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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 7 hits in this display   

TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50488611(CHEMBL2298806)
Affinity DataKi:  1.70nMAssay Description:Binding affinity to dopamine D2 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))TBA
LigandPNGBDBM50488611(CHEMBL2298806)
Affinity DataKi:  15nMAssay Description:Binding affinity to 5-HT2A receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))TBA
LigandPNGBDBM50488611(CHEMBL2298806)
Affinity DataKi:  65nMAssay Description:Binding affinity to 5-HT2C receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))TBA
LigandPNGBDBM50488611(CHEMBL2298806)
Affinity DataKi:  126nMAssay Description:Binding affinity to 5-HT1A receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetD(1A) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50488611(CHEMBL2298806)
Affinity DataKi:  3.98E+3nMAssay Description:Binding affinity to dopamine D1 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))TBA
LigandPNGBDBM50488611(CHEMBL2298806)
Affinity DataKi:  5.25E+3nMAssay Description:Binding affinity to 5-HT3 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetSodium-dependent serotonin transporter(Homo sapiens (Human))TBA
LigandPNGBDBM50488611(CHEMBL2298806)
Affinity DataIC50:  1.76E+3nMAssay Description:Inhibition of 5-HT uptake at SERT (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article