMAssay Description:All assays have been carried out using procedures previously described by our group (Srivastava et al., 2005a; 2005b; 2007)More data for this Ligand-Target Pair
DNA ligase(Bacteriophage T4)India Central Drug Research Institute
BDBM22986(18-[6-(piperidin-1-yl)hexyl]-8-thia-18-azatetracyc...)
IC50: 2.04E+5nMpH: 7.6 T: 2°CAssay Description:The assay was performed using a 40-bp double-stranded DNA substrate carrying a single-strand nick between bases 22 and 23. The reaction products were...More data for this Ligand-Target Pair
DNA ligase 1(Homo sapiens (Human))India Central Drug Research Institute
BDBM22986(18-[6-(piperidin-1-yl)hexyl]-8-thia-18-azatetracyc...)
IC50: 2.12E+5nMpH: 8.0 T: 2°CAssay Description:The assay was performed using a 40-bp double-stranded DNA substrate carrying a single-strand nick between bases 22 and 23. The reaction products were...More data for this Ligand-Target Pair