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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

Target5-hydroxytryptamine receptor 3A/3B(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50459885(CHEMBL1382868)
Affinity DataIC50:  430nMAssay Description:Inhibition of human 5-HT3AB receptor expressed in transient A201 cells after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50459885(CHEMBL1382868)
Affinity DataIC50:  620nMAssay Description:Inhibition of human 5-HT3A receptor expressed in transient A201 cells after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3E(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50459885(CHEMBL1382868)
Affinity DataIC50:  710nMAssay Description:Inhibition of human 5-HT3AE receptor expressed in transient A201 cells after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3C(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50459885(CHEMBL1382868)
Affinity DataIC50:  840nMAssay Description:Inhibition of human 5-HT3AC receptor expressed in transient A201 cells after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed