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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
10
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Target
5-hydroxytryptamine receptor 3A
(Homo sapiens (Human))
The University Of Louisiana At Monroe
Curated by
ChEMBL
Ligand
BDBM50103072
(1-Benzyl-2-piperazin-1-yl-1H-benzoimidazole | CHEM...)
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Affinity Data
Ki: 0.360nM
Assay Description:
Binding affinity of the compound against human 5-hydroxytryptamine 3A receptor
More data for this Ligand-Target Pair
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Target
5-hydroxytryptamine receptor 3A/3B
(Rattus norvegicus)
Universidad De Alcal£
Curated by
ChEMBL
Ligand
BDBM50103072
(1-Benzyl-2-piperazin-1-yl-1H-benzoimidazole | CHEM...)
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Affinity Data
Ki: 0.620nM
Assay Description:
Binding affinity towards rat 5-hydroxytryptamine 3 receptor was evaluated
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Target
5-hydroxytryptamine receptor 3A/3B
(Rattus norvegicus)
Universidad De Alcal£
Curated by
ChEMBL
Ligand
BDBM50103072
(1-Benzyl-2-piperazin-1-yl-1H-benzoimidazole | CHEM...)
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Affinity Data
Ki: 0.631nM
Assay Description:
In vitro by displacement of [3H]LY-278584 from 5-hydroxytryptamine 3 receptor on rat entorhinal cortex
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Target
5-hydroxytryptamine receptor 3A/3B
(Rattus norvegicus)
Universidad De Alcal£
Curated by
ChEMBL
Ligand
BDBM50103072
(1-Benzyl-2-piperazin-1-yl-1H-benzoimidazole | CHEM...)
Copy SMILES
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Affinity Data
Ki: 0.631nM
Assay Description:
Rat 5-hydroxytryptamine 3 receptor (5-HT3) antagonist
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Target
D(2) dopamine receptor
(Rattus norvegicus (rat))
Faes
Curated by
ChEMBL
Ligand
BDBM50103072
(1-Benzyl-2-piperazin-1-yl-1H-benzoimidazole | CHEM...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
In vitro by displacement of [3H]raclopride from Dopamine receptor D2 on rat striatal membrane
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Target
5-hydroxytryptamine receptor 4
(GUINEA PIG)
Faes
Curated by
ChEMBL
Ligand
BDBM50103072
(1-Benzyl-2-piperazin-1-yl-1H-benzoimidazole | CHEM...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
In vitro by displacement of [3H]GR-113808 from 5-hydroxytryptamine 4 receptor on guinea pig striatal membrane
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Target
5-hydroxytryptamine receptor 1A
(Rattus norvegicus (rat))
Faes
Curated by
ChEMBL
Ligand
BDBM50103072
(1-Benzyl-2-piperazin-1-yl-1H-benzoimidazole | CHEM...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
In vitro by displacement of [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor on rat cortical membrane
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Target
5-hydroxytryptamine receptor 2A
(Rattus norvegicus (rat))
Faes
Curated by
ChEMBL
Ligand
BDBM50103072
(1-Benzyl-2-piperazin-1-yl-1H-benzoimidazole | CHEM...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity was evaluated in vitro by displacement of [3H]ketanserin from 5-hydroxytryptamine 2A receptor on rat cortical membrane
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Target
5-hydroxytryptamine receptor 4
(GUINEA PIG)
Faes
Curated by
ChEMBL
Ligand
BDBM50103072
(1-Benzyl-2-piperazin-1-yl-1H-benzoimidazole | CHEM...)
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Affinity Data
IC50: >1.00E+3nM
Assay Description:
Binding affinity towards 5-hydroxytryptamine 4 receptor in striatum membranes of guinea-pig brain was evaluated
More data for this Ligand-Target Pair
Target Info
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Target
D(2) dopamine receptor
(Rattus norvegicus (rat))
Faes
Curated by
ChEMBL
Ligand
BDBM50103072
(1-Benzyl-2-piperazin-1-yl-1H-benzoimidazole | CHEM...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+3nM
Assay Description:
Binding affinity towards Dopamine receptor D2 in rat was evaluated
More data for this Ligand-Target Pair
Target Info
PDB
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KEGG
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CHEMBL
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