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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
5
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Target
Alpha-2B adrenergic receptor
(NEONATAL RAT)
University of Nebraska
Curated by
PDSP K
i
Database
Ligand
BDBM81805
(AZAPETINE | CAS_130-83-6 | NSC_8966)
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Affinity Data
Ki: 5.30nM
More data for this Ligand-Target Pair
Target Info
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KEGG
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Target
Alpha-2C adrenergic receptor
(OK)
University of Nebraska
Curated by
PDSP K
i
Database
Ligand
BDBM81805
(AZAPETINE | CAS_130-83-6 | NSC_8966)
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Affinity Data
Ki: 14nM
More data for this Ligand-Target Pair
Target Info
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Target
Alpha-2A adrenergic receptor
(Homo sapiens (Human))
University of Nebraska
Curated by
PDSP K
i
Database
Ligand
BDBM81805
(AZAPETINE | CAS_130-83-6 | NSC_8966)
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Affinity Data
Ki: 38nM
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
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Target
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Rattus norvegicus (rat))
TBA
Curated by
ChEMBL
Ligand
BDBM81805
(AZAPETINE | CAS_130-83-6 | NSC_8966)
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Affinity Data
IC50: 205nM
Assay Description:
Inhibition of specific [3H]-prazosin binding (0.2 nM) to rat brain membranes alpha-1 adrenergic receptor
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Target
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor
(RAT)
TBA
Curated by
ChEMBL
Ligand
BDBM81805
(AZAPETINE | CAS_130-83-6 | NSC_8966)
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Affinity Data
IC50: 1.30E+3nM
Assay Description:
Inhibition of specific [3H]clonidine binding (0.4 nM) to rat brain membranes alpha-2 adrenergic receptor
More data for this Ligand-Target Pair
Target Info
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GoogleScholar
Ligand Info
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Article
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