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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Histamine H3 receptor
(Homo sapiens (Human))
Meiji Seika Kaisha
Curated by
ChEMBL
Ligand
BDBM50326297
(3-((1H-imidazol-4-yl)methyl)pyridine | 3-(3H-Imida...)
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Affinity Data
Ki: 76nM
Assay Description:
Displacement of [3H]-(R)-alpha-methylhistamine from human histamine H3 receptor expressed in CHO cells by liquid scintillation counting
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
In Depth
Details
Article
PubMed
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Target
Histamine H4 receptor
(Homo sapiens (Human))
Vu University Amsterdam
Curated by
ChEMBL
Ligand
BDBM50326297
(3-((1H-imidazol-4-yl)methyl)pyridine | 3-(3H-Imida...)
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Copy InChI
Affinity Data
Ki: 100nM
Assay Description:
Displacement of [3H]histamine from human H4R receptor expressed in HEK293 cells at 10 uM after 1.5 hrs by liquid scintillation counting
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Histamine H3 receptor
(Homo sapiens (Human))
Meiji Seika Kaisha
Curated by
ChEMBL
Ligand
BDBM50326297
(3-((1H-imidazol-4-yl)methyl)pyridine | 3-(3H-Imida...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 140nM
Assay Description:
Agonist activity at human histamine H3 receptor expressed in CHO cells assessed as [35S]GTPgammaS binding
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI