Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50278526(4-((naphthalen-2-yloxy)methyl)piperidine | CHEMBL4...)
Affinity DataKi:  311nMAssay Description:Displacement of [3H]granisetron from human 5HT3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50278526(4-((naphthalen-2-yloxy)methyl)piperidine | CHEMBL4...)
Affinity DataKi:  3.80E+3nMAssay Description:Displacement of [3H]dofetilide from human ERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50278526(4-((naphthalen-2-yloxy)methyl)piperidine | CHEMBL4...)
Affinity DataIC50:  8nMAssay Description:Inhibition of radiolabeled serotonin reuptake at human SERT expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50278526(4-((naphthalen-2-yloxy)methyl)piperidine | CHEMBL4...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of radiolabeled noradrenaline reuptake at human NET expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50278526(4-((naphthalen-2-yloxy)methyl)piperidine | CHEMBL4...)
Affinity DataIC50: >7.00E+3nMAssay Description:Inhibition of radiolabeled dopamine reuptake at human DAT expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed