Home
About
Info
Download
WebServices
Contact
Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Histamine H4 receptor
(Homo sapiens (Human))
Bioprojet-Biotech
Curated by
ChEMBL
Ligand
BDBM50259264
(CHEMBL4100315)
Copy SMILES
Copy InChI
Affinity Data
Ki: 27nM
Assay Description:
Antagonist activity at H4 receptor in human SH-SY5Y cells assessed as inhibition of imetit-induced GTPgamma[35S] binding after 30 mins by microbeta s...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Histamine H4 receptor
(Homo sapiens (Human))
Bioprojet-Biotech
Curated by
ChEMBL
Ligand
BDBM50259264
(CHEMBL4100315)
Copy SMILES
Copy InChI
Affinity Data
Ki: 27nM
Assay Description:
Antagonist activity at human H4 receptor expressed in CHO cells co-expressing Galphai2 assessed as inhibition of imetit-induced GTPgamma[35S] binding...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Histamine H3 receptor
(Homo sapiens (Human))
Bioprojet-Biotech
Curated by
ChEMBL
Ligand
BDBM50259264
(CHEMBL4100315)
Copy SMILES
Copy InChI
Affinity Data
Ki: 118nM
Assay Description:
Antagonist activity at H3 receptor (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI